PT1819353E - Composi??o para inibi??o de proteassoma - Google Patents

Composi??o para inibi??o de proteassoma Download PDF

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Publication number
PT1819353E
PT1819353E PT05853385T PT05853385T PT1819353E PT 1819353 E PT1819353 E PT 1819353E PT 05853385 T PT05853385 T PT 05853385T PT 05853385 T PT05853385 T PT 05853385T PT 1819353 E PT1819353 E PT 1819353E
Authority
PT
Portugal
Prior art keywords
composition
compositions
proteasome inhibition
proteasome inhibitors
cyclodextrin
Prior art date
Application number
PT05853385T
Other languages
English (en)
Portuguese (pt)
Inventor
Evan R Lewis
Mark Nguyen Ho
Fabiana N Fonseca
Original Assignee
Proteolix Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36143200&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT1819353(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Proteolix Inc filed Critical Proteolix Inc
Publication of PT1819353E publication Critical patent/PT1819353E/pt

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    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/336Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having three-membered rings, e.g. oxirane, fumagillin
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/396Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having three-membered rings, e.g. aziridine
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
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    • C07K5/0812Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
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  • Biomedical Technology (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Inorganic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Biophysics (AREA)
PT05853385T 2004-12-07 2005-12-07 Composi??o para inibi??o de proteassoma PT1819353E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63436604P 2004-12-07 2004-12-07
US65593005P 2005-02-23 2005-02-23

Publications (1)

Publication Number Publication Date
PT1819353E true PT1819353E (pt) 2011-05-12

Family

ID=36143200

Family Applications (3)

Application Number Title Priority Date Filing Date
PT05853385T PT1819353E (pt) 2004-12-07 2005-12-07 Composi??o para inibi??o de proteassoma
PT101794220T PT2261236E (pt) 2004-12-07 2005-12-07 Composição para a inibição de proteassoma
PT101789980T PT2260835E (pt) 2004-12-07 2005-12-07 Composição para inibição do proteassoma

Family Applications After (2)

Application Number Title Priority Date Filing Date
PT101794220T PT2261236E (pt) 2004-12-07 2005-12-07 Composição para a inibição de proteassoma
PT101789980T PT2260835E (pt) 2004-12-07 2005-12-07 Composição para inibição do proteassoma

Country Status (17)

Country Link
US (1) US7737112B2 (enExample)
EP (3) EP2261236B1 (enExample)
JP (1) JP4990155B2 (enExample)
KR (1) KR101299821B1 (enExample)
CN (2) CN101180071A (enExample)
AT (1) ATE499109T1 (enExample)
AU (1) AU2005313975B2 (enExample)
CA (1) CA2589921C (enExample)
CY (1) CY1111489T1 (enExample)
DE (1) DE602005026556D1 (enExample)
DK (1) DK1819353T3 (enExample)
ES (2) ES2549763T3 (enExample)
HU (1) HUE027850T2 (enExample)
IL (1) IL183607A (enExample)
PL (3) PL2260835T3 (enExample)
PT (3) PT1819353E (enExample)
WO (1) WO2006063154A1 (enExample)

Families Citing this family (53)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5616569B2 (ja) 2004-04-15 2014-10-29 オニキス セラピューティクス, インク.Onyx Therapeutics, Inc. 酵素阻害のための化合物
US8198270B2 (en) * 2004-04-15 2012-06-12 Onyx Therapeutics, Inc. Compounds for proteasome enzyme inhibition
CN102875642A (zh) * 2004-05-10 2013-01-16 普罗特奥里克斯公司 用于酶抑制的化合物
US9034846B2 (en) * 2004-10-10 2015-05-19 Universite De Liege Use of cyclodextrin for treatment and prevention of bronchial inflammatory diseases
AU2006311584B2 (en) 2005-11-09 2012-03-08 Onyx Therapeutics, Inc. Compounds for enzyme inhibition
CN101506224B (zh) 2006-06-19 2016-03-30 欧尼斯治疗公司 蛋白酶体抑制用的肽环氧酮
PT2207791T (pt) 2007-10-04 2016-07-12 Onyx Therapeutics Inc Inibidores da epoxi cetona protease de péptido cristalino e a síntese de ceto-epóxidos de aminoácidos
US7635773B2 (en) 2008-04-28 2009-12-22 Cydex Pharmaceuticals, Inc. Sulfoalkyl ether cyclodextrin compositions
EP2344165A4 (en) * 2008-10-01 2012-12-05 Reddys Lab Ltd Dr PHARMACEUTICAL COMPOSITIONS COMPRISING BORONIC ACID COMPOUNDS
EP3090737A1 (en) * 2008-10-21 2016-11-09 Onyx Therapeutics, Inc. Combination therapy with peptide epoxyketones
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