MXPA04010625A - Antagonista de receptor de taquicinina. - Google Patents
Antagonista de receptor de taquicinina.Info
- Publication number
- MXPA04010625A MXPA04010625A MXPA04010625A MXPA04010625A MXPA04010625A MX PA04010625 A MXPA04010625 A MX PA04010625A MX PA04010625 A MXPA04010625 A MX PA04010625A MX PA04010625 A MXPA04010625 A MX PA04010625A MX PA04010625 A MXPA04010625 A MX PA04010625A
- Authority
- MX
- Mexico
- Prior art keywords
- receptor antagonists
- tachykinin receptor
- tachykinin
- tachykinins
- selective
- Prior art date
Links
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- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
- C07D249/06—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
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- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
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- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Otolaryngology (AREA)
- Addiction (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
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Abstract
La presente invencion se refiere a antagonistas del receptor NK-1 selectivos de la Formula (I); o una sal farmaceuticamente aceptable del mismo, para el tratamiento de trastornos asociados con un exceso de taquicininas.(ver formula I).
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US37612102P | 2002-04-26 | 2002-04-26 | |
US44086503P | 2003-01-16 | 2003-01-16 | |
PCT/US2003/010682 WO2003091227A1 (en) | 2002-04-26 | 2003-04-22 | Tachykinin receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA04010625A true MXPA04010625A (es) | 2004-12-13 |
Family
ID=29273048
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA04010625A MXPA04010625A (es) | 2002-04-26 | 2003-04-22 | Antagonista de receptor de taquicinina. |
Country Status (16)
Country | Link |
---|---|
US (1) | US7179804B2 (es) |
EP (1) | EP1501808B1 (es) |
JP (1) | JP4895476B2 (es) |
CN (1) | CN1313450C (es) |
AT (1) | ATE399770T1 (es) |
BR (1) | BR0309486A (es) |
CA (1) | CA2484188C (es) |
CY (1) | CY1108539T1 (es) |
DE (1) | DE60321907D1 (es) |
DK (1) | DK1501808T3 (es) |
ES (1) | ES2307925T3 (es) |
IL (1) | IL164787A0 (es) |
MX (1) | MXPA04010625A (es) |
PT (1) | PT1501808E (es) |
SI (1) | SI1501808T1 (es) |
WO (1) | WO2003091227A1 (es) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1312136C (zh) * | 2002-04-26 | 2007-04-25 | 伊莱利利公司 | 用作速激肽受体拮抗剂的三唑衍生物 |
WO2005000821A1 (en) * | 2003-06-12 | 2005-01-06 | Eli Lilly And Company | Tachykinin receptor antagonists |
US7932272B2 (en) * | 2003-09-30 | 2011-04-26 | Eisai R&D Management Co., Ltd. | Antifungal agent containing heterocyclic compound |
US20050241110A1 (en) * | 2004-04-09 | 2005-11-03 | Bruce Baker | Ergonomic handles, especially for garden tools |
US20090227799A1 (en) * | 2004-08-09 | 2009-09-10 | Kazutaka Nakamoto | Novel Antimalarial Agent Containing Heterocyclic Compound |
EP1864980A4 (en) | 2005-03-30 | 2010-08-18 | Eisai R&D Man Co Ltd | A PYRIDINE DERIVATIVE ANTIPILIC AGENT |
TW200716576A (en) * | 2005-06-07 | 2007-05-01 | Shionogi & Co | Heterocyclic derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1 |
US20110060017A1 (en) * | 2008-03-11 | 2011-03-10 | Neurosearch A/S | Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
CA2616576A1 (en) * | 2005-07-25 | 2007-02-01 | F. Hoffman-La Roche Ag | Substituted triazole derivatives and their use as neurokinin 3 receptor antagonists |
TWI385169B (zh) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | 經雜環取代之吡啶衍生物及含有彼之抗真菌劑 |
EP1946840B1 (en) * | 2005-11-04 | 2019-08-21 | NGK Insulators, Ltd. | Honeycomb structure and honeycomb catalyst |
EP2065377B1 (en) * | 2006-09-21 | 2011-11-23 | Eisai R&D Management Co., Ltd. | Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same |
EP2143723A4 (en) * | 2007-04-27 | 2011-05-18 | Eisai R&D Man Co Ltd | SALT OF A PYRIDINE DERIVATIVE SUBSTITUTED BY HETEROCYCLE OR CRYSTALS OF THE SAME |
TW200841879A (en) * | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
RU2501787C2 (ru) * | 2007-11-02 | 2013-12-20 | Метилджен Инк. | Ингибиторы гистондеацетилазы |
US8513287B2 (en) | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
AU2009263037B2 (en) * | 2008-06-26 | 2011-10-06 | Amgen Inc. | Alkynyl alcohols as kinase inhibitors |
JP2011530495A (ja) * | 2008-08-08 | 2011-12-22 | ノイロサーチ アクティーゼルスカブ | ニコチン性アセチルコリン受容体のモジュレーターとして有用な新規のジフェニル1,2,3−トリアゾール誘導体 |
US8188119B2 (en) * | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
WO2011115817A1 (en) | 2010-03-16 | 2011-09-22 | Isis Pharmaceuticals, Inc. | Methods of preparing 2'-o-substituted purine nucleosides |
US9109005B2 (en) * | 2012-02-23 | 2015-08-18 | Boehringer Ingelheim International Gmbh | Method for manufacturing of ciclesonide |
CN103073513B (zh) * | 2012-12-14 | 2015-12-02 | 雅本化学股份有限公司 | 1-取代-5-氯-2h-1,2,3-三氮唑-4-羧酸衍生物及其制备方法 |
EP3265087B1 (en) * | 2015-03-04 | 2020-07-22 | Vanda Pharmaceuticals Inc. | Method of treatment with tradipitant |
KR20200054232A (ko) | 2017-09-13 | 2020-05-19 | 반다 파마슈티칼즈, 인코퍼레이티드. | 트라디피탄트를 이용한 아토피 피부염의 개선된 치료 |
CN108516942B (zh) * | 2018-03-12 | 2021-04-20 | 中国科学院成都有机化学有限公司 | 一种左旋盐酸米那普仑的制备方法 |
WO2023041779A1 (en) * | 2021-09-20 | 2023-03-23 | Novaled Gmbh | Metal complex, semiconductor layer comprising a metal complex and organic electronic device |
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IL50699A0 (en) | 1975-10-28 | 1976-12-31 | Ici America Inc | Triazole derivatives |
WO1995011880A1 (en) * | 1993-10-27 | 1995-05-04 | Merck Sharp & Dohme Limited | Substituted amides as tachykinin antagonists |
US6175013B1 (en) * | 1994-06-10 | 2001-01-16 | Eli Lilly And Company | Imidazolinyl tachykinin receptor antagonists |
US5998444A (en) * | 1995-10-24 | 1999-12-07 | Zeneca Ltd. | Piperidinyl compounds as NK1 or NK2 antagonists |
AU2633897A (en) | 1996-04-19 | 1997-11-12 | Novo Nordisk A/S | Solid phase and combinatorial synthesis of substituted 1,2,3-triazoles and of arrays of substituted 1,2,3-triazoles |
US6060478A (en) | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
TR200000291T2 (tr) * | 1997-08-06 | 2000-07-21 | Eli Lilly And Company | Taşikinin reseptör antagonistleri olarak 2-asilaminopropanaminler. |
ATE318259T1 (de) * | 1999-12-17 | 2006-03-15 | Schering Corp | Selektive neurokinin-antagonisten |
TWI287003B (en) | 2000-07-24 | 2007-09-21 | Hoffmann La Roche | 4-phenyl-pyridine derivatives |
DE10036818A1 (de) * | 2000-07-28 | 2002-02-07 | Solvay Pharm Gmbh | Neue N-Triazolylmethyl-Piperazinderivate als Neurokininrezeptor-Antagonisten |
JP2002123925A (ja) | 2000-10-13 | 2002-04-26 | Fuji Photo Film Co Ltd | 磁気記録媒体 |
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- 2003-04-22 BR BR0309486-3A patent/BR0309486A/pt not_active IP Right Cessation
- 2003-04-22 WO PCT/US2003/010682 patent/WO2003091227A1/en active Application Filing
- 2003-04-22 ES ES03721561T patent/ES2307925T3/es not_active Expired - Lifetime
- 2003-04-22 AT AT03721561T patent/ATE399770T1/de not_active IP Right Cessation
- 2003-04-22 US US10/512,248 patent/US7179804B2/en not_active Expired - Fee Related
- 2003-04-22 JP JP2003587787A patent/JP4895476B2/ja not_active Expired - Fee Related
- 2003-04-22 CN CNB03809360XA patent/CN1313450C/zh not_active Expired - Fee Related
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- 2003-04-22 MX MXPA04010625A patent/MXPA04010625A/es active IP Right Grant
- 2003-04-22 SI SI200331308T patent/SI1501808T1/sl unknown
- 2003-04-22 DK DK03721561T patent/DK1501808T3/da active
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EP1501808A1 (en) | 2005-02-02 |
CY1108539T1 (el) | 2012-05-23 |
US20050239776A1 (en) | 2005-10-27 |
ATE399770T1 (de) | 2008-07-15 |
JP2005534627A (ja) | 2005-11-17 |
EP1501808B1 (en) | 2008-07-02 |
CA2484188A1 (en) | 2003-11-06 |
US7179804B2 (en) | 2007-02-20 |
AU2003224868A1 (en) | 2003-11-10 |
PT1501808E (pt) | 2008-09-26 |
IL164787A0 (en) | 2005-12-18 |
DK1501808T3 (da) | 2008-10-13 |
CN1313450C (zh) | 2007-05-02 |
WO2003091227A1 (en) | 2003-11-06 |
AU2003224868B2 (en) | 2008-11-20 |
JP4895476B2 (ja) | 2012-03-14 |
BR0309486A (pt) | 2005-02-09 |
ES2307925T3 (es) | 2008-12-01 |
CA2484188C (en) | 2010-11-09 |
DE60321907D1 (de) | 2008-08-14 |
CN1649849A (zh) | 2005-08-03 |
SI1501808T1 (sl) | 2008-10-31 |
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