PT946566E - Formas pro-farmacos e analogos da camptotecina sua aplicacao como medicamentos - Google Patents
Formas pro-farmacos e analogos da camptotecina sua aplicacao como medicamentosInfo
- Publication number
- PT946566E PT946566E PT97950235T PT97950235T PT946566E PT 946566 E PT946566 E PT 946566E PT 97950235 T PT97950235 T PT 97950235T PT 97950235 T PT97950235 T PT 97950235T PT 946566 E PT946566 E PT 946566E
- Authority
- PT
- Portugal
- Prior art keywords
- analogenic
- camptotecin
- medicines
- pharmacological
- pro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9615775A FR2757515B1 (fr) | 1996-12-20 | 1996-12-20 | Formes prodrogues et nouveaux analogues de la camptothecine, leurs procedes de preparation, leur application comme medicaments et les compositions pharmaceutiques les contenant |
FR9615945 | 1996-12-24 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT946566E true PT946566E (pt) | 2004-03-31 |
Family
ID=26233188
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT97950235T PT946566E (pt) | 1996-12-20 | 1997-12-05 | Formas pro-farmacos e analogos da camptotecina sua aplicacao como medicamentos |
Country Status (24)
Country | Link |
---|---|
EP (1) | EP0946566B1 (pt) |
JP (1) | JP3576174B2 (pt) |
KR (1) | KR100516873B1 (pt) |
CN (1) | CN1090634C (pt) |
AR (1) | AR005849A1 (pt) |
AT (1) | ATE253582T1 (pt) |
AU (1) | AU734512B2 (pt) |
BR (1) | BR9713977B1 (pt) |
CA (1) | CA2275345C (pt) |
CZ (1) | CZ299794B6 (pt) |
DE (1) | DE69726007T2 (pt) |
DK (1) | DK0946566T3 (pt) |
ES (1) | ES2206760T3 (pt) |
HK (1) | HK1024694A1 (pt) |
HU (1) | HUP0001385A3 (pt) |
IL (2) | IL129892A0 (pt) |
MY (1) | MY122042A (pt) |
NO (1) | NO324973B1 (pt) |
NZ (1) | NZ335938A (pt) |
PL (1) | PL188109B1 (pt) |
PT (1) | PT946566E (pt) |
TW (1) | TW410224B (pt) |
UA (1) | UA57757C2 (pt) |
WO (1) | WO1998028304A1 (pt) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2790261B1 (fr) * | 1999-02-26 | 2004-09-10 | Sod Conseils Rech Applic | Nouveaux analogues optiquement purs de la camptothecine et leurs procedes de preparation |
AU764123B2 (en) * | 1998-09-02 | 2003-08-07 | Pharmagenesis, Inc. | Triptolide prodrugs having high aqueous solubility |
US6207832B1 (en) | 1999-04-09 | 2001-03-27 | University Of Pittsburgh | Camptothecin analogs and methods of preparation thereof |
FR2801309B1 (fr) * | 1999-11-18 | 2002-01-04 | Adir | Nouveaux composes analogues de la camptothecine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
US6350756B1 (en) | 2001-01-18 | 2002-02-26 | California Pacific Medical Center | Camptothecin derivatives |
US6403604B1 (en) | 2001-03-01 | 2002-06-11 | California Pacific Medical Center | Nitrogen-based camptothecin derivatives |
US6855720B2 (en) | 2001-03-01 | 2005-02-15 | California Pacific Medical Center | Nitrogen-based camptothecin derivatives |
US20040077674A1 (en) * | 2002-03-01 | 2004-04-22 | Curran Dennis P. | Mappicine analogs, intermediates in the synthesis of mappicine analogs and methods of synthesis of mappicine analogs |
US6933302B2 (en) | 2002-06-03 | 2005-08-23 | California Pacific Medical Center | Nitrogen-based homo-camptothecin derivatives |
EP1694684B1 (en) * | 2003-12-17 | 2011-08-03 | Bionumerik Pharmaceuticals, Inc. | Process for making camptothecin derivatives |
WO2005097803A1 (ja) * | 2004-04-09 | 2005-10-20 | Chugai Seiyaku Kabushiki Kaisha | 新規水溶性プロドラッグ |
ITRM20040288A1 (it) * | 2004-06-11 | 2004-09-11 | Sigma Tau Ind Farmaceuti | Uso della 7-t-butossiimminometilcamptotecina per la preparazione di un medicamento per il trattamento delle neoplasie dell'utero. |
TW200744603A (en) | 2005-08-22 | 2007-12-16 | Chugai Pharmaceutical Co Ltd | Novel anticancer concomitant drug |
FR2892418B1 (fr) * | 2005-10-24 | 2010-10-22 | Servier Lab | Nouveaux composes aminoesterifies a cycle e hydrocarbone a six chainons analogues de la camptothecine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2892417B1 (fr) * | 2005-10-24 | 2010-10-22 | Servier Lab | Nouveaux composes aminoesterifies a cycle e hydrocarbone a sept chainons analogues de la camptothecine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
CN100465175C (zh) * | 2005-11-29 | 2009-03-04 | 中国人民解放军第二军医大学 | 7-位取代高喜树碱类化合物及作为药物的用途 |
CN100441580C (zh) * | 2006-07-14 | 2008-12-10 | 中山大学 | 喹啉二酮衍生物及其在制备抗菌药物中的应用 |
CN102746314B (zh) * | 2011-04-18 | 2016-07-06 | 华东师范大学 | 含有稳定7元内酯环的喜树碱类化合物、制备方法和用途 |
CN117164601A (zh) * | 2022-06-02 | 2023-12-05 | 华东师范大学 | 一种高喜树碱类小分子及其应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5391745A (en) * | 1992-07-23 | 1995-02-21 | Sloan-Kettering Institute For Cancer Research | Methods of preparation of camptothecin analogs |
CN1114608C (zh) * | 1995-06-21 | 2003-07-16 | 科学研究与运用咨询公司 | 喜树碱类似物、其制备方法和药物应用及其药物组合物 |
-
1997
- 1997-05-12 UA UA99063448A patent/UA57757C2/uk unknown
- 1997-12-05 ES ES97950235T patent/ES2206760T3/es not_active Expired - Lifetime
- 1997-12-05 CZ CZ0209299A patent/CZ299794B6/cs not_active IP Right Cessation
- 1997-12-05 EP EP97950235A patent/EP0946566B1/fr not_active Expired - Lifetime
- 1997-12-05 IL IL12989297A patent/IL129892A0/xx active IP Right Grant
- 1997-12-05 WO PCT/FR1997/002217 patent/WO1998028304A1/fr active IP Right Grant
- 1997-12-05 DK DK97950235T patent/DK0946566T3/da active
- 1997-12-05 PT PT97950235T patent/PT946566E/pt unknown
- 1997-12-05 DE DE69726007T patent/DE69726007T2/de not_active Expired - Lifetime
- 1997-12-05 NZ NZ335938A patent/NZ335938A/xx not_active IP Right Cessation
- 1997-12-05 PL PL97334092A patent/PL188109B1/pl not_active IP Right Cessation
- 1997-12-05 KR KR10-1999-7005604A patent/KR100516873B1/ko not_active IP Right Cessation
- 1997-12-05 CN CN97180816A patent/CN1090634C/zh not_active Expired - Fee Related
- 1997-12-05 HU HU0001385A patent/HUP0001385A3/hu unknown
- 1997-12-05 JP JP52844798A patent/JP3576174B2/ja not_active Expired - Fee Related
- 1997-12-05 BR BRPI9713977-7A patent/BR9713977B1/pt not_active IP Right Cessation
- 1997-12-05 AU AU53264/98A patent/AU734512B2/en not_active Ceased
- 1997-12-05 CA CA2275345A patent/CA2275345C/fr not_active Expired - Fee Related
- 1997-12-05 AT AT97950235T patent/ATE253582T1/de active
- 1997-12-19 AR ARP970106042A patent/AR005849A1/es active IP Right Grant
- 1997-12-19 TW TW086119342A patent/TW410224B/zh not_active IP Right Cessation
- 1997-12-20 MY MYPI97006216A patent/MY122042A/en unknown
-
1999
- 1999-05-11 IL IL129892A patent/IL129892A/en not_active IP Right Cessation
- 1999-06-18 NO NO19992997A patent/NO324973B1/no not_active IP Right Cessation
-
2000
- 2000-07-04 HK HK00104033A patent/HK1024694A1/xx not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PT946566E (pt) | Formas pro-farmacos e analogos da camptotecina sua aplicacao como medicamentos | |
PT1006110E (pt) | Derivados de acil-piperazinil-pirimidinas sua preparacao e aplicacao como medicamentos | |
BR9607317A (pt) | Peptídios e composição farmacêutica | |
BR9607318A (pt) | Peptidos e composição farmacêutica | |
DE69838386D1 (de) | Beleuchtungssystem und dessen anwendung | |
PT1119557E (pt) | Derivados de indeno- nafto- e benzociclohepta-di-hidrotiazole sua preparacao e sua utilizacao como medicamentos anorecticos | |
FI960635A0 (fi) | Elektrodi ja sen valmistus | |
PT937083E (pt) | Substancia cristalina de cefditoren pivoxil e sua producao | |
NO965103L (no) | Bicykliske aromatiske forbindelser, anvendelse derav, og farmasöytiske og kosmetiske preparater | |
BR9607851B1 (pt) | combinaÇço e formulaÇço farmacÊutica. | |
LV12624B (lv) | Tienilazolilalkosietanamini to iegusanas panemiens un pielietojums medikamentu legusana | |
DE69621221D1 (de) | Klebstoffzusammensetzung und luftreifen | |
FI965204A0 (fi) | Bromelaiinin lääkekäyttö | |
NO965102D0 (no) | Bicykliske aromatiske forbindelser, anvendelser derav, og farmasöytiske og kosmetiske preparater | |
KR960016892A (ko) | 약제의 신독성 경감제 | |
BR9509688A (pt) | Composto e composição farmacêutica | |
ID19147A (id) | Ksilanase dan pemakaiannya | |
PT858445E (pt) | Novos derivados de ¬(3-alcoxi-fenoxi)-etil|-dialquilamina e sua utilizacao como anrstesicos locais | |
DE69837507D1 (de) | Humanes Hedgehog-Protein | |
BR9609081A (pt) | Combinações de substáncias ativas | |
PT922703E (pt) | Benzocicloalcenos substituidos e sua utilizacao como substancias com efeito analgesico | |
EA199900672A1 (ru) | Гомеопатическое лекарственное средство | |
NO963482D0 (no) | Medisinsk anvendelse av bromelain | |
FR2752317B1 (fr) | Terminal medical et paramedical | |
KR960010685A (ko) | 펩티드 및 그 용도 |