JP2008543780A - グルココルチコイド模倣薬、それらの製造方法、医薬組成物及びそれらの使用 - Google Patents

グルココルチコイド模倣薬、それらの製造方法、医薬組成物及びそれらの使用 Download PDF

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JP2008543780A
JP2008543780A JP2008515997A JP2008515997A JP2008543780A JP 2008543780 A JP2008543780 A JP 2008543780A JP 2008515997 A JP2008515997 A JP 2008515997A JP 2008515997 A JP2008515997 A JP 2008515997A JP 2008543780 A JP2008543780 A JP 2008543780A
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indazol
trifluoro
fluorophenyl
propan
phenyl
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JP2008543780A5 (enExample
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インゴ アンドレアス ムゲ
マイケル ジェイソン バーク
マーク スティーブン ラルフ
ディヴィッド エス トムソン
アブデルハキム ハムマック
ジェニファー エイ コワルスキー
ヨルグ マルティン ベンツィエン
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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  • Chemical & Material Sciences (AREA)
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  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
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  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Otolaryngology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
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  • Communicable Diseases (AREA)
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  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
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JP2008515997A 2005-06-10 2006-06-08 グルココルチコイド模倣薬、それらの製造方法、医薬組成物及びそれらの使用 Pending JP2008543780A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68941205P 2005-06-10 2005-06-10
PCT/US2006/022651 WO2006135826A1 (en) 2005-06-10 2006-06-08 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

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Publication Number Publication Date
JP2008543780A true JP2008543780A (ja) 2008-12-04
JP2008543780A5 JP2008543780A5 (enExample) 2009-08-13

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US (1) US7622594B2 (enExample)
EP (1) EP1893588A1 (enExample)
JP (1) JP2008543780A (enExample)
KR (1) KR20080027828A (enExample)
CN (1) CN101193869B (enExample)
AR (1) AR058006A1 (enExample)
AU (1) AU2006257861A1 (enExample)
BR (1) BRPI0611620A2 (enExample)
CA (1) CA2610588A1 (enExample)
IL (1) IL187976A0 (enExample)
MX (1) MX2007014811A (enExample)
NZ (1) NZ564696A (enExample)
PE (1) PE20070112A1 (enExample)
RU (1) RU2007148225A (enExample)
TW (1) TW200716573A (enExample)
WO (1) WO2006135826A1 (enExample)
ZA (1) ZA200709430B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023535279A (ja) * 2020-06-22 2023-08-17 コーセプト セラピューティクス， インコーポレイテッド ４級インダゾールグルココルチコイド受容体アンタゴニスト

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JP4324480B2 (ja) * 2002-03-26 2009-09-02 ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド グルココルチコイドミメティクス、その製法、医薬組成物、及び使用
NZ538932A (en) * 2002-08-29 2007-04-27 Boehringer Ingelheim Pharma 3-(sulfonamidoethyl)-indole derivatives for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative disease
UY28526A1 (es) 2003-09-24 2005-04-29 Boehringer Ingelheim Pharma Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos
US7795272B2 (en) 2004-03-13 2010-09-14 Boehringer Ingelheim Pharmaceutical, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
PE20060776A1 (es) 2004-12-27 2006-09-26 Boehringer Ingelheim Pharma Mimeticos de glucocorticoides, metodos para prepararlos y composiciones farmaceuticas
JP2010500300A (ja) 2006-08-08 2010-01-07 サノフィ−アベンティス アリールアミノアリール−アルキル−置換イミダゾリジン−２，４−ジオン、それらの製造法、それらの化合物を含有する薬剤、およびそれらの使用
JP2010508358A (ja) * 2006-11-01 2010-03-18 ブリストル−マイヤーズ スクイブ カンパニー グルココルチコイド受容体、ＡＰ−１、および／またはＮＦ−κＢ活性の調節剤、並びにその使用
TW200829578A (en) 2006-11-23 2008-07-16 Astrazeneca Ab Chemical compounds 537
MX2009005264A (es) 2006-12-06 2009-05-28 Boehringer Ingelheim Int Mimeticos de glucocorticoides, metodos para su fabricacion, composiciones farmaceuticas y usos de los mismos.
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