RU2007148225A - Глюкокортикоидные миметики, способы их получения, фармацевтические композиции и их применение - Google Patents

Глюкокортикоидные миметики, способы их получения, фармацевтические композиции и их применение Download PDF

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RU2007148225A
RU2007148225A RU2007148225/04A RU2007148225A RU2007148225A RU 2007148225 A RU2007148225 A RU 2007148225A RU 2007148225/04 A RU2007148225/04 A RU 2007148225/04A RU 2007148225 A RU2007148225 A RU 2007148225A RU 2007148225 A RU2007148225 A RU 2007148225A
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Russia
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indazol
trifluoro
fluorophenyl
propan
phenyl
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RU2007148225/04A
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English (en)
Russian (ru)
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Инго Андреас МУГГЕ (US)
Инго Андреас МУГГЕ
Майкл Джейсон БЕРК (US)
Майкл Джейсон БЕРК
Марк Стивен РАЛФ (US)
Марк Стивен РАЛФ
Дейвид С. ТОМСОН (US)
Дейвид С. ТОМСОН
Абедельхаким ХАММАЧ (US)
Абедельхаким ХАММАЧ
Дженнифер А. КОВАЛЬСКИ (US)
Дженнифер А. Ковальски
Йерг Мартин БЕНТЦИН (US)
Йерг Мартин БЕНТЦИН
Original Assignee
БЕРИНГЕР ИНГЕЛЬХАЙМ ИНТЕРНАЦИОНАЛЬ ГмбХ (DE)
Берингер Ингельхайм Интернациональ Гмбх
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Publication of RU2007148225A publication Critical patent/RU2007148225A/ru

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Organic Chemistry (AREA)
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  • Medicinal Chemistry (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Otolaryngology (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Child & Adolescent Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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RU2007148225/04A 2005-06-10 2006-06-08 Глюкокортикоидные миметики, способы их получения, фармацевтические композиции и их применение RU2007148225A (ru)

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Application Number Priority Date Filing Date Title
US68941205P 2005-06-10 2005-06-10
US60/689,412 2005-06-10

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RU2007148225A true RU2007148225A (ru) 2009-07-20

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US (1) US7622594B2 (enExample)
EP (1) EP1893588A1 (enExample)
JP (1) JP2008543780A (enExample)
KR (1) KR20080027828A (enExample)
CN (1) CN101193869B (enExample)
AR (1) AR058006A1 (enExample)
AU (1) AU2006257861A1 (enExample)
BR (1) BRPI0611620A2 (enExample)
CA (1) CA2610588A1 (enExample)
IL (1) IL187976A0 (enExample)
MX (1) MX2007014811A (enExample)
NZ (1) NZ564696A (enExample)
PE (1) PE20070112A1 (enExample)
RU (1) RU2007148225A (enExample)
TW (1) TW200716573A (enExample)
WO (1) WO2006135826A1 (enExample)
ZA (1) ZA200709430B (enExample)

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KR20050036982A (ko) * 2002-08-29 2005-04-20 베링거 인겔하임 파마슈티칼즈, 인코포레이티드 염증, 알러지 및 증식성 질환의 치료에 글루코코르티코이드모사체로 사용하기 위한 3-(설폰아미도에틸)-인돌 유도체
UY28526A1 (es) * 2003-09-24 2005-04-29 Boehringer Ingelheim Pharma Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos
US7795272B2 (en) 2004-03-13 2010-09-14 Boehringer Ingelheim Pharmaceutical, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
ES2326907T3 (es) * 2004-12-27 2009-10-21 Boehringer Ingelheim Pharmaceuticals Inc. Mimeticos de glucocorticoides, metodos para su preparacion, composiciones farmaceuticas y su uso.
EP2061767B1 (de) 2006-08-08 2014-12-17 Sanofi Arylaminoaryl-alkyl-substituierte Imidazolidin-2,4-dione, Verfahren zu ihrer Herstellung, diese Verbindungen enthaltende Arzneimittel und ihre Verwendung
EP2099767A1 (en) * 2006-11-01 2009-09-16 Brystol-Myers Squibb Company Modulators of glucocorticoid receptor, ap-1, and/or nf- b activity and use thereof
TW200829578A (en) 2006-11-23 2008-07-16 Astrazeneca Ab Chemical compounds 537
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JO2754B1 (en) * 2006-12-21 2014-03-15 استرازينكا ايه بي Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders
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US7622594B2 (en) 2009-11-24
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CA2610588A1 (en) 2006-12-21
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AU2006257861A1 (en) 2006-12-21
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