RS56539B1 - Policiklična-karbamoilpiridonska jedinjenja i njihova upotreba za lečenje hiv infekcija - Google Patents

Policiklična-karbamoilpiridonska jedinjenja i njihova upotreba za lečenje hiv infekcija

Info

Publication number
RS56539B1
RS56539B1 RS20171143A RSP20171143A RS56539B1 RS 56539 B1 RS56539 B1 RS 56539B1 RS 20171143 A RS20171143 A RS 20171143A RS P20171143 A RSP20171143 A RS P20171143A RS 56539 B1 RS56539 B1 RS 56539B1
Authority
RS
Serbia
Prior art keywords
compound
mmol
pharmaceutically acceptable
concentrated
ethyl acetate
Prior art date
Application number
RS20171143A
Other languages
English (en)
Serbian (sr)
Inventor
Mingzhe Ji
Teresa Alejandra Trejo Martin
Manoj C Desai
Haolun Jin
Hyung Jung Pyun
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of RS56539B1 publication Critical patent/RS56539B1/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
RS20171143A 2013-07-12 2014-07-11 Policiklična-karbamoilpiridonska jedinjenja i njihova upotreba za lečenje hiv infekcija RS56539B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361845807P 2013-07-12 2013-07-12
EP14745053.0A EP3019499B1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections
PCT/US2014/046415 WO2015006733A1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections

Publications (1)

Publication Number Publication Date
RS56539B1 true RS56539B1 (sr) 2018-02-28

Family

ID=51257630

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20171143A RS56539B1 (sr) 2013-07-12 2014-07-11 Policiklična-karbamoilpiridonska jedinjenja i njihova upotreba za lečenje hiv infekcija

Country Status (18)

Country Link
US (6) US9458159B2 (en:Method)
EP (2) EP3252053B1 (en:Method)
JP (1) JP6411492B2 (en:Method)
AU (3) AU2014286995B2 (en:Method)
CA (1) CA2918055C (en:Method)
CY (1) CY1119545T1 (en:Method)
DK (1) DK3019499T3 (en:Method)
ES (2) ES2647216T3 (en:Method)
HR (1) HRP20171807T1 (en:Method)
HU (1) HUE037343T2 (en:Method)
LT (1) LT3019499T (en:Method)
NO (1) NO2865735T3 (en:Method)
PL (1) PL3019499T3 (en:Method)
PT (1) PT3019499T (en:Method)
RS (1) RS56539B1 (en:Method)
SI (2) SI3019499T1 (en:Method)
SM (1) SMT201700525T1 (en:Method)
WO (1) WO2015006733A1 (en:Method)

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RS56540B1 (sr) * 2013-07-12 2018-02-28 Gilead Sciences Inc Policiklična karbamoilpiridonska jedinjenja i njihova upotreba za lečenje hiv infekcija
NO2865735T3 (en:Method) * 2013-07-12 2018-07-21
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EP4222152A1 (en) * 2020-09-30 2023-08-09 Gilead Sciences, Inc. Bridged tricyclic carbamoylpyridone compounds and uses thereof
JP7591155B2 (ja) 2021-01-19 2024-11-27 ギリアード サイエンシーズ， インコーポレイテッド 置換ピリドトリアジン化合物及びその使用
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