SG11201806863WA - Tetracyclic pyridone compounds as antivirals - Google Patents
Tetracyclic pyridone compounds as antiviralsInfo
- Publication number
- SG11201806863WA SG11201806863WA SG11201806863WA SG11201806863WA SG11201806863WA SG 11201806863W A SG11201806863W A SG 11201806863WA SG 11201806863W A SG11201806863W A SG 11201806863WA SG 11201806863W A SG11201806863W A SG 11201806863WA SG 11201806863W A SG11201806863W A SG 11201806863WA
- Authority
- SG
- Singapore
- Prior art keywords
- novartis
- international
- emeryville
- chiron
- way
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/08—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with a hetero atom directly attached to the ring nitrogen atom
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
- C07D491/147—Ortho-condensed systems the condensed system containing one ring with oxygen as ring hetero atom and two rings with nitrogen as ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Virology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201662297590P | 2016-02-19 | 2016-02-19 | |
US201662434658P | 2016-12-15 | 2016-12-15 | |
PCT/EP2017/053568 WO2017140821A1 (fr) | 2016-02-19 | 2017-02-16 | Composés pyridones tétracycliques en tant qu'agents antiviraux |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11201806863WA true SG11201806863WA (en) | 2018-09-27 |
Family
ID=58046696
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201806863WA SG11201806863WA (en) | 2016-02-19 | 2017-02-16 | Tetracyclic pyridone compounds as antivirals |
Country Status (21)
Country | Link |
---|---|
US (3) | US20200270265A1 (fr) |
EP (1) | EP3416946B1 (fr) |
JP (1) | JP7016809B2 (fr) |
KR (1) | KR20180110131A (fr) |
CN (1) | CN109071447B (fr) |
AU (1) | AU2017219216B2 (fr) |
BR (1) | BR112018016842A2 (fr) |
CA (1) | CA3014369A1 (fr) |
CO (1) | CO2018008589A2 (fr) |
EA (1) | EA038098B1 (fr) |
EC (1) | ECSP18069924A (fr) |
ES (1) | ES2897913T3 (fr) |
IL (1) | IL261158B (fr) |
JO (1) | JOP20170045B1 (fr) |
MX (1) | MX2018010010A (fr) |
PH (1) | PH12018501736A1 (fr) |
SG (1) | SG11201806863WA (fr) |
TW (1) | TWI747879B (fr) |
UY (1) | UY37128A (fr) |
WO (1) | WO2017140821A1 (fr) |
ZA (1) | ZA201805032B (fr) |
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EA038098B1 (ru) * | 2016-02-19 | 2021-07-06 | Новартис Аг | Тетрациклические пиридоновые соединения в качестве противовирусных средств |
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CN106928215B (zh) * | 2017-03-06 | 2019-03-22 | 河南春风医药科技有限公司 | 一种喹嗪酮类化合物的制备方法 |
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2017
- 2017-02-16 EA EA201891876A patent/EA038098B1/ru unknown
- 2017-02-16 EP EP17705425.1A patent/EP3416946B1/fr active Active
- 2017-02-16 SG SG11201806863WA patent/SG11201806863WA/en unknown
- 2017-02-16 US US15/999,664 patent/US20200270265A1/en not_active Abandoned
- 2017-02-16 UY UY0001037128A patent/UY37128A/es not_active Application Discontinuation
- 2017-02-16 BR BR112018016842A patent/BR112018016842A2/pt not_active Application Discontinuation
- 2017-02-16 CN CN201780024193.6A patent/CN109071447B/zh active Active
- 2017-02-16 ES ES17705425T patent/ES2897913T3/es active Active
- 2017-02-16 CA CA3014369A patent/CA3014369A1/fr not_active Abandoned
- 2017-02-16 JP JP2018543679A patent/JP7016809B2/ja active Active
- 2017-02-16 JO JOP/2017/0045A patent/JOP20170045B1/ar active
- 2017-02-16 WO PCT/EP2017/053568 patent/WO2017140821A1/fr active Application Filing
- 2017-02-16 KR KR1020187026639A patent/KR20180110131A/ko unknown
- 2017-02-16 AU AU2017219216A patent/AU2017219216B2/en not_active Ceased
- 2017-02-16 MX MX2018010010A patent/MX2018010010A/es unknown
- 2017-02-16 US US15/435,137 patent/US9845325B2/en active Active
- 2017-02-18 TW TW106105419A patent/TWI747879B/zh active
- 2017-10-12 US US15/782,722 patent/US10093673B2/en active Active
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2018
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- 2018-08-14 IL IL261158A patent/IL261158B/en active IP Right Grant
- 2018-08-15 CO CONC2018/0008589A patent/CO2018008589A2/es unknown
- 2018-08-16 PH PH12018501736A patent/PH12018501736A1/en unknown
- 2018-09-14 EC ECSENADI201869924A patent/ECSP18069924A/es unknown
Also Published As
Publication number | Publication date |
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CN109071447A (zh) | 2018-12-21 |
JP7016809B2 (ja) | 2022-02-07 |
EA038098B1 (ru) | 2021-07-06 |
MX2018010010A (es) | 2018-11-09 |
EA201891876A1 (ru) | 2019-01-31 |
UY37128A (es) | 2017-09-29 |
US20180030053A1 (en) | 2018-02-01 |
EP3416946B1 (fr) | 2021-09-15 |
JOP20170045B1 (ar) | 2021-08-17 |
KR20180110131A (ko) | 2018-10-08 |
EP3416946A1 (fr) | 2018-12-26 |
CO2018008589A2 (es) | 2018-08-21 |
WO2017140821A1 (fr) | 2017-08-24 |
TWI747879B (zh) | 2021-12-01 |
AU2017219216B2 (en) | 2019-12-19 |
IL261158A (en) | 2018-10-31 |
PH12018501736A1 (en) | 2019-06-17 |
BR112018016842A2 (pt) | 2018-12-26 |
ZA201805032B (en) | 2019-08-28 |
US10093673B2 (en) | 2018-10-09 |
US20200270265A1 (en) | 2020-08-27 |
US20170240548A1 (en) | 2017-08-24 |
ECSP18069924A (es) | 2018-09-30 |
US9845325B2 (en) | 2017-12-19 |
AU2017219216A1 (en) | 2018-08-30 |
CA3014369A1 (fr) | 2017-08-24 |
JP2019509276A (ja) | 2019-04-04 |
ES2897913T3 (es) | 2022-03-03 |
TW201804995A (zh) | 2018-02-16 |
CN109071447B (zh) | 2022-04-22 |
IL261158B (en) | 2020-10-29 |
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