PT922703E - Benzocicloalcenos substituidos e sua utilizacao como substancias com efeito analgesico - Google Patents

Benzocicloalcenos substituidos e sua utilizacao como substancias com efeito analgesico

Info

Publication number
PT922703E
PT922703E PT98122218T PT98122218T PT922703E PT 922703 E PT922703 E PT 922703E PT 98122218 T PT98122218 T PT 98122218T PT 98122218 T PT98122218 T PT 98122218T PT 922703 E PT922703 E PT 922703E
Authority
PT
Portugal
Prior art keywords
benzocycloalcenses
substances
substituted
analgesic effect
analgesic
Prior art date
Application number
PT98122218T
Other languages
English (en)
Inventor
Zimmer Dr Oswald
Strassburger Prof Dr Wolfgang
Putz Dr Claudia
Englberger Dr Werner
Kogel Dr Babette-Yvonne
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of PT922703E publication Critical patent/PT922703E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D335/00Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/06Benzothiopyrans; Hydrogenated benzothiopyrans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D313/00Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
    • C07D313/02Seven-membered rings
    • C07D313/06Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D313/08Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D335/00Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/08Naphthothiopyrans; Hydrogenated naphthothiopyrans
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D337/00Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02Seven-membered rings
    • C07D337/06Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems
PT98122218T 1997-12-13 1998-11-23 Benzocicloalcenos substituidos e sua utilizacao como substancias com efeito analgesico PT922703E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19755480A DE19755480A1 (de) 1997-12-13 1997-12-13 Substituierte heterocyclische Benzocycloalkene und ihre Verwendung als analgetisch wirksame Substanzen

Publications (1)

Publication Number Publication Date
PT922703E true PT922703E (pt) 2003-04-30

Family

ID=7851818

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98122218T PT922703E (pt) 1997-12-13 1998-11-23 Benzocicloalcenos substituidos e sua utilizacao como substancias com efeito analgesico

Country Status (29)

Country Link
US (1) US6013809A (pt)
EP (1) EP0922703B1 (pt)
JP (1) JPH11246547A (pt)
KR (1) KR19990062982A (pt)
CN (1) CN100376564C (pt)
AR (1) AR017800A1 (pt)
AT (1) ATE229016T1 (pt)
AU (1) AU747979B2 (pt)
BR (1) BR9805437A (pt)
CA (1) CA2256007C (pt)
CO (1) CO4990950A1 (pt)
CZ (1) CZ294990B6 (pt)
DE (2) DE19755480A1 (pt)
DK (1) DK0922703T3 (pt)
ES (1) ES2189072T3 (pt)
HK (1) HK1020944A1 (pt)
HU (1) HU226014B1 (pt)
IL (1) IL127518A (pt)
MY (1) MY133169A (pt)
NO (1) NO985818L (pt)
NZ (1) NZ332622A (pt)
PE (1) PE133499A1 (pt)
PL (1) PL194934B1 (pt)
PT (1) PT922703E (pt)
RU (1) RU2197484C2 (pt)
SI (1) SI0922703T1 (pt)
SK (1) SK283366B6 (pt)
UY (1) UY25296A1 (pt)
ZA (1) ZA9811346B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6077850A (en) * 1997-04-21 2000-06-20 G.D. Searle & Co. Substituted benzopyran analogs for the treatment of inflammation
US6221897B1 (en) 1998-06-10 2001-04-24 Aventis Pharma Deutschland Gmbh Benzothiepine 1,1-dioxide derivatives, a process for their preparation, pharmaceuticals comprising these compounds, and their use
DE19830105C1 (de) * 1998-07-06 2000-02-17 Gruenenthal Gmbh Acridinderivate
AU5301599A (en) 1998-08-20 2000-03-14 Takeda Chemical Industries Ltd. Quaternary ammonium salts and their use
DE10033459A1 (de) * 2000-07-10 2002-01-24 Gruenenthal Gmbh Cyclische substituierte Aminomethylverbindungen und diese Verbindungen enthaltende Arzeimittel
US7289083B1 (en) * 2000-11-30 2007-10-30 Palm, Inc. Multi-sided display for portable computer
CA2722122C (en) * 2008-04-28 2017-01-03 Janssen Pharmaceutica Nv Benzocycloheptane and benzoxepine derivatives
US20140243281A1 (en) 2011-10-28 2014-08-28 Lumena Pharmaceuticals, Inc. Bile acid recycling inhibitors for treatment of pediatric cholestatic liver diseases
CN104844471B (zh) * 2015-04-21 2017-05-03 苏州远智医药科技有限公司 一种作为dor受体拮抗剂的化合物
CN109896991B (zh) * 2017-12-08 2020-11-20 苏州远智医药科技有限公司 一种δ阿片受体拮抗剂及其用途和药物组合物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3444176A (en) * 1967-04-28 1969-05-13 Mcneilab Inc Certain 4-diloweralkylamino-lower alkyl - 5 - pyridyl (or phenyl)-2,3-dihydro - 1 - benzothiepins and derivatives thereof
US4104280A (en) * 1977-02-04 1978-08-01 Syntex (U.S.A.) Inc. Dibenzo [b.f]thiepin and dibenzo[b.f]oxepin derivatives
JPS61130286A (ja) * 1984-11-28 1986-06-18 Suntory Ltd 2,3−ジヒドロ−1−ベンズオキセピン誘導体
JP3042156B2 (ja) * 1992-02-20 2000-05-15 田辺製薬株式会社 ナフタレン誘導体、その製法及びその合成中間体
US5482967A (en) * 1992-09-04 1996-01-09 Takeda Chemical Industries, Ltd. Condensed heterocyclic compounds, their production and use

Also Published As

Publication number Publication date
UY25296A1 (es) 2001-05-31
DK0922703T3 (da) 2003-03-17
PE133499A1 (es) 2000-02-02
NO985818D0 (no) 1998-12-11
PL330257A1 (en) 1999-06-21
EP0922703B1 (de) 2002-12-04
NZ332622A (en) 2000-03-27
AR017800A1 (es) 2001-10-24
HUP9802886A3 (en) 2001-09-28
CN1221743A (zh) 1999-07-07
CA2256007C (en) 2009-04-14
CZ407698A3 (cs) 1999-06-16
SK283366B6 (sk) 2003-06-03
HU9802886D0 (en) 1999-02-01
AU747979B2 (en) 2002-05-30
ES2189072T3 (es) 2003-07-01
HU226014B1 (en) 2008-02-28
IL127518A (en) 2003-05-29
JPH11246547A (ja) 1999-09-14
PL194934B1 (pl) 2007-07-31
BR9805437A (pt) 2000-05-02
US6013809A (en) 2000-01-11
SI0922703T1 (en) 2003-04-30
HK1020944A1 (en) 2000-05-26
DE19755480A1 (de) 1999-06-24
IL127518A0 (en) 1999-10-28
CN100376564C (zh) 2008-03-26
RU2197484C2 (ru) 2003-01-27
CZ294990B6 (cs) 2005-04-13
CA2256007A1 (en) 1999-06-13
DE59806523D1 (de) 2003-01-16
KR19990062982A (ko) 1999-07-26
ATE229016T1 (de) 2002-12-15
CO4990950A1 (es) 2000-12-26
NO985818L (no) 1999-06-14
MY133169A (en) 2007-10-31
EP0922703A1 (de) 1999-06-16
AU9707398A (en) 1999-07-01
HUP9802886A2 (hu) 2001-04-28
ZA9811346B (en) 1999-06-14
SK169998A3 (en) 1999-07-12

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