RU2019117451A - Способ и композиция для неочищенных препаратов обогащенного сахара для гликемического контроля - Google Patents
Способ и композиция для неочищенных препаратов обогащенного сахара для гликемического контроля Download PDFInfo
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- RU2019117451A RU2019117451A RU2019117451A RU2019117451A RU2019117451A RU 2019117451 A RU2019117451 A RU 2019117451A RU 2019117451 A RU2019117451 A RU 2019117451A RU 2019117451 A RU2019117451 A RU 2019117451A RU 2019117451 A RU2019117451 A RU 2019117451A
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- inhibition
- polyphenol
- sweetener
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- 238000000034 method Methods 0.000 title claims 3
- 238000002360 preparation method Methods 0.000 title claims 3
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- 230000002641 glycemic effect Effects 0.000 title claims 2
- 238000009472 formulation Methods 0.000 claims 23
- 230000005764 inhibitory process Effects 0.000 claims 8
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- 229920002472 Starch Polymers 0.000 claims 6
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- 235000019698 starch Nutrition 0.000 claims 6
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- 239000003765 sweetening agent Substances 0.000 claims 6
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Claims (18)
1. Препарат, содержащий подсластитель, полифенол и крахмал.
2. Препарат по п. 1, где данный препарат смягчает гипергликемические эффекты при введении индивиду, нуждающемуся в этом.
3. Препарат по п. 2, где гипергликемическое состояние выбрано из группы, состоящей из метаболического синдрома, ожирения, диабета и неврологического заболевания.
4. Препарат по п. 1, дополнительно содержащий продукт питания, включающий напитки, хлебобулочные изделия, сладости, кондитерские изделия, покрытия, лечебное питание и медицинские препараты.
5. Препарат по п. 1, где композицию нагревали, и подсластитель ожижали таким образом, что полифенол и крахмал заключаются в перекристаллизованную форму подсластителя.
6. Препарат по п. 5, где данный препарат был заключен в столовый сахар, напитки, хлебобулочные изделия, сладости, кондитерские изделия, покрытия, лечебное питание и медицинские препараты.
7. Препарат по п. 1, где данный препарат распределяется и переносится в жидкой фазе подсластителя, такого как кукурузный сироп.
8. Препарат по п. 7, где данный препарат включается в напитки, хлебобулочные изделия, сладости, кондитерские изделия, покрытия, лечебное питание и медицинские препараты.
9. Препарат по п. 1, где подсластитель представляет собой углеводную основу как природной, так и полусинтетической природы, включающую моносахариды, дисахариды, олигосахариды и природные подсластители, включающие фруктозу, галактозу, сахарозу, дезоксирибозу, диозу, триозу, тетрозу, пентозу, гексозу, альдозу, фуранозу, пиранозу, глюкофуранозу, глюкопиранозу, сахарозу, лактулозу, лактозу, мальтозу, целлобиозу, хитобиозу, койибиозу, нигерлозу, изомальтозу, софорозу, ламиниарибиозу, туранозу, мальтулозу, палатинозу, маннобиозу, мелибиозу, мелибиулозу, рунтинозу, ксилобиозу, фруктоолигосахарид, галактоолигосахарид, манноолигосахарид, аспартам, цикламат, сахарин, стевию, сукралозу, калия ацесульфам, ацетат свинца, могрозиды, браззеин, куркулин, эритритол, глицирризин, глицерин, инулин, изомальт, лактит, мабинлин, мальтит, миракулин, монатин, монеллин, осладин, пентадин, сорбит, тагетозу, тауматин, ксилит, адвантам, элитам, дульцин, глюцин, неогесперидин, дигидрохалкон, неотам, р-4000, сахарин, L-рамнозу, L-глюкозу, L-маннозу, L-фукозу.
10. Препарат по п. 1, где по меньшей мере один из подсластителя, полифенола и крахмала имеет биоактивную фенольную природу, которые включают фенолы, флавонали, флавоноиды, биофлавоноиды, антоксантины, флаваноны, флаванолы, флаваны, антоцианидины, но не ограничиваются ими, в частности: апиол, карнозол, карвакрол, диллапиол, розмаринол, кверцетин, кемпферол, мирицетин, дигидромирицетин, физетин, рутин, изорамнетин, гесперитин, гесперидин, нарингин, нарингенин, силибин, эриодиктиол, акацетин, апигенин, хризин, диосметин, тангеритин, лютеолин, хризантему, катехин, галлокатехин, эпикатехин, эпигаллокатехин, эпигаллокатехин галлат, теафлавин, теарубигины, проантоцианодины, пелагонидин, пеонидин, цианидин, дельфинидин, малвидин, петунидин, дайдзеин, генистеин, глицитин, изофлаваны, изофлавандиолы, изофлавены, птерокарпаны, ауроны, халконоиды, резевератрол, птеростильбен, пицеатаннол, пиносильван, эллагиктаннин, пуникалагин, касталагин, вескалагин, касталин, казуариктин, грандинин, пуникалины, робурин, теллимаграндин, терфлавин, галлотаннин, проантоцианидин, полифлавоноид, пирокатехольное соединение, флаволан, салициловую кислоту, ваниллин, галловую кислоту, эллаговую кислоту, дигалловую кислоту, кофеиновую кислоту, хлорогеновую кислоту, феруловую кислоту, кумарин, тирозол, гидрокситирозол, олеокантол, олеуропеин, капсаицин, гингерол, мальтодекстрин, декстрозу, стерубин, азалеин, галангин, госсипетин, гиперозид, икариин, изокверцетин, изорамнетин, кемпферид, кемпферитрин, морин, мирицитрин, кверцитрин, пахиподол, рамназин, робинии, робинозу, спиреозид, спиренозид, троксерутин, вогонин, стерубин, понцирин, эупафолин, апигенин.
11. Препарат по п. 1, где крахмал выбран из группы, состоящей из полимерного углевода или полисахарида, включающего глюкопиранозу, амилозу, амилопектин, гликоген, арабиноксилан, целлюлозу, хитин, пектин, кислотные полисахариды.
12. Препарат по п. 1, где полифенол адаптирован, при введении препарата индивиду, для контроля отрицательных эффектов гипергликемии посредством одного или более чем одного из следующих способов: ингибирование провоспалительного TNF-α (фактор некроза опухолей-альфа), ингибирование альфа-амилазы, ингибирование глюкозидазы, ингибирование транспорта glut 2 в жировую ткань, стимуляция транспорта glut 4 в мышечную ткань и/или стимуляция образования митохондрий в мышечной ткани.
13. Препарат по п. 1, где данный препарат, при введении индивиду, ингибирует гликемическое влияние сахаров посредством одного или более чем одного из следующих способов: прямое ингибирование фермента альфа-амилазы, прямое ингибирование фермента глюкозидазы, ингибирование и буферизация кислот желудка.
14. Препарат по п. 1, где данный препарат, при введении индивиду, нуждающемуся в этом, предупреждает образование полости во рту посредством предупреждения или уменьшения уровня кислот, разрушающих эмаль, от побочного продукта амилазной активности.
15. Препарат по п. 1, где полифенол готовят для ингибирования амилазной активности в полости рта при введении препарата индивиду, нуждающемуся в этом.
16. Препарат по п. 1, который, при введении пациенту, нуждающемуся в этом, приводит к улучшенному препарату сахара, который будет вызывать потерю массы тела или предупреждать набор веса через прямое взаимодействие уменьшения накопления жира посредством ингибирования пути glut 2 жировых тканей и прямой стимуляции повышенного потребления энергии/углеводов посредством активации пути glut 4.
17. Препарат по п. 1, где полифенол представляет собой гесперитин или гесперидин, и крахмал представляет собой инулин.
18. Препарат по п. 1, где полифенол представляет собой галловую кислоту, и крахмал представляет собой арабиноксилан.
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CN111096986A (zh) * | 2019-12-31 | 2020-05-05 | 江门民康生物科技研究有限公司 | 一种以神秘果果核为原料的提取物及其在制备具有降血糖作用的药物或保健品中的应用 |
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US20030004211A1 (en) * | 2001-05-25 | 2003-01-02 | Frank Corsini | Carbohydrate modifying agent and drinks containing the modifying agent |
US20030017219A1 (en) * | 2001-05-25 | 2003-01-23 | Frank Corsini | Carbohydrate modifying agent and drinks containing the modifying agent |
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CA3051413A1 (en) | 2018-05-24 |
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EP3541207A4 (en) | 2020-05-20 |
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