MEP30608A - Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics - Google Patents

Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics

Info

Publication number
MEP30608A
MEP30608A MEP-306/08A MEP30608A MEP30608A ME P30608 A MEP30608 A ME P30608A ME P30608 A MEP30608 A ME P30608A ME P30608 A MEP30608 A ME P30608A
Authority
ME
Montenegro
Prior art keywords
phenyl
ethylcarbamate
alkyl
optionally substituted
nitrophenyl
Prior art date
Application number
MEP-306/08A
Other languages
Bosnian (bs)
English (en)
Inventor
Ahmed Abouabdellah
Garcia Antonio Almario
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MEP30608A publication Critical patent/MEP30608A/xx

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/40Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/42Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/44Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/325Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • AHUMAN NECESSITIES
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    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/12Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/24Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/40Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/42Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/48Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by singly-bound oxygen atoms
MEP-306/08A 2003-10-03 2004-10-01 Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics MEP30608A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0311615A FR2860514A1 (fr) 2003-10-03 2003-10-03 Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique
PCT/FR2004/002486 WO2005033066A2 (fr) 2003-10-03 2004-10-01 Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique sanofi-synthelabo
YUP-2006/0239A RS20060239A (xx) 2003-10-03 2004-10-01 Derivati arilalkilkarbamata, njihovo dobijanje i njihova primena kao terapeutika

Publications (1)

Publication Number Publication Date
MEP30608A true MEP30608A (en) 2010-10-10

Family

ID=34307401

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-306/08A MEP30608A (en) 2003-10-03 2004-10-01 Arylalkylcarbamate derivatives, preparation method thereof and use of same in therapeutics

Country Status (21)

Country Link
US (1) US7696374B2 (xx)
EP (2) EP1972616A1 (xx)
JP (1) JP4822351B2 (xx)
KR (2) KR20110093928A (xx)
CN (1) CN1878750B (xx)
AT (1) ATE534621T1 (xx)
AU (2) AU2004277436B2 (xx)
BR (1) BRPI0414855A (xx)
CA (1) CA2539849A1 (xx)
FR (1) FR2860514A1 (xx)
HK (1) HK1097250A1 (xx)
IL (1) IL174555A0 (xx)
MA (1) MA28074A1 (xx)
ME (1) MEP30608A (xx)
MX (1) MXPA06003751A (xx)
NO (1) NO20061982L (xx)
NZ (1) NZ546309A (xx)
RS (1) RS20060239A (xx)
RU (1) RU2400472C2 (xx)
SG (1) SG139760A1 (xx)
WO (1) WO2005033066A2 (xx)

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FR2864080B1 (fr) * 2003-12-23 2006-02-03 Sanofi Synthelabo Derives de 1-piperazine-et-1-homopiperazine-carboxylates, leur preparation et leur application en therapeutique
FR2866885B1 (fr) 2004-02-26 2007-08-31 Sanofi Synthelabo Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique
FR2885364B1 (fr) * 2005-05-03 2007-06-29 Sanofi Aventis Sa Derives d'alkyl-, alkenyl-et alkynylcarbamates, leur preparation et leur application en therapeutique
CN101253173A (zh) * 2005-09-02 2008-08-27 辉瑞有限公司 羟基取代的1h-咪唑并吡啶和方法
WO2007047575A2 (en) * 2005-10-14 2007-04-26 The Board Of Trustees Of The University Of Illinois Pharmacological treatments for sleep-related breathing disorders
US20080089845A1 (en) * 2006-09-07 2008-04-17 N.V. Organon Methods for determining effective doses of fatty acid amide hydrolase inhibitors in vivo
WO2008042892A2 (en) * 2006-10-02 2008-04-10 N.V. Organon Fatty acid amide hydrolase inhibitors for energy metabolism disorders
EP2096915A1 (en) * 2006-11-20 2009-09-09 N.V. Organon Metabolically-stabilized inhibitors of fatty acid amide hydrolase
WO2009009041A2 (en) * 2007-07-06 2009-01-15 Kinex Pharmaceuticals, Llc Compositions and methods for modulating a kinase cascade
US8207226B1 (en) 2008-06-03 2012-06-26 Alcon Research, Ltd. Use of FAAH antagonists for treating dry eye and ocular pain
WO2012058115A2 (en) * 2010-10-28 2012-05-03 Benjamin Cravatt Anti-cancer serine hydrolase inhibitory carbamates
CA2883144C (en) 2012-08-30 2023-01-17 Kinex Pharmaceuticals, Llc N-(3-fluorobenzyl)-2-(5-(4-morpholinophenyl)pyridin-2-yl) acetamide as protein|tyrosine kinase modulators
CN105418460B (zh) * 2014-08-11 2017-04-12 苏州鹏旭医药科技有限公司 匹莫范色林及其类似化合物中间体,其制备方法和制备匹莫范色林及其类似化合物的方法
JP6980534B2 (ja) 2015-06-25 2021-12-15 ザ チルドレンズ メディカル センター コーポレーション 造血幹細胞の増大、富化、および維持に関する方法および組成物
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JP2007507474A (ja) 2007-03-29
KR20110093928A (ko) 2011-08-18
KR20060100373A (ko) 2006-09-20
MA28074A1 (fr) 2006-08-01
BRPI0414855A (pt) 2006-11-21
WO2005033066A3 (fr) 2006-05-11
RU2400472C2 (ru) 2010-09-27
AU2004277436A1 (en) 2005-04-14
CN1878750B (zh) 2011-04-20
US7696374B2 (en) 2010-04-13
EP1673337B1 (fr) 2011-11-23
IL174555A0 (en) 2006-08-20
MXPA06003751A (es) 2006-06-23
HK1097250A1 (en) 2007-06-22
NO20061982L (no) 2006-07-03
WO2005033066A2 (fr) 2005-04-14
JP4822351B2 (ja) 2011-11-24
US20060223805A1 (en) 2006-10-05
AU2011201012A1 (en) 2011-03-31
EP1972616A1 (fr) 2008-09-24
AU2011201012B2 (en) 2011-12-15
SG139760A1 (en) 2008-02-29
ATE534621T1 (de) 2011-12-15
RU2006114700A (ru) 2007-11-20
AU2004277436B2 (en) 2011-04-14
EP1673337A2 (fr) 2006-06-28
RS20060239A (xx) 2008-06-05
CA2539849A1 (fr) 2005-04-14
CN1878750A (zh) 2006-12-13
NZ546309A (en) 2010-01-29

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