ZA200610835B - Diamine ß2 adrenergic receptor agonists - Google Patents

Diamine ß2 adrenergic receptor agonists

Info

Publication number
ZA200610835B
ZA200610835B ZA200610835A ZA200610835A ZA200610835B ZA 200610835 B ZA200610835 B ZA 200610835B ZA 200610835 A ZA200610835 A ZA 200610835A ZA 200610835 A ZA200610835 A ZA 200610835A ZA 200610835 B ZA200610835 B ZA 200610835B
Authority
ZA
South Africa
Prior art keywords
diamine
receptor agonists
adrenergic receptor
adrenergic
agonists
Prior art date
Application number
ZA200610835A
Other languages
English (en)
Inventor
Martin S Linsell
Original Assignee
Theravance Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theravance Inc filed Critical Theravance Inc
Publication of ZA200610835B publication Critical patent/ZA200610835B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/24—Oxygen atoms attached in position 8
    • C07D215/26—Alcohols; Ethers thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Quinoline Compounds (AREA)
ZA200610835A 2004-06-03 2006-12-21 Diamine ß2 adrenergic receptor agonists ZA200610835B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57656004P 2004-06-03 2004-06-03

Publications (1)

Publication Number Publication Date
ZA200610835B true ZA200610835B (en) 2007-11-28

Family

ID=35115813

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200610835A ZA200610835B (en) 2004-06-03 2006-12-21 Diamine ß2 adrenergic receptor agonists

Country Status (14)

Country Link
US (2) US7402673B2 (enExample)
EP (1) EP1751086A2 (enExample)
JP (1) JP2008501705A (enExample)
CN (1) CN1984876A (enExample)
AU (1) AU2005252226A1 (enExample)
BR (1) BRPI0511695A (enExample)
CA (1) CA2569395A1 (enExample)
IL (1) IL179631A0 (enExample)
MA (1) MA28902B1 (enExample)
MX (1) MXPA06013916A (enExample)
NO (1) NO20066016L (enExample)
RU (1) RU2006146042A (enExample)
WO (1) WO2005121065A2 (enExample)
ZA (1) ZA200610835B (enExample)

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CN102272104B (zh) 2008-12-30 2014-07-09 帕尔马根治疗(炎症)有限公司 用于治疗呼吸疾病的磺酰胺化合物
EP2228368A1 (en) 2009-03-12 2010-09-15 Almirall, S.A. Process for manufacturing 5-(2-{[6-(2,2-difluoro-2-phenylethoxy) hexyl]amino}-1-hydroxyethyl)-8-hydroxyquinolin-2(1H)-one
WO2010150014A1 (en) 2009-06-24 2010-12-29 Pulmagen Therapeutics (Inflammation) Limited 5r- 5 -deuterated glitazones for respiratory disease treatment
GB0918923D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Aminothiazole derivatives
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WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
WO2011098746A1 (en) 2010-02-09 2011-08-18 Pulmagen Therapeutics (Inflammation) Limited Crystalline acid addition salts of ( 5r) -enanti0mer of pioglitazone
GB201002243D0 (en) 2010-02-10 2010-03-31 Argenta Therapeutics Ltd Respiratory disease treatment
GB201002224D0 (en) 2010-02-10 2010-03-31 Argenta Therapeutics Ltd Respiratory disease treatment
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
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EA201391230A1 (ru) 2011-02-25 2014-01-30 АйАрЭм ЭлЭлСи Соединения и композиции в качестве ингибиторов trk
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Also Published As

Publication number Publication date
MXPA06013916A (es) 2007-03-07
EP1751086A2 (en) 2007-02-14
US20050272769A1 (en) 2005-12-08
IL179631A0 (en) 2007-05-15
WO2005121065A3 (en) 2006-02-09
WO2005121065A2 (en) 2005-12-22
US20080039495A1 (en) 2008-02-14
CN1984876A (zh) 2007-06-20
RU2006146042A (ru) 2008-07-20
BRPI0511695A (pt) 2008-01-08
AU2005252226A1 (en) 2005-12-22
CA2569395A1 (en) 2005-12-22
NO20066016L (no) 2007-02-27
MA28902B1 (fr) 2007-10-01
JP2008501705A (ja) 2008-01-24
US7402673B2 (en) 2008-07-22

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