PT1411057E - Derivados de [3,4-a:3,4-c]carbazole processo para a sua preparacao e as composicoes farmaceuticas que os contem - Google Patents

Derivados de [3,4-a:3,4-c]carbazole processo para a sua preparacao e as composicoes farmaceuticas que os contem

Info

Publication number
PT1411057E
PT1411057E PT03292545T PT03292545T PT1411057E PT 1411057 E PT1411057 E PT 1411057E PT 03292545 T PT03292545 T PT 03292545T PT 03292545 T PT03292545 T PT 03292545T PT 1411057 E PT1411057 E PT 1411057E
Authority
PT
Portugal
Prior art keywords
contain
preparation
pharmaceutical compositions
carbazole derivatives
derivatives process
Prior art date
Application number
PT03292545T
Other languages
English (en)
Inventor
Alain Pierre
Bruno Pfeiffer
Pierre Renard
Michelle Prudhomme
Fabrice Anizon
John Hickman
Hugon Bernadette
Golsteyn Roy
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of PT1411057E publication Critical patent/PT1411057E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/23Heterocyclic radicals containing two or more heterocyclic rings condensed among themselves or condensed with a common carbocyclic ring system, not provided for in groups C07H19/14 - C07H19/22
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT03292545T 2002-10-16 2003-10-14 Derivados de [3,4-a:3,4-c]carbazole processo para a sua preparacao e as composicoes farmaceuticas que os contem PT1411057E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0212847A FR2845996A1 (fr) 2002-10-16 2002-10-16 Nouveaux derives de[3,4-a:3,4-c]carbazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
PT1411057E true PT1411057E (pt) 2005-08-31

Family

ID=29725330

Family Applications (1)

Application Number Title Priority Date Filing Date
PT03292545T PT1411057E (pt) 2002-10-16 2003-10-14 Derivados de [3,4-a:3,4-c]carbazole processo para a sua preparacao e as composicoes farmaceuticas que os contem

Country Status (26)

Country Link
US (1) US7151108B2 (pt)
EP (1) EP1411057B1 (pt)
JP (1) JP2004277404A (pt)
KR (1) KR100502250B1 (pt)
CN (1) CN1241925C (pt)
AR (1) AR041618A1 (pt)
AT (1) ATE294181T1 (pt)
AU (1) AU2003254746A1 (pt)
BR (1) BR0304575A (pt)
CA (1) CA2443585A1 (pt)
DE (1) DE60300571T2 (pt)
DK (1) DK1411057T3 (pt)
EA (1) EA007250B1 (pt)
ES (1) ES2240927T3 (pt)
FR (1) FR2845996A1 (pt)
HK (1) HK1063321A1 (pt)
MA (1) MA27007A1 (pt)
MX (1) MXPA03009362A (pt)
MY (1) MY134620A (pt)
NO (1) NO20034614L (pt)
NZ (1) NZ528902A (pt)
PL (1) PL362885A1 (pt)
PT (1) PT1411057E (pt)
SG (1) SG131765A1 (pt)
SI (1) SI1411057T1 (pt)
ZA (1) ZA200308053B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI499414B (zh) 2006-09-29 2015-09-11 Lexicon Pharmaceuticals Inc 鈉與葡萄糖第2型共同運輸體(co-transporter 2)的抑制物與其應用方法
US7846945B2 (en) 2007-03-08 2010-12-07 Lexicon Pharmaceuticals, Inc. Piperdine-based inhibitors of sodium glucose co-transporter 2 and methods of their use
CA2939164A1 (en) 2014-02-12 2015-08-20 Iteos Therapeutics Novel 3-(indol-3-yl)-pyridine derivatives, pharmaceutical compositions and methods for use
CN103804278B (zh) * 2014-02-19 2016-04-13 西北大学 一种天然产物2-甲基-3-甲氧基-咔唑-1,4-苯醌的制备方法
EA201650031A1 (ru) * 2014-05-15 2017-06-30 Итеос Терапьютик Производные пирролидин-2,5-диона, фармацевтические композиции и способы применения в качестве ингибиторов ido1
SG11201706992TA (en) 2015-03-17 2017-09-28 Pfizer Novel 3-indol substituted derivatives, pharmaceutical compositions and methods for use
JP2016216446A (ja) * 2015-05-14 2016-12-22 ファイザー・インク ピロリジン−2,5−ジオン誘導体の多形形態、医薬組成物、およびido1阻害薬としての使用方法
JP2018527336A (ja) 2015-08-10 2018-09-20 ファイザー・インク 3−インドール置換誘導体、医薬組成物、および使用方法
CN106832175B (zh) * 2017-02-17 2019-10-18 华南理工大学 一种基于咔唑衍生物的双羟基荧光扩链剂及其制备与应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3010675B2 (ja) * 1989-03-23 2000-02-21 萬有製薬株式会社 抗腫瘍性物質be―13793c

Also Published As

Publication number Publication date
KR20040034472A (ko) 2004-04-28
AU2003254746A1 (en) 2004-05-06
SG131765A1 (en) 2007-05-28
NO20034614L (no) 2004-04-19
EP1411057B1 (fr) 2005-04-27
CN1496989A (zh) 2004-05-19
MA27007A1 (fr) 2004-12-20
DE60300571D1 (de) 2005-06-02
EA007250B1 (ru) 2006-08-25
PL362885A1 (en) 2004-04-19
HK1063321A1 (en) 2004-12-24
ATE294181T1 (de) 2005-05-15
DK1411057T3 (da) 2005-08-29
ES2240927T3 (es) 2005-10-16
ZA200308053B (en) 2004-07-08
NZ528902A (en) 2004-09-24
CN1241925C (zh) 2006-02-15
FR2845996A1 (fr) 2004-04-23
US7151108B2 (en) 2006-12-19
NO20034614D0 (no) 2003-10-15
MY134620A (en) 2007-12-31
BR0304575A (pt) 2004-07-20
DE60300571T2 (de) 2006-02-23
KR100502250B1 (ko) 2005-07-20
EA200301020A1 (ru) 2004-04-29
CA2443585A1 (fr) 2004-04-16
US20040077672A1 (en) 2004-04-22
SI1411057T1 (pt) 2005-08-31
JP2004277404A (ja) 2004-10-07
AR041618A1 (es) 2005-05-26
EP1411057A1 (fr) 2004-04-21
MXPA03009362A (es) 2004-04-28

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