PT1245565E - Derivados de indenoindolonas processo para a sua preparacao e as composicoes farmaceuticas que os contem - Google Patents
Derivados de indenoindolonas processo para a sua preparacao e as composicoes farmaceuticas que os contemInfo
- Publication number
- PT1245565E PT1245565E PT02290668T PT02290668T PT1245565E PT 1245565 E PT1245565 E PT 1245565E PT 02290668 T PT02290668 T PT 02290668T PT 02290668 T PT02290668 T PT 02290668T PT 1245565 E PT1245565 E PT 1245565E
- Authority
- PT
- Portugal
- Prior art keywords
- indenoindolon
- contain
- preparation
- pharmaceutical compositions
- derivatives process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Reproductive Health (AREA)
- Emergency Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pregnancy & Childbirth (AREA)
- Anesthesiology (AREA)
- Psychology (AREA)
- Gynecology & Obstetrics (AREA)
- Child & Adolescent Psychology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0103667A FR2822153B1 (fr) | 2001-03-19 | 2001-03-19 | Nouveaux derives d'indenoindolones, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1245565E true PT1245565E (pt) | 2003-12-31 |
Family
ID=8861264
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT02290668T PT1245565E (pt) | 2001-03-19 | 2002-03-18 | Derivados de indenoindolonas processo para a sua preparacao e as composicoes farmaceuticas que os contem |
Country Status (24)
Country | Link |
---|---|
US (1) | US6844445B2 (pt) |
EP (1) | EP1245565B1 (pt) |
JP (1) | JP3886829B2 (pt) |
KR (1) | KR100453979B1 (pt) |
CN (1) | CN1185214C (pt) |
AR (1) | AR034861A1 (pt) |
AT (1) | ATE250578T1 (pt) |
AU (1) | AU780027B2 (pt) |
BR (1) | BR0200871A (pt) |
CA (1) | CA2378628C (pt) |
DE (1) | DE60200041T2 (pt) |
DK (1) | DK1245565T3 (pt) |
EA (1) | EA004711B1 (pt) |
ES (1) | ES2207629T3 (pt) |
FR (1) | FR2822153B1 (pt) |
HK (1) | HK1049159B (pt) |
HU (1) | HU226674B1 (pt) |
MX (1) | MXPA02002816A (pt) |
NO (1) | NO321890B1 (pt) |
NZ (1) | NZ517855A (pt) |
PL (1) | PL352866A1 (pt) |
PT (1) | PT1245565E (pt) |
SI (1) | SI1245565T1 (pt) |
ZA (1) | ZA200202220B (pt) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102006047231B4 (de) * | 2006-10-04 | 2009-02-12 | Hemmerling, Hans-Jörg, Dr. | Substituierte Indeno[1,2-b]indolderivate als neue Hemmstoffe der Protein Kinase CK2 und ihre Verwendung als Tumor Therapeutika, Cytostatika und Diagnostika |
JP4831077B2 (ja) * | 2008-01-15 | 2011-12-07 | 三菱電機株式会社 | 燃料圧力調整器およびそれを用いた燃料供給装置 |
ES2580702B1 (es) | 2015-02-25 | 2017-06-08 | Palobiofarma, S.L. | Derivados de 2-aminopiridina como antagonistas del receptor A2b de adenosina y ligandos del receptor MT3 de melatonina |
CA3073656C (en) | 2017-09-22 | 2024-03-05 | Jubilant Epipad LLC | Heterocyclic compounds as pad inhibitors |
CN111225915B (zh) | 2017-10-18 | 2023-03-07 | 朱比兰特埃皮帕德有限公司 | 作为pad抑制剂的咪唑并吡啶化合物 |
EP3707135A1 (en) | 2017-11-06 | 2020-09-16 | Jubilant Prodel LLC | Pyrimidine derivatives as inhibitors of pd1/pd-l1 activation |
BR112020010322A2 (pt) | 2017-11-24 | 2020-11-17 | Jubilant Episcribe Llc | composto da fórmula i; composto da fórmula ia; composto da fórmula ib; processo de preparação de compostos da fórmula i; composição farmacêutica; método para o tratamento e/ou prevenção de várias doenças; uso dos compostos; método para o tratamento de câncer; e método para o tratamento e/ou prevenção de uma afecção mediada por prmt5 ou um distúrbio proliferativo ou câncer |
SG11202008950PA (en) | 2018-03-13 | 2020-10-29 | Jubilant Prodel LLC | Bicyclic compounds as inhibitors of pd1/pd-l1 interaction/activation |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL99750A0 (en) * | 1990-10-16 | 1992-08-18 | Univ Bath | Indenoindole compounds |
-
2001
- 2001-03-19 FR FR0103667A patent/FR2822153B1/fr not_active Expired - Fee Related
-
2002
- 2002-03-14 MX MXPA02002816A patent/MXPA02002816A/es active IP Right Grant
- 2002-03-18 AT AT02290668T patent/ATE250578T1/de not_active IP Right Cessation
- 2002-03-18 PT PT02290668T patent/PT1245565E/pt unknown
- 2002-03-18 AR ARP020100952A patent/AR034861A1/es unknown
- 2002-03-18 NO NO20021330A patent/NO321890B1/no not_active IP Right Cessation
- 2002-03-18 SI SI200230003T patent/SI1245565T1/xx unknown
- 2002-03-18 EP EP02290668A patent/EP1245565B1/fr not_active Expired - Lifetime
- 2002-03-18 NZ NZ517855A patent/NZ517855A/xx unknown
- 2002-03-18 CN CNB021075778A patent/CN1185214C/zh not_active Expired - Fee Related
- 2002-03-18 JP JP2002073851A patent/JP3886829B2/ja not_active Expired - Fee Related
- 2002-03-18 DK DK02290668T patent/DK1245565T3/da active
- 2002-03-18 ES ES02290668T patent/ES2207629T3/es not_active Expired - Lifetime
- 2002-03-18 DE DE60200041T patent/DE60200041T2/de not_active Expired - Fee Related
- 2002-03-18 EA EA200200263A patent/EA004711B1/ru unknown
- 2002-03-19 KR KR10-2002-0014738A patent/KR100453979B1/ko not_active IP Right Cessation
- 2002-03-19 BR BR0200871-8A patent/BR0200871A/pt not_active IP Right Cessation
- 2002-03-19 US US10/100,784 patent/US6844445B2/en not_active Expired - Fee Related
- 2002-03-19 HU HU0201024A patent/HU226674B1/hu not_active IP Right Cessation
- 2002-03-19 CA CA002378628A patent/CA2378628C/fr not_active Expired - Fee Related
- 2002-03-19 PL PL02352866A patent/PL352866A1/xx not_active IP Right Cessation
- 2002-03-19 ZA ZA200202220A patent/ZA200202220B/xx unknown
- 2002-03-19 AU AU27469/02A patent/AU780027B2/en not_active Ceased
-
2003
- 2003-02-18 HK HK03101148.6A patent/HK1049159B/zh not_active IP Right Cessation
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