RS64591B1 - Derivati bipirazola kao inhibitori jak - Google Patents

Derivati bipirazola kao inhibitori jak

Info

Publication number
RS64591B1
RS64591B1 RS20230782A RSP20230782A RS64591B1 RS 64591 B1 RS64591 B1 RS 64591B1 RS 20230782 A RS20230782 A RS 20230782A RS P20230782 A RSP20230782 A RS P20230782A RS 64591 B1 RS64591 B1 RS 64591B1
Authority
RS
Serbia
Prior art keywords
jak inhibitors
bipyrazole derivatives
bipyrazole
derivatives
jak
Prior art date
Application number
RS20230782A
Other languages
English (en)
Inventor
Yun-Long Li
Jincong Zhuo
Ding-Quan Qian
Song Mei
Ganfeng Cao
Yongchun Pan
Qun Li
Zhongjiang Jia
Original Assignee
Incyte Holdings Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Holdings Corp filed Critical Incyte Holdings Corp
Publication of RS64591B1 publication Critical patent/RS64591B1/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
RS20230782A 2013-05-17 2014-05-16 Derivati bipirazola kao inhibitori jak RS64591B1 (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361824683P 2013-05-17 2013-05-17
EP20201593.9A EP3786162B1 (en) 2013-05-17 2014-05-16 Bipyrazole derivatives as jak inhibitors

Publications (1)

Publication Number Publication Date
RS64591B1 true RS64591B1 (sr) 2023-10-31

Family

ID=50983151

Family Applications (4)

Application Number Title Priority Date Filing Date
RS20190315A RS58743B1 (sr) 2013-05-17 2014-05-16 Soli bipirazola kao inhibitori jak
RS20210074A RS61482B1 (sr) 2013-05-17 2014-05-16 Derivati bipirazola kao inhibitori jak
RS20230782A RS64591B1 (sr) 2013-05-17 2014-05-16 Derivati bipirazola kao inhibitori jak
RS20170526A RS56012B1 (sr) 2013-05-17 2014-05-16 Derivati bipirazola kao inhibitori jak

Family Applications Before (2)

Application Number Title Priority Date Filing Date
RS20190315A RS58743B1 (sr) 2013-05-17 2014-05-16 Soli bipirazola kao inhibitori jak
RS20210074A RS61482B1 (sr) 2013-05-17 2014-05-16 Derivati bipirazola kao inhibitori jak

Family Applications After (1)

Application Number Title Priority Date Filing Date
RS20170526A RS56012B1 (sr) 2013-05-17 2014-05-16 Derivati bipirazola kao inhibitori jak

Country Status (35)

Country Link
US (6) US9382231B2 (sr)
EP (5) EP3527263B1 (sr)
JP (4) JP6415543B2 (sr)
KR (3) KR102442747B1 (sr)
CN (2) CN105452239B (sr)
AR (2) AR096330A1 (sr)
AU (5) AU2014265279B2 (sr)
BR (1) BR112015028501B8 (sr)
CA (1) CA2911536C (sr)
CL (1) CL2015003355A1 (sr)
CR (2) CR20190156A (sr)
CY (3) CY1119105T1 (sr)
DK (3) DK3527263T3 (sr)
EA (2) EA039660B1 (sr)
ES (4) ES2626793T3 (sr)
FI (1) FI3786162T3 (sr)
HK (2) HK1221466A1 (sr)
HR (4) HRP20231048T1 (sr)
HU (4) HUE063817T2 (sr)
IL (4) IL242453B (sr)
LT (4) LT3786162T (sr)
ME (2) ME02763B (sr)
MX (2) MX2020004506A (sr)
MY (1) MY174788A (sr)
PE (2) PE20160126A1 (sr)
PH (2) PH12015502563B1 (sr)
PL (4) PL3786162T3 (sr)
PT (4) PT3231801T (sr)
RS (4) RS58743B1 (sr)
SG (2) SG10201709469SA (sr)
SI (4) SI3231801T1 (sr)
TR (1) TR201905814T4 (sr)
TW (2) TWI719401B (sr)
UA (1) UA117830C2 (sr)
WO (1) WO2014186706A1 (sr)

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