EA200000261A2 - Новые замещенные димерные соединения, способ их получения и содержащая их фармацевтическая композиция - Google Patents

Новые замещенные димерные соединения, способ их получения и содержащая их фармацевтическая композиция

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Publication number
EA200000261A2
EA200000261A2 EA200000261A EA200000261A EA200000261A2 EA 200000261 A2 EA200000261 A2 EA 200000261A2 EA 200000261 A EA200000261 A EA 200000261A EA 200000261 A EA200000261 A EA 200000261A EA 200000261 A2 EA200000261 A2 EA 200000261A2
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Prior art keywords
preparation
pharmaceutical compositions
compositions containing
new substituted
dimeric compounds
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EA200000261A
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English (en)
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EA003300B1 (ru
EA200000261A3 (ru
Inventor
Даниель Лезьер
Саид Иус
Кароль Декамп-Франсуа
Франсуа Лефулон
Жераль Гийоме
Мари-Клод Вио
Каролин Беннежан
Филипп Делягранж
Пьер Ренар
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Адир Э Компани
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Publication of EA200000261A2 publication Critical patent/EA200000261A2/ru
Publication of EA200000261A3 publication Critical patent/EA200000261A3/ru
Publication of EA003300B1 publication Critical patent/EA003300B1/ru

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Abstract

Изобретение относится к соединениям формулы (I)A-G-Cy-G-Cy-G-B (I)где A представляет собой группу NRC(Q)R, NRC(Q)NRRили C(Q)NRR,B представляет собой группу NRC(Q)R, C(Q)NRR, NRC(Q)NRR, C(Q)OR, NRC(Q)ORи NRR,Gи Cявляются необязательно замещенной алкиленовой цепью,Cy представляет собой циклическую структуруGпредставляет собой цепьЛекарственные препараты.
EA200000261A 1999-03-25 2000-03-24 Новые замещенные димерные соединения, способ их получения и содержащая их фармацевтическая композиция EA003300B1 (ru)

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FR9903717A FR2791344B1 (fr) 1999-03-25 1999-03-25 Nouveaux derives dimeriques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

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EA200000261A2 true EA200000261A2 (ru) 2000-10-30
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US7078541B2 (en) * 2002-02-07 2006-07-18 Galileo Pharmaceuticals, Inc. Benzofuran derivatives
US6653346B1 (en) * 2002-02-07 2003-11-25 Galileo Pharmaceuticals, Inc. Cytoprotective benzofuran derivatives
BR0316962A (pt) * 2002-12-03 2005-10-25 Hoffmann La Roche Aminoalcoxiindóis como ligantes para o receptor de 5-ht6 para o tratamento de distúrbios do snc
EP2352501B1 (en) * 2008-11-03 2014-01-01 ChemoCentryx, Inc. Compounds for use in the treatment of osteoporosis
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US5273999A (en) * 1991-09-10 1993-12-28 Hoffmann-La Roche Inc. Carboxylic acid leukotriene B4 antagonists
DK78692D0 (da) * 1992-06-12 1992-06-12 Lundbeck & Co As H Dimere piperidin- og piperazinderivater
FR2713636B1 (fr) * 1993-12-07 1996-01-05 Adir Nouveaux dérivés naphtaléniques, leur procédé de préparation, et les compositions pharmaceutiques qui les contiennent.
US5753700A (en) * 1994-12-28 1998-05-19 Ono Pharmaceutical Co., Ltd. Naphthyloxyacetic acid derivatives
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HU0001249D0 (en) 2000-06-28
FR2791344A1 (fr) 2000-09-29
JP3688549B2 (ja) 2005-08-31
ZA200001502B (en) 2000-10-24
EP1038863A2 (fr) 2000-09-27
DK1038863T3 (da) 2003-09-22
CA2301990C (fr) 2004-01-06
PL339184A1 (en) 2000-10-09
AU761605B2 (en) 2003-06-05
HUP0001249A2 (hu) 2000-10-28
CN1273967A (zh) 2000-11-22
US6319930B1 (en) 2001-11-20
PT1038863E (pt) 2003-09-30
CA2301990A1 (fr) 2000-09-25
CN1181050C (zh) 2004-12-22
KR100450314B1 (ko) 2004-09-30
ATE242201T1 (de) 2003-06-15
KR20010006873A (ko) 2001-01-26
EP1038863B1 (fr) 2003-06-04
EP1038863A3 (fr) 2000-11-02
SI1038863T1 (en) 2003-10-31
JP2000319242A (ja) 2000-11-21
BR0001419A (pt) 2000-09-26
US20020035114A1 (en) 2002-03-21
ES2200794T3 (es) 2004-03-16
FR2791344B1 (fr) 2002-02-15
NZ503587A (en) 2001-05-25
US6635650B2 (en) 2003-10-21
EA003300B1 (ru) 2003-04-24
NO20001541D0 (no) 2000-03-24
NO20001541L (no) 2000-09-26
DE60003103T2 (de) 2004-05-19
HUP0001249A3 (en) 2003-05-28
AU2257700A (en) 2000-10-05
EA200000261A3 (ru) 2000-12-25
HK1032042A1 (en) 2001-07-06
DE60003103D1 (de) 2003-07-10

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