SG10201406805RA - Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one - Google Patents

Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one

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Publication number
SG10201406805RA
SG10201406805RA SG10201406805RA SG10201406805RA SG10201406805RA SG 10201406805R A SG10201406805R A SG 10201406805RA SG 10201406805R A SG10201406805R A SG 10201406805RA SG 10201406805R A SG10201406805R A SG 10201406805RA SG 10201406805R A SG10201406805R A SG 10201406805RA
Authority
SG
Singapore
Prior art keywords
azepino
polymorphs
indol
methylamino
tetrahydro
Prior art date
Application number
SG10201406805RA
Other languages
English (en)
Inventor
Patricia Ann Basford
Anthony Michael Campeta
Adam Gillmore
Matthew Cameron Jones
Robert Walton
Eleftherios Kougoulos
Suman Luthra
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43859823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201406805R(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of SG10201406805RA publication Critical patent/SG10201406805RA/en

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/19—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
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    • C07C57/145—Maleic acid
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    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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SG10201406805RA 2010-02-12 2011-02-10 Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one SG10201406805RA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30427710P 2010-02-12 2010-02-12

Publications (1)

Publication Number Publication Date
SG10201406805RA true SG10201406805RA (en) 2014-11-27

Family

ID=43859823

Family Applications (2)

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SG2012052171A SG182533A1 (en) 2010-02-12 2011-02-10 Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one
SG10201406805RA SG10201406805RA (en) 2010-02-12 2011-02-10 Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one

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SG2012052171A SG182533A1 (en) 2010-02-12 2011-02-10 Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one

Country Status (31)

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US (5) US8754072B2 (zh)
EP (4) EP3597651A1 (zh)
JP (6) JP5745283B2 (zh)
KR (2) KR20120127495A (zh)
CN (2) CN104876937B (zh)
AR (2) AR080164A1 (zh)
AU (1) AU2011213944B2 (zh)
BR (1) BR112012019050B1 (zh)
CA (2) CA3024216C (zh)
CY (3) CY1118319T1 (zh)
DK (2) DK2534153T3 (zh)
ES (2) ES2753748T3 (zh)
HK (1) HK1176617A1 (zh)
HR (2) HRP20161742T1 (zh)
HU (3) HUE047248T2 (zh)
IL (1) IL220921B (zh)
LT (3) LT3150610T (zh)
LU (1) LUC00093I2 (zh)
MX (1) MX343383B (zh)
NL (1) NL300958I2 (zh)
NO (1) NO2018039I1 (zh)
NZ (1) NZ601445A (zh)
PL (2) PL3150610T3 (zh)
PT (2) PT2534153T (zh)
RS (2) RS59494B1 (zh)
RU (1) RU2570198C2 (zh)
SG (2) SG182533A1 (zh)
SI (2) SI2534153T1 (zh)
SM (1) SMT201600462B (zh)
TW (1) TWI545123B (zh)
WO (1) WO2011098971A1 (zh)

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