RU93004666A - Сульфонамидокарбоксимиды - Google Patents

Сульфонамидокарбоксимиды

Info

Publication number
RU93004666A
RU93004666A RU93004666/04A RU93004666A RU93004666A RU 93004666 A RU93004666 A RU 93004666A RU 93004666/04 A RU93004666/04 A RU 93004666/04A RU 93004666 A RU93004666 A RU 93004666A RU 93004666 A RU93004666 A RU 93004666A
Authority
RU
Russia
Prior art keywords
sulphonamidokarboximides
sulfonamidocarboxamides
amidation
fibrinogen
thrombin
Prior art date
Application number
RU93004666/04A
Other languages
English (en)
Other versions
RU2133739C1 (ru
Inventor
Акерманн Жан
Баннер Давид
Губернатор Клаус
Хильперт Курт
Шмид Жерар
Original Assignee
Ф.Хоффманн Ля Рош АГ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ф.Хоффманн Ля Рош АГ filed Critical Ф.Хоффманн Ля Рош АГ
Publication of RU93004666A publication Critical patent/RU93004666A/ru
Application granted granted Critical
Publication of RU2133739C1 publication Critical patent/RU2133739C1/ru

Links

Claims (1)

  1. Предложены новые сульфонамидокарбоксамиды формулы
    Figure 00000001

    где A, M, Q, X и Y имеют значения, указанные в описании, а также их гидраты или сольваты, подавляющие вызванное тромбинами скопление тромбоцитов и свертывание фибриногенов в плазме. Их получают путем амидирования циклической аминогруппы, служащей для образования группы X или образования амидов через C(O)N(Q).
RU93004666A 1992-03-06 1993-03-04 Сульфонамидокарбоксамиды, их гидраты и физиологически приемлемые соли, фармацевтическая композиция на их основе RU2133739C1 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH728/92 1992-03-04
CH72892 1992-03-06
CH18093 1993-01-21
CH180/93 1993-01-21

Publications (2)

Publication Number Publication Date
RU93004666A true RU93004666A (ru) 1996-04-27
RU2133739C1 RU2133739C1 (ru) 1999-07-27

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
RU93004666A RU2133739C1 (ru) 1992-03-06 1993-03-04 Сульфонамидокарбоксамиды, их гидраты и физиологически приемлемые соли, фармацевтическая композиция на их основе

Country Status (24)

Country Link
US (4) US5405854A (ru)
EP (1) EP0559046B1 (ru)
JP (1) JPH0780848B2 (ru)
CN (1) CN1076690A (ru)
AT (1) ATE203013T1 (ru)
AU (1) AU665230B2 (ru)
BG (1) BG61506B1 (ru)
CA (1) CA2089972C (ru)
CZ (1) CZ286926B6 (ru)
DE (1) DE59310186D1 (ru)
DK (1) DK0559046T3 (ru)
ES (1) ES2161217T3 (ru)
FI (1) FI103880B1 (ru)
GR (1) GR3036870T3 (ru)
HU (2) HUT70156A (ru)
IL (3) IL104893A0 (ru)
IS (1) IS3983A (ru)
MY (1) MY131303A (ru)
NO (1) NO302818B1 (ru)
NZ (1) NZ247014A (ru)
PT (1) PT559046E (ru)
RO (1) RO112863B1 (ru)
RU (1) RU2133739C1 (ru)
TW (1) TW223629B (ru)

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