PT1853241E - Utilização de 2-(2-nitro-4-trifluorometilbenzoil)-1,3- ciclohexanodiona no tratamento de doença de parkinson - Google Patents
Utilização de 2-(2-nitro-4-trifluorometilbenzoil)-1,3- ciclohexanodiona no tratamento de doença de parkinson Download PDFInfo
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- PT1853241E PT1853241E PT06709910T PT06709910T PT1853241E PT 1853241 E PT1853241 E PT 1853241E PT 06709910 T PT06709910 T PT 06709910T PT 06709910 T PT06709910 T PT 06709910T PT 1853241 E PT1853241 E PT 1853241E
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- compound
- effective amount
- pharmaceutically acceptable
- alkyl
- pharmaceutically effective
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/12—Ketones
- A61K31/122—Ketones having the oxygen directly attached to a ring, e.g. quinones, vitamin K1, anthralin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
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- Engineering & Computer Science (AREA)
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- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
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| GBGB0504103.3A GB0504103D0 (en) | 2005-02-28 | 2005-02-28 | Novel method |
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Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2748599T3 (es) | 2007-08-27 | 2020-03-17 | Dart Neuroscience Cayman Ltd | Compuestos terapéuticos de isoxazol |
| CA2709784A1 (en) * | 2007-12-21 | 2009-07-09 | University Of Rochester | Method for altering the lifespan of eukaryotic organisms |
| CN102395595A (zh) * | 2008-11-06 | 2012-03-28 | 生物链接治疗股份有限公司 | 不宁腿综合症和睡眠障碍的治疗 |
| JP6038132B2 (ja) | 2011-06-23 | 2016-12-07 | スウェディッシュ オーファン バイオビトラム インターナショナル アクチエボラグ | ニチシノンを含む液体薬学的組成物 |
| CN103622942A (zh) * | 2013-11-04 | 2014-03-12 | 江苏大学 | 左旋多巴/卡比多巴复方缓释混悬剂及其制备方法 |
| WO2017017165A1 (en) * | 2015-07-29 | 2017-02-02 | Takeda Gmbh | Pde4 inhibitor for the treatment of diabetic nephropathy |
| ITUB20160650A1 (it) | 2016-02-11 | 2017-08-11 | Dipharma S A | Formulazioni farmaceutiche solide stabili contenenti 2-(2-nitro-4-trifluorometilbenzoil)-1,3-cicloesandione |
| US9783485B1 (en) | 2016-11-30 | 2017-10-10 | Dipharma S.A. | Crystalline inhibitor of 4-hydroxyphenylpyruvate dioxygenase, and a process of synthesis and crystallization thereof |
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| US4780127A (en) * | 1982-03-25 | 1988-10-25 | Stauffer Chemical Company | Certain 2-(substituted benzoyl)-1,3-cyclohexanediones and their use as herbicides |
| US5092919A (en) * | 1991-01-15 | 1992-03-03 | Imperial Chemical Industries Plc | Certain 2-(2'-methyl-3',4'-trisubstituted benzoyl)-1,3-cyclohexanediones |
| AU672361B2 (en) * | 1991-06-24 | 1996-10-03 | Swedish Orphan Biovitrum International Ab | Use of 2-(2-nitro-4-trifluoromethylbenzoyl)-1,3-cyclohexanedione in the treatment of tyrosinaemia and pharmaceutical compositions |
| FR2777781B1 (fr) * | 1998-04-24 | 2004-04-09 | Rhone Poulenc Rorer Sa | Associations riluzole et l-dopa pour le traitement de la maladie de parkinson |
| US20050288187A1 (en) * | 2002-07-03 | 2005-12-29 | Hanauske-Abel Hartmut M | Inhibitor development for 4-hydroxyphenylpyruvate dioxygenase, employing tyrosinemia 1 as a model for human diseases mediated by 2-oxoacid utilizing dioxygenases |
| US20060166972A1 (en) * | 2003-07-11 | 2006-07-27 | Conn P J | Treatment of movement disorders with a metabotropic glutamate 4 receptor positive allosteric modulator |
| EP2233136A1 (en) * | 2006-08-18 | 2010-09-29 | Syngenta Limited | Use of HPPD Inhibitors in the Treatment of Depression and/or Withdrawal Symptoms Associated with Addictive Drugs |
| CN102395595A (zh) * | 2008-11-06 | 2012-03-28 | 生物链接治疗股份有限公司 | 不宁腿综合症和睡眠障碍的治疗 |
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2005
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2006
- 2006-02-27 JP JP2007557572A patent/JP2008531665A/ja active Pending
- 2006-02-27 PT PT06709910T patent/PT1853241E/pt unknown
- 2006-02-27 MX MX2007010480A patent/MX2007010480A/es not_active Application Discontinuation
- 2006-02-27 DK DK06709910.1T patent/DK1853241T3/da active
- 2006-02-27 CN CN2006800133878A patent/CN101163466B/zh not_active Expired - Fee Related
- 2006-02-27 BR BRPI0609177-6A patent/BRPI0609177A2/pt not_active IP Right Cessation
- 2006-02-27 WO PCT/GB2006/000684 patent/WO2006090177A1/en not_active Ceased
- 2006-02-27 AT AT06709910T patent/ATE524171T1/de active
- 2006-02-27 ZA ZA200707486A patent/ZA200707486B/xx unknown
- 2006-02-27 AU AU2006217650A patent/AU2006217650B2/en not_active Ceased
- 2006-02-27 US US12/090,645 patent/US20090326072A1/en not_active Abandoned
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- 2006-02-27 CA CA002598517A patent/CA2598517A1/en not_active Abandoned
- 2006-02-27 EP EP06709910A patent/EP1853241B1/en active Active
- 2006-02-27 RU RU2007131934/15A patent/RU2420272C2/ru not_active IP Right Cessation
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Also Published As
| Publication number | Publication date |
|---|---|
| RU2420272C2 (ru) | 2011-06-10 |
| CA2598517A1 (en) | 2006-08-31 |
| EP1853241A1 (en) | 2007-11-14 |
| JP2008531665A (ja) | 2008-08-14 |
| WO2006090177A1 (en) | 2006-08-31 |
| ES2374761T3 (es) | 2012-02-21 |
| CN101163466B (zh) | 2011-12-07 |
| BRPI0609177A2 (pt) | 2010-02-23 |
| EP1853241B1 (en) | 2011-09-14 |
| CN101163466A (zh) | 2008-04-16 |
| AU2006217650A1 (en) | 2006-08-31 |
| AU2006217650B2 (en) | 2011-06-09 |
| RU2007131934A (ru) | 2009-02-27 |
| US20090326072A1 (en) | 2009-12-31 |
| ZA200707486B (en) | 2009-02-25 |
| IL185410A0 (en) | 2008-08-07 |
| DK1853241T3 (da) | 2012-01-16 |
| GB0504103D0 (en) | 2005-04-06 |
| ATE524171T1 (de) | 2011-09-15 |
| HK1110211A1 (en) | 2008-07-11 |
| MX2007010480A (es) | 2008-02-07 |
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