RU95107706A - Пиридоиндолобензодиазепины и их производные, фармацевтическая композиция антипсихоточеского действия на их основе и способ лечения - Google Patents

Пиридоиндолобензодиазепины и их производные, фармацевтическая композиция антипсихоточеского действия на их основе и способ лечения

Info

Publication number
RU95107706A
RU95107706A RU95107706/14A RU95107706A RU95107706A RU 95107706 A RU95107706 A RU 95107706A RU 95107706/14 A RU95107706/14 A RU 95107706/14A RU 95107706 A RU95107706 A RU 95107706A RU 95107706 A RU95107706 A RU 95107706A
Authority
RU
Russia
Prior art keywords
medical treatment
pyridoindolobenzodiazepines
derivatives
pharmaceutical composition
activity based
Prior art date
Application number
RU95107706/14A
Other languages
English (en)
Russian (ru)
Inventor
Партасарати Раджагопалан
Us]
Original Assignee
Дю Пон Мерк Фармацьютикал Компани (US)
Дю Пон Мерк Фармацьютикал Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Дю Пон Мерк Фармацьютикал Компани (US), Дю Пон Мерк Фармацьютикал Компани filed Critical Дю Пон Мерк Фармацьютикал Компани (US)
Publication of RU95107706A publication Critical patent/RU95107706A/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A61P39/02—Antidotes

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Toxicology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
RU95107706/14A 1992-07-29 1993-07-23 Пиридоиндолобензодиазепины и их производные, фармацевтическая композиция антипсихоточеского действия на их основе и способ лечения RU95107706A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/921,051 1992-07-29
US07/921,051 US5321023A (en) 1992-07-29 1992-07-29 Pyridoindolobenzodiazepines and derivatives as antipsychotics

Publications (1)

Publication Number Publication Date
RU95107706A true RU95107706A (ru) 1997-03-20

Family

ID=25444846

Family Applications (1)

Application Number Title Priority Date Filing Date
RU95107706/14A RU95107706A (ru) 1992-07-29 1993-07-23 Пиридоиндолобензодиазепины и их производные, фармацевтическая композиция антипсихоточеского действия на их основе и способ лечения

Country Status (22)

Country Link
US (1) US5321023A (enExample)
EP (1) EP0652878A1 (enExample)
JP (1) JPH08500579A (enExample)
KR (1) KR950702562A (enExample)
CN (1) CN1100424A (enExample)
AU (1) AU4685393A (enExample)
BR (1) BR9306896A (enExample)
CA (1) CA2141332A1 (enExample)
CZ (1) CZ19895A3 (enExample)
FI (1) FI950303A7 (enExample)
HR (1) HRP931082A2 (enExample)
HU (1) HUT69393A (enExample)
IL (1) IL106352A0 (enExample)
MX (1) MX9304552A (enExample)
NO (1) NO950327D0 (enExample)
NZ (1) NZ254650A (enExample)
PL (1) PL307231A1 (enExample)
RU (1) RU95107706A (enExample)
SK (1) SK40395A3 (enExample)
TW (1) TW260670B (enExample)
WO (1) WO1994003455A1 (enExample)
ZA (1) ZA935486B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19546297C2 (de) 1995-12-12 2003-12-04 Temic Bayern Chem Airbag Gmbh Airbagsystem mit variablem Auslösezeitpunkt
US8367655B2 (en) * 2009-07-03 2013-02-05 Daya Drug Discoveries, Inc. Pyridoindolobenzox—and thiazepine derivatives and uses thereof
WO2014137849A1 (en) * 2013-03-04 2014-09-12 Daya Drug Discoveries, Inc Pentacyclic pyridoindolo[b,e]azepine derivatives and uses thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3373168A (en) * 1964-06-02 1968-03-12 Hoffmann La Roche Certain benzazepinoxyridoindole compounds and their preparation
US3457271A (en) * 1964-06-02 1969-07-22 Hoffmann La Roche 11-lower alkyl-hexahydro-1-benzazepino (3,2,1-h,i)pyrido(4,3-b)indole
US3764684A (en) * 1971-08-11 1973-10-09 M Finizio Novel indolobenzazepine derivatives, useful as tranquilizers
US3790675A (en) * 1972-04-19 1974-02-05 Endo Lab Certain indolobenzazepine derivatives as analgesics
US3932650A (en) * 1973-01-22 1976-01-13 E. I. Du Pont De Nemours & Company Trans-octahydropyridoindolobenzazepines as central nervous system depressants
US3890327A (en) * 1973-05-11 1975-06-17 Du Pont Trans-1,2,3,4,4a,8,9,14a-octahydropyrido(r',3':2,3)indolo(1,7-ab)+8 1)benzazepine
US3983123A (en) * 1973-01-22 1976-09-28 Endo Laboratories, Inc. Trans-octahydropyridoindolobenzazepines
CA1026331A (en) * 1973-12-06 1978-02-14 Joel G. Berger Substituted indolobenzazepines
US4438120A (en) * 1982-11-12 1984-03-20 E. I. Du Pont De Nemours & Company Pyridoindolobenzodiazepine tranquilizers

Also Published As

Publication number Publication date
US5321023A (en) 1994-06-14
NO950327L (no) 1995-01-27
FI950303L (fi) 1995-01-24
FI950303A0 (fi) 1995-01-24
AU4685393A (en) 1994-03-03
TW260670B (enExample) 1995-10-21
NO950327D0 (no) 1995-01-27
ZA935486B (en) 1995-01-30
CN1100424A (zh) 1995-03-22
PL307231A1 (en) 1995-05-15
BR9306896A (pt) 1998-12-08
HRP931082A2 (en) 1997-06-30
NZ254650A (en) 1996-03-26
WO1994003455A1 (en) 1994-02-17
HUT69393A (en) 1995-09-28
SK40395A3 (en) 1995-12-06
KR950702562A (ko) 1995-07-29
MX9304552A (es) 1994-05-31
EP0652878A1 (en) 1995-05-17
CA2141332A1 (en) 1994-02-17
FI950303A7 (fi) 1995-01-24
IL106352A0 (en) 1993-11-15
CZ19895A3 (en) 1995-11-15
HU9500193D0 (en) 1995-03-28
JPH08500579A (ja) 1996-01-23

Similar Documents

Publication Publication Date Title
RU94038043A (ru) Применение замещенных производных аденина для лечения множественного склероза
BG103417A (en) Condensed pyrimidine bicyclic derivatives
UA41297C2 (uk) Похідні індолу, фармацевтична композиція і спосіб лікування
ATE4903T1 (de) 1-, 6- und 2-substituierte 1-carba-2-penem-3carbons[ure, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen.
RU94042922A (ru) Новые соединения, способы их получения, фармацевтическая композиция
MXPA05009245A (es) Nuevos compuestos de pirazina como inhibidores del factor de crecimiento transformante (tgf).
BR0014596A (pt) Derivado de pirimidina, uso do mesmo, composição farmacêutica, e, método de tratar doenças ou condições médicas mediadas por citocinas
NZ225344A (en) 3-demethylmevalonic acid derivatives and lactones and pharmaceutical compositions; intermediates for the preparation thereof
FI946073A0 (fi) Vitamiini D-sarjan, 20-asemassa modifioituja johdannaisia, menetelmä tällaisten johdannaisten valmistamiseksi, menetelmässä käytettäviä välituotteita, mainittuja johdannaisia sisältäviä farmaseuttisia valmisteita ja johdannaisten käyttö lääkeaineiden valmistamiseen
EA200100127A1 (ru) Производные фенилксантина
JPS57501963A (enExample)
ATE226953T1 (de) 3-,8-substituierte deuteroporphyrinderivate, diese enthaltende pharmazeutische mittel und verfahren zu ihrer herstellung
RU95110937A (ru) Хинолоновые и акридиноновые соединения, способ их получения, фармацевтическая композиция и промежуточные соединения
RU95111308A (ru) Производные 2-амино-4-фенил-4-оксомасляной кислоты, способы получения, фармацевтическая композиция
MX9203417A (es) Compuestos de diarilo antiateroescleroticos.
CA2238875A1 (en) Tri-aryl ethane derivatives as pde iv inhibitors
MX9706605A (es) Derivados de indol como antagonistas de los aminoacidos exitadores.
EE03771B1 (et) Tetrahüdropüridoühendid, neid sisaldav ravim ja nende kasutamine
AU611113B2 (en) Basically substituted phenylacetonitriles, their preparation and drugs containing these compounds
NO883074L (no) Fremgangsmaate til fremstilling av 3-desmetyl-4-fluor-mevalonsyrederivater.
DE3686979D1 (de) Cephemverbindungen und verfahren zu ihrer herstellung.
UA48958C2 (uk) 9-o-оксимові похідні еритроміцину а та фармацевтична композиція на їх основі
ZA826453B (en) Tricyclic thiazolyloxamic acids and their derivatives,their preparation,and therapeutic agents containing these compounds
IL89335A (en) 6-oxo-pyridazine derivatives, a process for their preparation and pharmaceutical compositions containing these compounds
TNSN01001A1 (fr) NOUVELLES PYRAZOLO [4,3-e] DIAZEPINES SUBSTITUEES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, UTILISATION A TITRE DE MEDICAMENT ET PROCEDES POUR LEUR PREPARATION