SG11201708793SA - Crystals of azabicyclic compound - Google Patents

Crystals of azabicyclic compound

Info

Publication number
SG11201708793SA
SG11201708793SA SG11201708793SA SG11201708793SA SG11201708793SA SG 11201708793S A SG11201708793S A SG 11201708793SA SG 11201708793S A SG11201708793S A SG 11201708793SA SG 11201708793S A SG11201708793S A SG 11201708793SA SG 11201708793S A SG11201708793S A SG 11201708793SA
Authority
SG
Singapore
Prior art keywords
crystals
azabicyclic compound
azabicyclic
compound
Prior art date
Application number
SG11201708793SA
Other languages
English (en)
Inventor
Takao Uno
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of SG11201708793SA publication Critical patent/SG11201708793SA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
SG11201708793SA 2015-05-12 2016-05-11 Crystals of azabicyclic compound SG11201708793SA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2015097521 2015-05-12
PCT/JP2016/063989 WO2016181990A1 (ja) 2015-05-12 2016-05-11 アザ二環式化合物の結晶

Publications (1)

Publication Number Publication Date
SG11201708793SA true SG11201708793SA (en) 2017-11-29

Family

ID=57248173

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201708793SA SG11201708793SA (en) 2015-05-12 2016-05-11 Crystals of azabicyclic compound

Country Status (20)

Country Link
US (2) US10526324B2 (ru)
EP (1) EP3296299B1 (ru)
JP (1) JP6537601B2 (ru)
KR (1) KR102089254B1 (ru)
CN (1) CN107531707B (ru)
AU (1) AU2016260279B2 (ru)
BR (1) BR112017024367B1 (ru)
CA (1) CA2985033C (ru)
DK (1) DK3296299T3 (ru)
ES (1) ES2760503T3 (ru)
HU (1) HUE047855T2 (ru)
MX (1) MX2017014438A (ru)
MY (1) MY189352A (ru)
PH (1) PH12017502007A1 (ru)
PL (1) PL3296299T3 (ru)
PT (1) PT3296299T (ru)
RU (1) RU2697521C2 (ru)
SG (1) SG11201708793SA (ru)
TW (1) TWI659954B (ru)
WO (1) WO2016181990A1 (ru)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2020002886A (es) * 2017-09-15 2020-10-01 Taiho Pharmaceutical Co Ltd Agente profilactico y/o terapeutico para enfermedades que involucran la expresion de ido.
CN112584837A (zh) 2018-08-31 2021-03-30 细胞内治疗公司 新方法
CA3108558A1 (en) 2018-08-31 2020-03-05 Intra-Cellular Therapies, Inc. Novel methods
US11753419B2 (en) 2019-12-11 2023-09-12 Intra-Cellular Therapies, Inc. 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3′4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)phenyl)butan-1-one for treating conditions of the central nervous system and cardiac disorders
CN114685492A (zh) * 2020-12-31 2022-07-01 杭州领业医药科技有限公司 Tas-116的晶型及其制备方法、药物组合物和用途
TW202404585A (zh) * 2022-06-10 2024-02-01 日商大鵬藥品工業股份有限公司 含有匹密特匹(Pimitespib)之醫藥組合物
WO2023238930A1 (ja) * 2022-06-10 2023-12-14 大鵬薬品工業株式会社 アザ二環式化合物の類縁物質
CN115960100B (zh) * 2022-12-28 2023-08-18 北京康立生医药技术开发有限公司 一种治疗胃肠道间质瘤药物皮咪特昔布的合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL375993A1 (en) 2002-09-16 2005-12-12 Glaxo Group Limited Pyrazolo[3,4-b]pyridine compounds, and their use as phosphodiesterase inhibitors
RU2357967C2 (ru) * 2002-09-16 2009-06-10 Глаксо Груп Лимитед ПРОИЗВОДНЫЕ ПИРАЗОЛО[3, 4-b]ПИРИДИНА, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ (ВАРИАНТЫ), ПРИМЕНЕНИЕ (ВАРИАНТЫ), КОМПОЗИЦИЯ (ВАРИАНТЫ)
WO2011004610A1 (ja) * 2009-07-10 2011-01-13 大鵬薬品工業株式会社 アザ二環式化合物又はその塩
MX2013007938A (es) 2011-01-07 2013-11-01 Taiho Pharmaceutical Co Ltd Compuesto biciclico novedoso o sal del mismo.
AU2014325016C1 (en) * 2013-09-30 2021-10-07 Taiho Pharmaceutical Co., Ltd. Combination therapy using azabicyclo compound for cancer

Also Published As

Publication number Publication date
JP6537601B2 (ja) 2019-07-03
KR102089254B1 (ko) 2020-03-16
BR112017024367A2 (pt) 2018-07-31
HUE047855T2 (hu) 2020-05-28
WO2016181990A1 (ja) 2016-11-17
RU2017142958A3 (ru) 2019-06-13
TW201704234A (zh) 2017-02-01
BR112017024367B1 (pt) 2023-05-09
ES2760503T3 (es) 2020-05-14
US20200102304A1 (en) 2020-04-02
CA2985033A1 (en) 2016-11-17
CN107531707B (zh) 2020-01-10
PT3296299T (pt) 2019-12-13
EP3296299A4 (en) 2018-10-24
US10526324B2 (en) 2020-01-07
CN107531707A (zh) 2018-01-02
MY189352A (en) 2022-02-07
AU2016260279A1 (en) 2017-11-30
KR20180003558A (ko) 2018-01-09
DK3296299T3 (da) 2019-12-16
EP3296299B1 (en) 2019-10-02
TWI659954B (zh) 2019-05-21
US20180148443A1 (en) 2018-05-31
JPWO2016181990A1 (ja) 2018-03-01
US10947233B2 (en) 2021-03-16
PH12017502007A1 (en) 2018-03-26
PL3296299T3 (pl) 2020-04-30
CA2985033C (en) 2020-02-25
RU2697521C2 (ru) 2019-08-15
EP3296299A1 (en) 2018-03-21
MX2017014438A (es) 2018-03-02
RU2017142958A (ru) 2019-06-13
AU2016260279B2 (en) 2019-03-14

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