RU2017109814A3 - - Google Patents

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Publication number
RU2017109814A3
RU2017109814A3 RU2017109814A RU2017109814A RU2017109814A3 RU 2017109814 A3 RU2017109814 A3 RU 2017109814A3 RU 2017109814 A RU2017109814 A RU 2017109814A RU 2017109814 A RU2017109814 A RU 2017109814A RU 2017109814 A3 RU2017109814 A3 RU 2017109814A3
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RU
Russia
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RU2017109814A
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RU2017109814A (ru
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Publication of RU2017109814A publication Critical patent/RU2017109814A/ru
Publication of RU2017109814A3 publication Critical patent/RU2017109814A3/ru

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
RU2017109814A 2011-11-10 2012-11-09 Кристаллическая 7-{ (3s,4s)-3-[(циклопропиламино)метил]-4-фторпирролидин-1-ил} -6-фтор-1-(2-фторэтил)-8-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновая кислота RU2017109814A (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2011-246209 2011-11-10
JP2011246209 2011-11-10
JP2012-071739 2012-03-27
JP2012071739 2012-03-27

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
RU2014123567A Division RU2615509C2 (ru) 2011-11-10 2012-11-09 Кристаллическая 7-{ (3s,4s)-3-[(циклопропиламино)метил]-4-фторпирролидин-1-ил} -6-фтор-1-(2-фторэтил)-8-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновая кислота

Publications (2)

Publication Number Publication Date
RU2017109814A RU2017109814A (ru) 2019-01-23
RU2017109814A3 true RU2017109814A3 (ru) 2020-04-08

Family

ID=48289529

Family Applications (2)

Application Number Title Priority Date Filing Date
RU2017109814A RU2017109814A (ru) 2011-11-10 2012-11-09 Кристаллическая 7-{ (3s,4s)-3-[(циклопропиламино)метил]-4-фторпирролидин-1-ил} -6-фтор-1-(2-фторэтил)-8-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновая кислота
RU2014123567A RU2615509C2 (ru) 2011-11-10 2012-11-09 Кристаллическая 7-{ (3s,4s)-3-[(циклопропиламино)метил]-4-фторпирролидин-1-ил} -6-фтор-1-(2-фторэтил)-8-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновая кислота

Family Applications After (1)

Application Number Title Priority Date Filing Date
RU2014123567A RU2615509C2 (ru) 2011-11-10 2012-11-09 Кристаллическая 7-{ (3s,4s)-3-[(циклопропиламино)метил]-4-фторпирролидин-1-ил} -6-фтор-1-(2-фторэтил)-8-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновая кислота

Country Status (16)

Country Link
US (3) US9090587B2 (ru)
EP (2) EP3112359B1 (ru)
JP (4) JP5871948B2 (ru)
KR (2) KR102162208B1 (ru)
CN (2) CN104945375B (ru)
AU (1) AU2016273899B2 (ru)
BR (1) BR112014010765B1 (ru)
CA (1) CA2855022C (ru)
ES (2) ES2747303T3 (ru)
IN (1) IN2014DN03277A (ru)
NZ (1) NZ623808A (ru)
RU (2) RU2017109814A (ru)
SA (1) SA112330992B1 (ru)
SG (2) SG10201608167UA (ru)
TW (1) TWI547492B (ru)
WO (1) WO2013069297A1 (ru)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SA112330992B1 (ar) * 2011-11-10 2015-09-13 كيورين فارماسوتيكال كو.، ليمتد صورة متبلرة من 7-{(s4، s3)-3-[(سيكلو بروبيل أمينو) ميثيل]-4-فلورو بيروليدين-1-يل}-6-فلورو-1-(2-فلورو إيثيل)- 8-ميثوكسي-4-أوكسو-1، 4-داي هيدرو كينولين-3- حمض كربوكسيلي
CN105338982B (zh) * 2013-04-25 2017-10-10 杏林制药株式会社 固体药用组合物
JP5700740B1 (ja) * 2013-04-25 2015-04-15 杏林製薬株式会社 固形医薬組成物
WO2014174848A1 (ja) * 2013-04-25 2014-10-30 杏林製薬株式会社 錠剤
GB201402071D0 (en) * 2014-02-07 2014-03-26 Galapagos Nv Novel salts and pharmaceutical compositions thereof for the treatment of inflammatory disorders
WO2016063542A1 (ja) * 2014-10-23 2016-04-28 杏林製薬株式会社 固形医薬組成物
EP3210608A4 (en) * 2014-10-23 2018-06-20 Kyorin Pharmaceutical Co., Ltd. Solid pharmaceutical composition
CN113975277A (zh) 2015-03-13 2022-01-28 杏林制药株式会社 呼吸器官感染治疗剂
WO2016195014A1 (ja) * 2015-06-02 2016-12-08 杏林製薬株式会社 水性液剤
EP3305295A4 (en) * 2015-06-02 2019-02-20 Kyorin Pharmaceutical Co., Ltd. AQUEOUS MEDICINE
EP3305296A4 (en) * 2015-06-02 2019-02-13 Kyorin Pharmaceutical Co., Ltd. AQUEOUS LIQUID FORMULATION
TWI818910B (zh) 2017-06-16 2023-10-21 日商杏林製藥股份有限公司 吸入性肺炎、肺化膿症或肺膿瘍之治療劑
EA202090066A1 (ru) 2018-03-30 2020-04-15 Керин Фармасьютикал Ко., Лтд. Терапевтическое средство для лечения аспирационной пневмонии, легочного нагноения или абсцесса легких

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA944369B (en) * 1993-08-27 1995-02-13 Hokuriku Seuyaku Co Ltd 5-amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid derivative
CN1158846A (zh) * 1995-05-09 1997-09-10 昆山市康壮达兽药厂 盐酸氟哌酸的合成工艺
US20030119060A1 (en) * 2001-08-10 2003-06-26 Desrosiers Peter J. Apparatuses and methods for creating and testing pre-formulations and systems for same
WO2003076428A1 (fr) * 2002-03-08 2003-09-18 Daiichi Pharmaceutical Co., Ltd. Derive d'acide quinolone-carboxylique
PT1666477E (pt) * 2003-09-10 2013-08-28 Kyorin Seiyaku Kk Derivado de 7-(4-substituído-3-ciclopropilaminometil-1- pirrolidinil) quinolonecarboxílico
CN101003540A (zh) * 2006-01-18 2007-07-25 广州白云山制药股份有限公司广州白云山制药总厂 一种抗感染化合物和用途
SA112330992B1 (ar) * 2011-11-10 2015-09-13 كيورين فارماسوتيكال كو.، ليمتد صورة متبلرة من 7-{(s4، s3)-3-[(سيكلو بروبيل أمينو) ميثيل]-4-فلورو بيروليدين-1-يل}-6-فلورو-1-(2-فلورو إيثيل)- 8-ميثوكسي-4-أوكسو-1، 4-داي هيدرو كينولين-3- حمض كربوكسيلي

Also Published As

Publication number Publication date
TWI547492B (zh) 2016-09-01
CN103930414A (zh) 2014-07-16
KR20140098074A (ko) 2014-08-07
SA112330992B1 (ar) 2015-09-13
KR20190065456A (ko) 2019-06-11
EP3112359A1 (en) 2017-01-04
US9090587B2 (en) 2015-07-28
US20140288310A1 (en) 2014-09-25
SG11201401817TA (en) 2014-08-28
EP2778159A1 (en) 2014-09-17
RU2014123567A (ru) 2015-12-20
CA2855022C (en) 2019-05-07
AU2012337206B2 (en) 2016-09-15
EP2778159A4 (en) 2015-06-03
AU2012337206A8 (en) 2016-09-22
JP6349435B2 (ja) 2018-06-27
JP2017160243A (ja) 2017-09-14
JP5871948B2 (ja) 2016-03-01
TW201332991A (zh) 2013-08-16
KR102162208B1 (ko) 2020-10-06
BR112014010765B1 (pt) 2020-07-14
CA2855022A1 (en) 2013-05-16
RU2615509C2 (ru) 2017-04-05
USRE47785E1 (en) 2019-12-31
US9328089B2 (en) 2016-05-03
JP6514069B2 (ja) 2019-05-15
JP2018158949A (ja) 2018-10-11
JPWO2013069297A1 (ja) 2015-04-02
SG10201608167UA (en) 2016-11-29
WO2013069297A1 (ja) 2013-05-16
EP3112359B1 (en) 2019-08-21
JP2016027045A (ja) 2016-02-18
ES2621664T3 (es) 2017-07-04
CN104945375A (zh) 2015-09-30
EP2778159B1 (en) 2017-03-01
JP6818719B2 (ja) 2021-01-20
AU2016273899A1 (en) 2017-01-12
AU2012337206A1 (en) 2014-05-22
NZ623808A (en) 2015-07-31
RU2017109814A (ru) 2019-01-23
US20150284361A1 (en) 2015-10-08
CN104945375B (zh) 2017-07-04
IN2014DN03277A (ru) 2015-05-22
AU2016273899B2 (en) 2017-07-27
ES2747303T3 (es) 2020-03-10
CN103930414B (zh) 2016-01-20
BR112014010765A2 (pt) 2017-06-13

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