RS20060239A - Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics - Google Patents
Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeuticsInfo
- Publication number
- RS20060239A RS20060239A YUP-2006/0239A YUP20060239A RS20060239A RS 20060239 A RS20060239 A RS 20060239A YU P20060239 A YUP20060239 A YU P20060239A RS 20060239 A RS20060239 A RS 20060239A
- Authority
- RS
- Serbia
- Prior art keywords
- therapeutics
- preparation
- same
- arylalkylcarbamate
- derivatives
- Prior art date
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- C07C271/06—Esters of carbamic acids
- C07C271/40—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
- C07C271/42—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/44—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
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Abstract
Jedinjenje koje odgovara opštoj formuli (I) : u kome n predstavja ceo broj između 1 i 6: A je odabrano između jedne ili više grupa X, I i/ili Z; X predstavja eventualno supstituisanu alkilensku grupu Cl-2-; I predstavja eventualno supstituisanu C2-alkenilensku grupu ili grupu -C≡C-; Z predstavlja C3-7 cikloalkil, gde m predstavlja ceo broj od 1 do 5; P i q predstavljaju cele brojeve i definisani su tako da p+q bude ceo broj od I do 5; R1 predstavlja atom vodonika, halogena ili hidroksilnu, cijano, nitro, Cl-3-alkil, C1-3-alkoksi, C1-3-tioalkil, C1-3-f1uoroalkil, C1-3-f1uoroalkoksi, C1-3-f1uorotioalkil grupu; R2 predstavlja atom vodonika, halogena ili cijano, nitro, hidroksilnu, C1-3-alkil, C1-3-alkoksi, C1-3-tioalkil, C1-3-fluoroalkil, C1-3-fluoroalkoksi, Cl-3-f1uorotioalkil grupu ili aromatičnu ili heteroaromatičnu, eventualno supstituisanu grupu; R3 predstavlja ili 2,2,2-trif1uoroetil grupu, ili eventualno supstituisanu fenil grupu; a R6 i R7 predstavljaju, nezavisno jedan od drugog, C 1-3-alkil i fenil; u vidu baze, adicione soli kiseline, hidrata ili solvata. Primena u terapeutici.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MEP-306/08A MEP30608A (en) | 2003-10-03 | 2004-10-01 | Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0311615A FR2860514A1 (fr) | 2003-10-03 | 2003-10-03 | Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique |
PCT/FR2004/002486 WO2005033066A2 (fr) | 2003-10-03 | 2004-10-01 | Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique sanofi-synthelabo |
Publications (1)
Publication Number | Publication Date |
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RS20060239A true RS20060239A (en) | 2008-06-05 |
Family
ID=34307401
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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YUP-2006/0239A RS20060239A (en) | 2003-10-03 | 2004-10-01 | Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics |
Country Status (21)
Country | Link |
---|---|
US (1) | US7696374B2 (sr) |
EP (2) | EP1972616A1 (sr) |
JP (1) | JP4822351B2 (sr) |
KR (2) | KR20110093928A (sr) |
CN (1) | CN1878750B (sr) |
AT (1) | ATE534621T1 (sr) |
AU (2) | AU2004277436B2 (sr) |
BR (1) | BRPI0414855A (sr) |
CA (1) | CA2539849A1 (sr) |
FR (1) | FR2860514A1 (sr) |
HK (1) | HK1097250A1 (sr) |
IL (1) | IL174555A0 (sr) |
MA (1) | MA28074A1 (sr) |
ME (1) | MEP30608A (sr) |
MX (1) | MXPA06003751A (sr) |
NO (1) | NO20061982L (sr) |
NZ (1) | NZ546309A (sr) |
RS (1) | RS20060239A (sr) |
RU (1) | RU2400472C2 (sr) |
SG (1) | SG139760A1 (sr) |
WO (1) | WO2005033066A2 (sr) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2864080B1 (fr) * | 2003-12-23 | 2006-02-03 | Sanofi Synthelabo | Derives de 1-piperazine-et-1-homopiperazine-carboxylates, leur preparation et leur application en therapeutique |
FR2866885B1 (fr) | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique |
FR2885364B1 (fr) * | 2005-05-03 | 2007-06-29 | Sanofi Aventis Sa | Derives d'alkyl-, alkenyl-et alkynylcarbamates, leur preparation et leur application en therapeutique |
CN101253173A (zh) * | 2005-09-02 | 2008-08-27 | 辉瑞有限公司 | 羟基取代的1h-咪唑并吡啶和方法 |
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-
2003
- 2003-10-03 FR FR0311615A patent/FR2860514A1/fr not_active Withdrawn
-
2004
- 2004-10-01 KR KR1020117015377A patent/KR20110093928A/ko not_active Application Discontinuation
- 2004-10-01 NZ NZ546309A patent/NZ546309A/en not_active IP Right Cessation
- 2004-10-01 SG SG200800743-7A patent/SG139760A1/en unknown
- 2004-10-01 EP EP08012005A patent/EP1972616A1/fr not_active Withdrawn
- 2004-10-01 EP EP04817093A patent/EP1673337B1/fr active Active
- 2004-10-01 MX MXPA06003751A patent/MXPA06003751A/es active IP Right Grant
- 2004-10-01 ME MEP-306/08A patent/MEP30608A/xx unknown
- 2004-10-01 KR KR1020067006449A patent/KR20060100373A/ko not_active Application Discontinuation
- 2004-10-01 CA CA002539849A patent/CA2539849A1/fr not_active Abandoned
- 2004-10-01 AU AU2004277436A patent/AU2004277436B2/en not_active Ceased
- 2004-10-01 AT AT04817093T patent/ATE534621T1/de active
- 2004-10-01 CN CN2004800327944A patent/CN1878750B/zh not_active Expired - Fee Related
- 2004-10-01 JP JP2006530410A patent/JP4822351B2/ja not_active Expired - Fee Related
- 2004-10-01 BR BRPI0414855-0A patent/BRPI0414855A/pt not_active IP Right Cessation
- 2004-10-01 WO PCT/FR2004/002486 patent/WO2005033066A2/fr active Search and Examination
- 2004-10-01 RS YUP-2006/0239A patent/RS20060239A/sr unknown
- 2004-10-01 RU RU2006114700/04A patent/RU2400472C2/ru not_active IP Right Cessation
-
2006
- 2006-03-26 IL IL174555A patent/IL174555A0/en unknown
- 2006-03-27 MA MA28890A patent/MA28074A1/fr unknown
- 2006-03-31 US US11/395,942 patent/US7696374B2/en not_active Expired - Fee Related
- 2006-05-03 NO NO20061982A patent/NO20061982L/no not_active Application Discontinuation
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2007
- 2007-04-20 HK HK07104181.4A patent/HK1097250A1/xx not_active IP Right Cessation
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2011
- 2011-03-08 AU AU2011201012A patent/AU2011201012B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
FR2860514A1 (fr) | 2005-04-08 |
JP2007507474A (ja) | 2007-03-29 |
KR20110093928A (ko) | 2011-08-18 |
MEP30608A (en) | 2010-10-10 |
KR20060100373A (ko) | 2006-09-20 |
MA28074A1 (fr) | 2006-08-01 |
BRPI0414855A (pt) | 2006-11-21 |
WO2005033066A3 (fr) | 2006-05-11 |
RU2400472C2 (ru) | 2010-09-27 |
AU2004277436A1 (en) | 2005-04-14 |
CN1878750B (zh) | 2011-04-20 |
US7696374B2 (en) | 2010-04-13 |
EP1673337B1 (fr) | 2011-11-23 |
IL174555A0 (en) | 2006-08-20 |
MXPA06003751A (es) | 2006-06-23 |
HK1097250A1 (en) | 2007-06-22 |
NO20061982L (no) | 2006-07-03 |
WO2005033066A2 (fr) | 2005-04-14 |
JP4822351B2 (ja) | 2011-11-24 |
US20060223805A1 (en) | 2006-10-05 |
AU2011201012A1 (en) | 2011-03-31 |
EP1972616A1 (fr) | 2008-09-24 |
AU2011201012B2 (en) | 2011-12-15 |
SG139760A1 (en) | 2008-02-29 |
ATE534621T1 (de) | 2011-12-15 |
RU2006114700A (ru) | 2007-11-20 |
AU2004277436B2 (en) | 2011-04-14 |
EP1673337A2 (fr) | 2006-06-28 |
CA2539849A1 (fr) | 2005-04-14 |
CN1878750A (zh) | 2006-12-13 |
NZ546309A (en) | 2010-01-29 |
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