SE0301372D0 - Novel compounds - Google Patents

Novel compounds

Info

Publication number
SE0301372D0
SE0301372D0 SE0301372A SE0301372A SE0301372D0 SE 0301372 D0 SE0301372 D0 SE 0301372D0 SE 0301372 A SE0301372 A SE 0301372A SE 0301372 A SE0301372 A SE 0301372A SE 0301372 D0 SE0301372 D0 SE 0301372D0
Authority
SE
Sweden
Prior art keywords
novel compounds
methods
pharmaceutical compositions
relates
present
Prior art date
Application number
SE0301372A
Other languages
English (en)
Swedish (sv)
Inventor
Peter Hansen
David Laurent
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0301372A priority Critical patent/SE0301372D0/xx
Publication of SE0301372D0 publication Critical patent/SE0301372D0/xx
Priority to ES04731527T priority patent/ES2286634T3/es
Priority to AU2004236146A priority patent/AU2004236146B2/en
Priority to MXPA05012026A priority patent/MXPA05012026A/es
Priority to PCT/SE2004/000696 priority patent/WO2004099205A1/en
Priority to US10/556,227 priority patent/US20060287354A1/en
Priority to JP2006508046A priority patent/JP2006525998A/ja
Priority to CA002523922A priority patent/CA2523922A1/en
Priority to BRPI0410117-0A priority patent/BRPI0410117A/pt
Priority to CNA2004800126269A priority patent/CN1784403A/zh
Priority to AT04731527T priority patent/ATE362932T1/de
Priority to EP04731527A priority patent/EP1625127B1/en
Priority to DE602004006618T priority patent/DE602004006618T2/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SE0301372A 2003-05-09 2003-05-09 Novel compounds SE0301372D0 (sv)

Priority Applications (13)

Application Number Priority Date Filing Date Title
SE0301372A SE0301372D0 (sv) 2003-05-09 2003-05-09 Novel compounds
DE602004006618T DE602004006618T2 (de) 2003-05-09 2004-05-06 Azaindolverbindungen als kinaseinhibitoren
PCT/SE2004/000696 WO2004099205A1 (en) 2003-05-09 2004-05-06 Azaindole compounds as kinase inhibitors
AU2004236146A AU2004236146B2 (en) 2003-05-09 2004-05-06 Azaindole compounds as kinase inhibitors
MXPA05012026A MXPA05012026A (es) 2003-05-09 2004-05-06 Compuestos de azaindol como inhibidores de cinasa.
ES04731527T ES2286634T3 (es) 2003-05-09 2004-05-06 Compuestos de azaindol como inhibidores de quinasas.
US10/556,227 US20060287354A1 (en) 2003-05-09 2004-05-06 Azaindole compounds as kinase inhibitors
JP2006508046A JP2006525998A (ja) 2003-05-09 2004-05-06 キナーゼ阻害剤としてのアザインドール化合物
CA002523922A CA2523922A1 (en) 2003-05-09 2004-05-06 Azaindole compounds as kinase inhibitors
BRPI0410117-0A BRPI0410117A (pt) 2003-05-09 2004-05-06 composto, composição farmacêutica, método para o tratamento de uma doença ou condição mediada por jak3, e, processo para a preparação de um composto
CNA2004800126269A CN1784403A (zh) 2003-05-09 2004-05-06 作为激酶抑制剂的吖吲哚化合物
AT04731527T ATE362932T1 (de) 2003-05-09 2004-05-06 Azaindolverbindungen als kinaseinhibitoren
EP04731527A EP1625127B1 (en) 2003-05-09 2004-05-06 Azaindole compounds as kinase inhibitors

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0301372A SE0301372D0 (sv) 2003-05-09 2003-05-09 Novel compounds

Publications (1)

Publication Number Publication Date
SE0301372D0 true SE0301372D0 (sv) 2003-05-09

Family

ID=20291270

Family Applications (1)

Application Number Title Priority Date Filing Date
SE0301372A SE0301372D0 (sv) 2003-05-09 2003-05-09 Novel compounds

Country Status (13)

Country Link
US (1) US20060287354A1 (es)
EP (1) EP1625127B1 (es)
JP (1) JP2006525998A (es)
CN (1) CN1784403A (es)
AT (1) ATE362932T1 (es)
AU (1) AU2004236146B2 (es)
BR (1) BRPI0410117A (es)
CA (1) CA2523922A1 (es)
DE (1) DE602004006618T2 (es)
ES (1) ES2286634T3 (es)
MX (1) MXPA05012026A (es)
SE (1) SE0301372D0 (es)
WO (1) WO2004099205A1 (es)

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EP2274288A2 (en) 2008-04-24 2011-01-19 Incyte Corporation Macrocyclic compounds and their use as kinase inhibitors
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WO2010058846A1 (ja) * 2008-11-21 2010-05-27 アステラス製薬株式会社 ４，６-ジアミノニコチンアミド化合物
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CN106967070A (zh) 2009-05-22 2017-07-21 因塞特控股公司 作为jak抑制剂的化合物
KR101771401B1 (ko) 2009-05-22 2017-08-25 인사이트 홀딩스 코포레이션 야누스 키나제 억제제로서 피라졸­４­일­피롤로［２,３­ｄ］피리미딘 및 피롤­３­일­피롤로［２,３­ｄ］피리미딘의 Ｎ­(헤테로)아릴­피롤리딘 유도체
US8299103B2 (en) 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
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UA110324C2 (en) * 2009-07-02 2015-12-25 Genentech Inc Jak inhibitory compounds based on pyrazolo pyrimidine
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US9315454B2 (en) 2010-01-15 2016-04-19 Boehringer Ingelheim International Gmbh Compounds which modulate the CB2 receptor
US8329735B2 (en) 2010-03-05 2012-12-11 Boehringer Ingelheim International Gmbh Tetrazole compounds which selectively modulate the CB2 receptor
SI3050882T1 (en) 2010-03-10 2018-06-29 Incyte Holdings Corporation Piperidin-4-yl azetidine derivatives, as inhibitors of JAK1
EA202091303A3 (ru) 2010-05-21 2021-05-31 Инсайт Холдингс Корпорейшн Композиция ингибитора jak для местного применения
WO2012012307A1 (en) 2010-07-22 2012-01-26 Boehringer Ingelheim International Gmbh Sulfonyl compounds which modulate the cb2 rece
AR083933A1 (es) 2010-11-19 2013-04-10 Incyte Corp Derivados de pirrolopiridina y pirrolopirimidina sustituidos con ciclobutilo como inhibidores de jak
WO2012068440A1 (en) 2010-11-19 2012-05-24 Incyte Corporation Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
WO2012093169A1 (en) 2011-01-07 2012-07-12 Leo Pharma A/S Novel sulfamide piperazine derivatives as protein tyrosine kinase inhibitors and pharmaceutical use thereof
EP2675451B9 (en) 2011-02-18 2017-07-26 Novartis Pharma AG mTOR/JAK INHIBITOR COMBINATION THERAPY
JP6277121B2 (ja) 2011-03-22 2018-02-07 アドヴィナス・セラピューティックス・リミテッド 置換された縮合三環式化合物、その組成物および医学的応用
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SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
SE0301373D0 (sv) * 2003-05-09 2003-05-09 Astrazeneca Ab Novel compounds

Also Published As

Publication number Publication date
EP1625127A1 (en) 2006-02-15
US20060287354A1 (en) 2006-12-21
ATE362932T1 (de) 2007-06-15
AU2004236146A1 (en) 2004-11-18
JP2006525998A (ja) 2006-11-16
CA2523922A1 (en) 2004-11-18
EP1625127B1 (en) 2007-05-23
CN1784403A (zh) 2006-06-07
DE602004006618D1 (de) 2007-07-05
MXPA05012026A (es) 2006-02-03
WO2004099205A1 (en) 2004-11-18
BRPI0410117A (pt) 2006-05-23
ES2286634T3 (es) 2007-12-01
DE602004006618T2 (de) 2008-01-31
AU2004236146B2 (en) 2007-12-13

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