RS50396B - Mezoprogestini (progesteron receptor modulatori) kao komponente kompozicija za terapiju zamene hormona (hrt) - Google Patents

Mezoprogestini (progesteron receptor modulatori) kao komponente kompozicija za terapiju zamene hormona (hrt)

Info

Publication number
RS50396B
RS50396B YUP-141/02A YUP14102A RS50396B RS 50396 B RS50396 B RS 50396B YU P14102 A YUP14102 A YU P14102A RS 50396 B RS50396 B RS 50396B
Authority
RS
Serbia
Prior art keywords
hrt
replacement therapy
hormone replacement
mesoprogestins
compositions
Prior art date
Application number
YUP-141/02A
Other languages
English (en)
Inventor
Walter Elger
Gerd SCHUBERT
Kristof Chwalisz
Original Assignee
Bayer Schering Pharma Aktiengesellschaft,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Aktiengesellschaft, filed Critical Bayer Schering Pharma Aktiengesellschaft,
Publication of YU14102A publication Critical patent/YU14102A/sh
Publication of RS50396B publication Critical patent/RS50396B/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34—Gestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Upotreba mezoprogestina odabranog od grupe koja se sastoji od[4-[17ß-Metoksi-17ß -(metoksimetil)-3-oksoestra-4,9-dien-11ß-il]benzaldehid-(1E)-oksim] (J867),[4-[17ß-Hidroksi-17ß -(metoksimetil)-3-oksoestra-4,9-dien-11ß-il]benzaldehid-(1 E)-oksim] (912) i [4-[17ß -Metoksi-17ß -(metoksimetil)-3-oksoestra-4,9-dien-11ß -il]benzaldehid-(1E)-[0-(etilamino)karbonil]oksim] (J956) kao farmaceutske komponente za proizvodnju medikamenta za terapiju zamene hormona (HRT). Prijava sadrži još 5 zavisnih zahteva
YUP-141/02A 1999-08-31 2000-08-31 Mezoprogestini (progesteron receptor modulatori) kao komponente kompozicija za terapiju zamene hormona (hrt) RS50396B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US38614099A 1999-08-31 1999-08-31

Publications (2)

Publication Number Publication Date
YU14102A YU14102A (sh) 2006-01-16
RS50396B true RS50396B (sr) 2009-12-31

Family

ID=23524333

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-141/02A RS50396B (sr) 1999-08-31 2000-08-31 Mezoprogestini (progesteron receptor modulatori) kao komponente kompozicija za terapiju zamene hormona (hrt)

Country Status (33)

Country Link
EP (1) EP1605924B1 (sr)
JP (1) JP2003513908A (sr)
KR (1) KR100729311B1 (sr)
CN (1) CN1454088A (sr)
AR (1) AR025456A1 (sr)
AT (1) ATE413168T1 (sr)
AU (1) AU781836B2 (sr)
BG (1) BG65846B1 (sr)
BR (1) BR0013710A (sr)
CA (1) CA2383659C (sr)
CO (1) CO5200773A1 (sr)
CZ (1) CZ301412B6 (sr)
DE (1) DE60040764D1 (sr)
EA (1) EA007840B1 (sr)
EE (1) EE200200102A (sr)
ES (1) ES2316402T3 (sr)
HR (1) HRP20020266A2 (sr)
HU (1) HUP0202460A3 (sr)
IL (2) IL148417A0 (sr)
LT (1) LT5011B (sr)
LV (1) LV12942B (sr)
MX (1) MXPA02002190A (sr)
NO (1) NO20021000L (sr)
NZ (1) NZ517469A (sr)
PE (1) PE20010581A1 (sr)
PL (1) PL198798B1 (sr)
RO (1) RO122180B1 (sr)
RS (1) RS50396B (sr)
SI (1) SI20851B (sr)
SK (1) SK287121B6 (sr)
UA (1) UA75339C2 (sr)
WO (1) WO2001034126A2 (sr)
ZA (1) ZA200201621B (sr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1525215B1 (de) * 2002-08-02 2006-09-06 Schering Aktiengesellschaft Progesteronrezeptormodulatoren mit erhöhter antigonadotroper aktivität für die weibliche fertilitätskontrolle und hormonersatztherapie
DE10236405A1 (de) 2002-08-02 2004-02-19 Schering Ag Progesteronrezeptormodulatoren mit erhöhter antigonadotroper Aktivität für die weibliche Fertilitätskontrolle und Hormonersatztherapie
US20040097591A1 (en) * 2002-11-18 2004-05-20 Kristof Chwalisz Use of selective progesterone receptor modulators for the treatment of androgen deficiency
RU2611370C1 (ru) * 2016-01-12 2017-02-21 Общество с ограниченной ответственностью Медицинская Корпорация "РАНА" Применение препарата Лаеннек для уменьшения или устранения проявления менопаузальных симптомов (варианты)

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2054271A (en) 1932-05-17 1936-09-15 Schering Kahlbaum Ag Production of crystallized hormone esters
DE699310C (de) 1936-11-20 1940-11-27 Chemische Ind Ges Verfahren zur Herstellung von in 3-Stellung veresterten Verbindungen vom Typus des Oestradiols
US2225419A (en) 1937-03-01 1940-12-17 Schering Corp Process for the conversion of 17-cisalcohols of the cyclopentanopolyhydrophenanthrene series into the corresponding 17-trans-alcohols
US2611773A (en) 1951-08-21 1952-09-23 Upjohn Co Estradiol 17-cyclopenetanepropionate
US2990414A (en) 1957-03-26 1961-06-27 Syntex Sa 17-undecenoate of estradiol
US4729999A (en) * 1984-10-12 1988-03-08 Bcm Technologies Antiestrogen therapy for symptoms of estrogen deficiency
MX9301121A (es) * 1992-03-02 1993-09-01 Schering Ag Metodo y equipo para la contracepcion oral y regulacion de la menstruacion con estrogeno/progestina/aniprogestina.
TW366342B (en) * 1992-07-28 1999-08-11 Lilly Co Eli The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss
DE4225623C2 (de) * 1992-08-03 1994-06-30 Karl Hehl Verfahren zur Herstellung einer pulverförmigen Spritzgußmasse für die Herstellung von Porzellan und deren Verwendung
US5468736A (en) * 1993-02-25 1995-11-21 The Medical College Of Hampton Road Hormone replacement therapy
DE4332284C2 (de) 1993-09-20 1997-05-28 Jenapharm Gmbh 11-Benzaldoxim-17beta-methoxy-17alpha-methoxymethyl-estradien-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE4332283A1 (de) * 1993-09-20 1995-04-13 Jenapharm Gmbh Neue 11-Benzaldoximestradien-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
US5391557A (en) * 1993-10-15 1995-02-21 Eli Lilly And Company Methods for the treatment of peri-menopausal syndrome
JPH10507461A (ja) * 1994-10-24 1998-07-21 シエーリング アクチエンゲゼルシヤフト 必要に応じて女性の稔性を調節するための競合的プロゲステロン拮抗物質
DE19610635A1 (de) * 1996-03-11 1997-09-18 Schering Ag Sequentielle Estrogen/Progesteronantagonist-Kombination für die Hormonersatz-Therapie
TR199802705T2 (xx) * 1996-06-25 1999-03-22 Akzo Nobel N.V. Progestojen-anti-progestojen k�r�
WO1998005679A2 (en) * 1996-08-05 1998-02-12 Duke University Mixed agonists of the progesterone receptor and assays therefor
DE19809845A1 (de) * 1998-03-03 1999-09-09 Jenapharm Gmbh S-substituierte 11beta-Benzaldoxim-estra-4,9-dien-kohlensäurethiolester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Zubereitungen
EP1144396A2 (en) * 1999-01-14 2001-10-17 Bayer Corporation Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents

Also Published As

Publication number Publication date
KR20020027618A (ko) 2002-04-13
LT2002037A (en) 2002-11-25
EA007840B1 (ru) 2007-02-27
EE200200102A (et) 2003-04-15
ES2316402T3 (es) 2009-04-16
DE60040764D1 (de) 2008-12-18
AU3633201A (en) 2001-06-06
CN1454088A (zh) 2003-11-05
WO2001034126A2 (en) 2001-05-17
BG65846B1 (bg) 2010-03-31
HUP0202460A3 (en) 2004-04-28
AR025456A1 (es) 2002-11-27
SI20851A (sl) 2002-10-31
HRP20020266A2 (en) 2004-08-31
HUP0202460A2 (hu) 2002-12-28
MXPA02002190A (es) 2002-09-30
WO2001034126A3 (en) 2001-11-22
NO20021000D0 (no) 2002-02-28
CA2383659A1 (en) 2001-05-17
NZ517469A (en) 2004-01-30
NO20021000L (no) 2002-03-14
PL198798B1 (pl) 2008-07-31
BG106443A (bg) 2002-09-30
CZ2002706A3 (cs) 2002-10-16
SI20851B (sl) 2009-06-30
IL148417A (en) 2010-11-30
CA2383659C (en) 2009-02-10
PL353931A1 (en) 2003-12-15
EP1605924B1 (en) 2008-11-05
CO5200773A1 (es) 2002-09-27
LT5011B (lt) 2003-04-25
CZ301412B6 (cs) 2010-02-24
UA75339C2 (en) 2006-04-17
SK287121B6 (sk) 2009-12-07
ATE413168T1 (de) 2008-11-15
PE20010581A1 (es) 2001-06-04
EP1605924A2 (en) 2005-12-21
WO2001034126A9 (en) 2002-09-12
YU14102A (sh) 2006-01-16
RO122180B1 (ro) 2009-02-27
KR100729311B1 (ko) 2007-06-19
ZA200201621B (en) 2004-08-25
JP2003513908A (ja) 2003-04-15
SK2972002A3 (en) 2002-07-02
IL148417A0 (en) 2002-09-12
AU781836B2 (en) 2005-06-16
LV12942B (en) 2003-06-20
EA200200285A1 (ru) 2002-08-29
BR0013710A (pt) 2002-05-07

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