SG149879A1 - OPTICALLY ACTIVE QUATERNARY AMMONIUM SALT HAVING AXIAL ASYMMETRY AND PROCESS FOR PRODUCING α - AMINO ACID AND DERIVATIVE THEREOF WITH THE SAME - Google Patents
OPTICALLY ACTIVE QUATERNARY AMMONIUM SALT HAVING AXIAL ASYMMETRY AND PROCESS FOR PRODUCING α - AMINO ACID AND DERIVATIVE THEREOF WITH THE SAMEInfo
- Publication number
- SG149879A1 SG149879A1 SG200900527-3A SG2009005273A SG149879A1 SG 149879 A1 SG149879 A1 SG 149879A1 SG 2009005273 A SG2009005273 A SG 2009005273A SG 149879 A1 SG149879 A1 SG 149879A1
- Authority
- SG
- Singapore
- Prior art keywords
- derivative
- producing
- amino acid
- quaternary ammonium
- ammonium salt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
- B01J31/02—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides
- B01J31/0234—Nitrogen-, phosphorus-, arsenic- or antimony-containing compounds
- B01J31/0235—Nitrogen containing compounds
- B01J31/0237—Amines
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
- B01J31/02—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides
- B01J31/0234—Nitrogen-, phosphorus-, arsenic- or antimony-containing compounds
- B01J31/0235—Nitrogen containing compounds
- B01J31/0239—Quaternary ammonium compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2231/00—Catalytic reactions performed with catalysts classified in B01J31/00
- B01J2231/40—Substitution reactions at carbon centres, e.g. C-C or C-X, i.e. carbon-hetero atom, cross-coupling, C-H activation or ring-opening reactions
- B01J2231/42—Catalytic cross-coupling, i.e. connection of previously not connected C-atoms or C- and X-atoms without rearrangement
- B01J2231/4205—C-C cross-coupling, e.g. metal catalyzed or Friedel-Crafts type
- B01J2231/4272—C-C cross-coupling, e.g. metal catalyzed or Friedel-Crafts type via enolates or aza-analogues, added as such or made in-situ, e.g. ArY + R2C=C(OM)Z -> ArR2C-C(O)Z, in which R is H or alkyl, M is Na, K or SiMe3, Y is the leaving group, Z is Ar or OR' and R' is alkyl
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2531/00—Additional information regarding catalytic systems classified in B01J31/00
- B01J2531/90—Catalytic systems characterized by the solvent or solvent system used
- B01J2531/98—Phase-transfer catalysis in a mixed solvent system containing at least 2 immiscible solvents or solvent phases
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Polarising Elements (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2004023317 | 2004-01-30 | ||
JP2004056659 | 2004-03-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG149879A1 true SG149879A1 (en) | 2009-02-27 |
Family
ID=34829419
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG200900527-3A SG149879A1 (en) | 2004-01-30 | 2005-01-27 | OPTICALLY ACTIVE QUATERNARY AMMONIUM SALT HAVING AXIAL ASYMMETRY AND PROCESS FOR PRODUCING α - AMINO ACID AND DERIVATIVE THEREOF WITH THE SAME |
Country Status (7)
Country | Link |
---|---|
US (3) | US7928224B2 (zh) |
EP (1) | EP1712549B1 (zh) |
JP (2) | JP4605606B2 (zh) |
CN (1) | CN1914177B (zh) |
CA (1) | CA2549431C (zh) |
SG (1) | SG149879A1 (zh) |
WO (1) | WO2005073196A1 (zh) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1712549B1 (en) * | 2004-01-30 | 2018-04-11 | Nagase & Company, Ltd. | Optically active quaternary ammonium salt having axial asymmetry and process for producing alpha-amino acid and derivative thereof with the same |
JP4779109B2 (ja) * | 2004-11-17 | 2011-09-28 | 国立大学法人京都大学 | 軸不斉を有する光学活性アミノ酸誘導体及び該アミノ酸誘導体を不斉触媒として用いる光学活性化合物の製造方法 |
JP5296375B2 (ja) | 2005-03-03 | 2013-09-25 | 日本曹達株式会社 | 2つの軸不斉を有する光学活性アンモニウム塩化合物の製造方法 |
JP5008553B2 (ja) * | 2005-03-29 | 2012-08-22 | 長瀬産業株式会社 | 軸不斉を有する光学活性な4級アンモニウム塩およびそれを用いたα−アミノ酸およびその誘導体の製造方法 |
JP4879896B2 (ja) * | 2005-07-29 | 2012-02-22 | 長瀬産業株式会社 | アルジミンまたはその誘導体を用いる一置換アルキル化化合物の製造方法 |
JP4802191B2 (ja) * | 2005-07-29 | 2011-10-26 | 長瀬産業株式会社 | 軸不斉を有する光学活性な4級アンモニウム塩およびそれを用いたα−アミノ酸およびその誘導体の製造方法 |
JP5344523B2 (ja) * | 2005-12-26 | 2013-11-20 | 長瀬産業株式会社 | 立体選択的にストレッカー反応を進行させ得る触媒、およびそれを用いたα−アミノニトリル誘導体を立体選択的に製造するための方法 |
DE102006009518A1 (de) * | 2006-03-01 | 2007-09-06 | Studiengesellschaft Kohle Mbh | Organische Salze sowie Verfahren zur Herstellung von chiralen organischen Verbindungen |
JP5108777B2 (ja) | 2006-09-28 | 2012-12-26 | 長瀬産業株式会社 | 軸不斉を有する光学活性な4級アンモニウム塩およびそれを用いたα−アミノ酸およびその誘導体の製造方法 |
JP5112670B2 (ja) * | 2006-10-03 | 2013-01-09 | 日本曹達株式会社 | 置換アミノ酸シッフ塩基化合物の製造方法 |
US8507669B2 (en) | 2008-04-11 | 2013-08-13 | Nippon Soda Co., Ltd. | Optically active dibenzazepine derivatives |
CN102267946B (zh) * | 2010-06-07 | 2014-09-10 | 中国科学院上海药物研究所 | 高光学纯度含手性联萘骨架的α-季碳氨基酸酯类化合物、其制备方法及用途 |
JP5673169B2 (ja) | 2011-02-08 | 2015-02-18 | 住友化学株式会社 | 4級アンモニウム塩及びそれを用いたシクロプロパン化合物の製造方法 |
ES2804528T3 (es) | 2011-07-05 | 2021-02-08 | Vertex Pharma | Procesos y productos intermedios para la producción de azaindoles |
JP2015003861A (ja) * | 2011-10-18 | 2015-01-08 | 株式会社カネカ | (r)−2−アミノ−2−エチルヘキサノールの製造法 |
WO2013148550A1 (en) * | 2012-03-30 | 2013-10-03 | Merck Sharp & Dohme Corp. | Asymmetric synthesis for preparing fluoroleucine alkyl esters |
JP6119022B2 (ja) * | 2012-06-05 | 2017-04-26 | 国立大学法人 岡山大学 | 軸不斉を有するピリジン誘導体又はその塩、及びその製造方法並びにそれからなる不斉触媒 |
JP5963140B2 (ja) * | 2012-10-12 | 2016-08-03 | 国立大学法人金沢大学 | 不斉脱水縮合剤 |
JP2016074605A (ja) * | 2013-02-18 | 2016-05-12 | 長瀬産業株式会社 | アミノ酸の製造方法およびアミノ酸合成キット |
CN103193673B (zh) * | 2013-03-19 | 2014-07-23 | 淮海工学院 | 季铵盐支载(水杨醛缩氨基酸)的功能配体及其制备方法 |
JP2017014109A (ja) * | 2013-11-21 | 2017-01-19 | 株式会社カネカ | 光学活性2,6−ジメチルチロシン誘導体の製造法 |
CN108940361B (zh) * | 2018-08-02 | 2020-12-01 | 吉林大学 | 一种手性离子型多孔有机聚合物材料及其制备方法与应用 |
CN112916042B (zh) * | 2021-01-29 | 2021-10-22 | 兰州交通大学 | 基于四甲基螺二氢茚骨架的手性季铵盐相转移催化剂及制备方法 |
CN113354681A (zh) * | 2021-05-07 | 2021-09-07 | 佛山奕安赛医药科技有限公司 | L-络氨酸衍生物不对称催化合成方法 |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6340753B1 (en) * | 2000-04-21 | 2002-01-22 | Nagase & Co., Ltd. | Optically active quarternary ammonium salt with axial chirality, method for producing thereof, and application thereof for asymmetric synthesis of α-amino acid |
JP4502293B2 (ja) * | 1999-06-04 | 2010-07-14 | 長瀬産業株式会社 | 軸不斉を有する光学活性な4級アンモニウム塩、その製法およびα−アミノ酸誘導体の不斉合成への応用 |
US6441231B1 (en) * | 2000-07-13 | 2002-08-27 | Nagase & Co., Ltd. | Optically active quarternary ammonium salt with axial chirality, method for producing thereof, and application thereof for asymmetric synthesis of α-amino acid |
JP2002173492A (ja) | 2000-12-07 | 2002-06-21 | Nagase & Co Ltd | 軸不斉を有する光学活性な4級アンモニウム塩とそれを用いたβ−ヒドロキシケトンの立体選択的合成 |
JP2002326992A (ja) * | 2001-05-02 | 2002-11-15 | Nagase & Co Ltd | ビナフチル基およびビフェニル基を含むn−スピロ不斉相間移動触媒 |
JP4782329B2 (ja) | 2001-07-02 | 2011-09-28 | 長瀬産業株式会社 | キラル相間移動触媒およびそれを用いた不斉ペプチドの製造方法 |
JP4415543B2 (ja) | 2002-12-13 | 2010-02-17 | 三菱化学株式会社 | 光学活性6,6’−ジメチル−1,1’−ビフェニル−2,2’−ジオール誘導体の製造方法 |
JP4360096B2 (ja) | 2003-02-07 | 2009-11-11 | 東ソー株式会社 | 光学活性四級アンモニウム塩、その製造方法、及びこれを相間移動触媒として用いた光学活性α−アミノ酸誘導体の製造方法 |
JP4322051B2 (ja) | 2003-06-03 | 2009-08-26 | 日本曹達株式会社 | 光学活性4級アンモニウム塩化合物およびその合成中間体 |
JP4474861B2 (ja) | 2003-07-23 | 2010-06-09 | 東ソー株式会社 | 光学活性四級アンモニウム塩、その製造法、並びにそれを用いた光学活性α−アミノ酸誘導体の製造法 |
EP1650212B1 (en) * | 2003-07-23 | 2012-11-14 | Tosoh Corporation | Optically active quaternary ammonium salt, process for producing the same, and process for producing optically active alpha-amino acid derivative with the same |
EP1712549B1 (en) * | 2004-01-30 | 2018-04-11 | Nagase & Company, Ltd. | Optically active quaternary ammonium salt having axial asymmetry and process for producing alpha-amino acid and derivative thereof with the same |
WO2006054366A1 (ja) * | 2004-11-22 | 2006-05-26 | Nagase & Co., Ltd. | 軸不斉を有する光学活性な4級アンモニウム塩を用いたアミノ酸およびその誘導体の製造方法 |
JP5296375B2 (ja) | 2005-03-03 | 2013-09-25 | 日本曹達株式会社 | 2つの軸不斉を有する光学活性アンモニウム塩化合物の製造方法 |
JP5008553B2 (ja) * | 2005-03-29 | 2012-08-22 | 長瀬産業株式会社 | 軸不斉を有する光学活性な4級アンモニウム塩およびそれを用いたα−アミノ酸およびその誘導体の製造方法 |
JP4879896B2 (ja) * | 2005-07-29 | 2012-02-22 | 長瀬産業株式会社 | アルジミンまたはその誘導体を用いる一置換アルキル化化合物の製造方法 |
JP5108777B2 (ja) * | 2006-09-28 | 2012-12-26 | 長瀬産業株式会社 | 軸不斉を有する光学活性な4級アンモニウム塩およびそれを用いたα−アミノ酸およびその誘導体の製造方法 |
-
2005
- 2005-01-27 EP EP05704383.8A patent/EP1712549B1/en not_active Not-in-force
- 2005-01-27 WO PCT/JP2005/001623 patent/WO2005073196A1/ja not_active Application Discontinuation
- 2005-01-27 CA CA2549431A patent/CA2549431C/en active Active
- 2005-01-27 JP JP2005517573A patent/JP4605606B2/ja active Active
- 2005-01-27 CN CN2005800037166A patent/CN1914177B/zh active Active
- 2005-01-27 US US10/587,467 patent/US7928224B2/en active Active
- 2005-01-27 SG SG200900527-3A patent/SG149879A1/en unknown
-
2007
- 2007-01-23 US US11/626,228 patent/US8697910B2/en active Active
-
2010
- 2010-04-16 JP JP2010095535A patent/JP5244149B2/ja active Active
-
2011
- 2011-03-03 US US13/039,645 patent/US8716524B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
WO2005073196A1 (ja) | 2005-08-11 |
CA2549431C (en) | 2010-09-14 |
EP1712549B1 (en) | 2018-04-11 |
CA2549431A1 (en) | 2005-08-11 |
US20110152562A1 (en) | 2011-06-23 |
US7928224B2 (en) | 2011-04-19 |
EP1712549A4 (en) | 2009-08-05 |
CN1914177A (zh) | 2007-02-14 |
US8716524B2 (en) | 2014-05-06 |
JP4605606B2 (ja) | 2011-01-05 |
JP2010222358A (ja) | 2010-10-07 |
JPWO2005073196A1 (ja) | 2007-11-15 |
JP5244149B2 (ja) | 2013-07-24 |
CN1914177B (zh) | 2011-10-12 |
US20070135654A1 (en) | 2007-06-14 |
EP1712549A1 (en) | 2006-10-18 |
US20070161624A1 (en) | 2007-07-12 |
US8697910B2 (en) | 2014-04-15 |
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