RU2006146042A - Диаминные агонисты 2-адренергических рецепторов - Google Patents

Диаминные агонисты 2-адренергических рецепторов Download PDF

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Publication number
RU2006146042A
RU2006146042A RU2006146042/04A RU2006146042A RU2006146042A RU 2006146042 A RU2006146042 A RU 2006146042A RU 2006146042/04 A RU2006146042/04 A RU 2006146042/04A RU 2006146042 A RU2006146042 A RU 2006146042A RU 2006146042 A RU2006146042 A RU 2006146042A
Authority
RU
Russia
Prior art keywords
compound according
compound
hydrogen atom
hydroxy
formula
Prior art date
Application number
RU2006146042/04A
Other languages
English (en)
Russian (ru)
Inventor
Мартин С. ЛИНСЕЛЛ (US)
Мартин С. Линселл
Original Assignee
Тереванс
Тереванс, Инк.
Инк. (US)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Тереванс, Тереванс, Инк., Инк. (US) filed Critical Тереванс
Publication of RU2006146042A publication Critical patent/RU2006146042A/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/24—Oxygen atoms attached in position 8
    • C07D215/26—Alcohols; Ethers thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Quinoline Compounds (AREA)
RU2006146042/04A 2004-06-03 2005-06-02 Диаминные агонисты 2-адренергических рецепторов RU2006146042A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US57656004P 2004-06-03 2004-06-03
US60/576,560 2004-06-03

Publications (1)

Publication Number Publication Date
RU2006146042A true RU2006146042A (ru) 2008-07-20

Family

ID=35115813

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2006146042/04A RU2006146042A (ru) 2004-06-03 2005-06-02 Диаминные агонисты 2-адренергических рецепторов

Country Status (14)

Country Link
US (2) US20080039495A1 (enExample)
EP (1) EP1751086A2 (enExample)
JP (1) JP2008501705A (enExample)
CN (1) CN1984876A (enExample)
AU (1) AU2005252226A1 (enExample)
BR (1) BRPI0511695A (enExample)
CA (1) CA2569395A1 (enExample)
IL (1) IL179631A0 (enExample)
MA (1) MA28902B1 (enExample)
MX (1) MXPA06013916A (enExample)
NO (1) NO20066016L (enExample)
RU (1) RU2006146042A (enExample)
WO (1) WO2005121065A2 (enExample)
ZA (1) ZA200610835B (enExample)

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Also Published As

Publication number Publication date
WO2005121065A3 (en) 2006-02-09
AU2005252226A1 (en) 2005-12-22
IL179631A0 (en) 2007-05-15
US20050272769A1 (en) 2005-12-08
JP2008501705A (ja) 2008-01-24
US7402673B2 (en) 2008-07-22
WO2005121065A2 (en) 2005-12-22
NO20066016L (no) 2007-02-27
CA2569395A1 (en) 2005-12-22
EP1751086A2 (en) 2007-02-14
US20080039495A1 (en) 2008-02-14
MXPA06013916A (es) 2007-03-07
BRPI0511695A (pt) 2008-01-08
CN1984876A (zh) 2007-06-20
MA28902B1 (fr) 2007-10-01
ZA200610835B (en) 2007-11-28

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