PT1656345E - Derivados cíclicos como moduladores da actividade de receptores de quimioquinas - Google Patents

Derivados cíclicos como moduladores da actividade de receptores de quimioquinas Download PDF

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Publication number
PT1656345E
PT1656345E PT47818067T PT04781806T PT1656345E PT 1656345 E PT1656345 E PT 1656345E PT 47818067 T PT47818067 T PT 47818067T PT 04781806 T PT04781806 T PT 04781806T PT 1656345 E PT1656345 E PT 1656345E
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Portugal
Prior art keywords
modulators
chemokine receptor
receptor activity
cyclic derivatives
cyclic
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PT47818067T
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English (en)
Inventor
Douglas G Batt
Percy H Carter
Robert J Cherney
John V Duncia
Daniel S Gardner
Soo S Ko
Anurag S Srivastava
Michael G Yang
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Bristol Myers Squibb Co
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34228609&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT1656345(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of PT1656345E publication Critical patent/PT1656345E/pt

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    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
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    • C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
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    • C07D487/04—Ortho-condensed systems
PT47818067T 2003-08-21 2004-08-20 Derivados cíclicos como moduladores da actividade de receptores de quimioquinas PT1656345E (pt)

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Application Number Priority Date Filing Date Title
US49694703P 2003-08-21 2003-08-21
US10/923,619 US7163937B2 (en) 2003-08-21 2004-08-19 Cyclic derivatives as modulators of chemokine receptor activity

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EP (1) EP1656345B1 (pt)
JP (1) JP4795238B2 (pt)
KR (1) KR101120338B1 (pt)
AU (1) AU2004268968B2 (pt)
BR (1) BRPI0413713A (pt)
CA (1) CA2536384C (pt)
DK (1) DK1656345T3 (pt)
ES (1) ES2437104T3 (pt)
HK (1) HK1087712A1 (pt)
HR (1) HRP20131048T1 (pt)
IL (2) IL173824A (pt)
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NO (1) NO335946B1 (pt)
NZ (1) NZ545317A (pt)
PL (1) PL1656345T3 (pt)
PT (1) PT1656345E (pt)
RS (1) RS20060116A (pt)
RU (1) RU2006108867A (pt)
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AU2002241724A1 (en) 2000-12-20 2002-07-01 Bristol-Myers Squibb Company Diamines as modulators of chemokine receptor activity
US7087604B2 (en) * 2002-03-08 2006-08-08 Bristol-Myers Squibb Company Cyclic derivatives as modulators of chemokine receptor activity
US7291615B2 (en) 2003-05-01 2007-11-06 Bristol-Myers Squibb Company Cyclic derivatives as modulators of chemokine receptor activity
US7317019B2 (en) * 2003-08-21 2008-01-08 Bristol Myers Squibb Co. N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity
US7163937B2 (en) * 2003-08-21 2007-01-16 Bristol-Myers Squibb Company Cyclic derivatives as modulators of chemokine receptor activity
US7825244B2 (en) 2005-06-10 2010-11-02 Janssen Pharmaceutica Nv Intermediates useful in the synthesis of alkylquinoline and alkylquinazoline kinase modulators, and related methods of synthesis
US8071768B2 (en) 2005-06-10 2011-12-06 Janssen Pharmaceutica, N.V. Alkylquinoline and alkylquinazoline kinase modulators
JP2009503107A (ja) * 2005-08-04 2009-01-29 アポジー・バイオテクノロジー・コーポレイション スフィンゴシンキナーゼ阻害剤およびそれらの使用方法
US20100016289A1 (en) * 2005-11-01 2010-01-21 Kevin Sprott Compounds Useful as Antagonists of CCR2
WO2007053498A1 (en) * 2005-11-01 2007-05-10 Millennium Pharmaceuticals, Inc. Compounds useful as antagonists of ccr2
US8067415B2 (en) * 2005-11-01 2011-11-29 Millennium Pharmaceuticals, Inc. Compounds useful as antagonists of CCR2
GB0524786D0 (en) * 2005-12-05 2006-01-11 Glaxo Group Ltd Compounds
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