RU2007133655A - Замещенные бис-арильные и гетероарильные соединения в качестве селективных антагонистов 5нт2а - Google Patents

Замещенные бис-арильные и гетероарильные соединения в качестве селективных антагонистов 5нт2а Download PDF

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RU2007133655A
RU2007133655A RU2007133655/04A RU2007133655A RU2007133655A RU 2007133655 A RU2007133655 A RU 2007133655A RU 2007133655/04 A RU2007133655/04 A RU 2007133655/04A RU 2007133655 A RU2007133655 A RU 2007133655A RU 2007133655 A RU2007133655 A RU 2007133655A
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Russia
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fluoro
benzyl
indol
ylmethyl
phenyl
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RU2007133655/04A
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English (en)
Russian (ru)
Inventor
Дэвид Марк ФИНК (US)
Дэвид Марк ФИНК
Хелен Катерин СМИТ (GB)
Хелен Катерин СМИТ
Ричард Саймон ТОДД (GB)
Ричард Саймон Тодд
Пол Роберт ИСТВУД (ES)
Пол Роберт Иствуд
Хейзел ХАНТ (GB)
Хейзел ХАНТ
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Авентис Фармасьютикалз Инк. (Us)
Авентис Фармасьютикалз Инк.
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Publication of RU2007133655A publication Critical patent/RU2007133655A/ru

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    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C07D239/72—Quinazolines; Hydrogenated quinazolines
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    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
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    • C07D277/62—Benzothiazoles
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Organic Chemistry (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Psychiatry (AREA)
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  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
RU2007133655/04A 2005-02-10 2006-02-10 Замещенные бис-арильные и гетероарильные соединения в качестве селективных антагонистов 5нт2а RU2007133655A (ru)

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US65191105P 2005-02-10 2005-02-10
US60/651,911 2005-02-10

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RU2007133655A true RU2007133655A (ru) 2009-03-20

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US (1) US7625889B2 (OSRAM)
EP (1) EP1851199B1 (OSRAM)
JP (1) JP5419355B2 (OSRAM)
KR (1) KR20070107037A (OSRAM)
CN (1) CN101115717A (OSRAM)
AR (1) AR052903A1 (OSRAM)
AU (1) AU2006213634A1 (OSRAM)
BR (1) BRPI0606740A2 (OSRAM)
CA (1) CA2598429A1 (OSRAM)
CR (1) CR9260A (OSRAM)
DO (1) DOP2006000032A (OSRAM)
GT (1) GT200600042A (OSRAM)
IL (1) IL185173A0 (OSRAM)
MA (1) MA29289B1 (OSRAM)
MX (1) MX2007008606A (OSRAM)
NO (1) NO20074583L (OSRAM)
PA (1) PA8662501A1 (OSRAM)
PE (1) PE20061088A1 (OSRAM)
RU (1) RU2007133655A (OSRAM)
TN (1) TNSN07272A1 (OSRAM)
TW (1) TW200640859A (OSRAM)
UY (1) UY29372A1 (OSRAM)
WO (1) WO2006086705A1 (OSRAM)

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