PL91512B1 - - Google Patents

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Publication number
PL91512B1
PL91512B1 PL1974173564A PL17356474A PL91512B1 PL 91512 B1 PL91512 B1 PL 91512B1 PL 1974173564 A PL1974173564 A PL 1974173564A PL 17356474 A PL17356474 A PL 17356474A PL 91512 B1 PL91512 B1 PL 91512B1
Authority
PL
Poland
Prior art keywords
acid
pyridyl
formula
compounds
hydrochloride
Prior art date
Application number
PL1974173564A
Other languages
English (en)
Polish (pl)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of PL91512B1 publication Critical patent/PL91512B1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
PL1974173564A 1973-08-20 1974-08-19 PL91512B1 (instruction)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2341965A DE2341965C3 (de) 1973-08-20 1973-08-20 4- [N- (o-PyridyD- N-acyl] -aminolphenäthylpiperidine, Verfahren zu deren Herstellung sowie deren Verwendung bei der Bekämpfung von Schmerzzuständen

Publications (1)

Publication Number Publication Date
PL91512B1 true PL91512B1 (instruction) 1977-02-28

Family

ID=5890196

Family Applications (2)

Application Number Title Priority Date Filing Date
PL1974173565A PL91562B1 (instruction) 1973-08-20 1974-08-19
PL1974173564A PL91512B1 (instruction) 1973-08-20 1974-08-19

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PL1974173565A PL91562B1 (instruction) 1973-08-20 1974-08-19

Country Status (26)

Country Link
US (1) US3933832A (instruction)
JP (1) JPS5049285A (instruction)
AT (2) AT334901B (instruction)
BE (1) BE818989A (instruction)
BG (1) BG24669A3 (instruction)
CA (1) CA1041513A (instruction)
CH (2) CH603631A5 (instruction)
CS (2) CS181767B2 (instruction)
DD (1) DD114260A5 (instruction)
DE (1) DE2341965C3 (instruction)
DK (1) DK141097C (instruction)
ES (2) ES429234A1 (instruction)
FI (1) FI57749C (instruction)
FR (1) FR2241314B1 (instruction)
GB (1) GB1468283A (instruction)
HU (1) HU167563B (instruction)
IE (1) IE40511B1 (instruction)
IL (1) IL45494A (instruction)
NL (1) NL7410989A (instruction)
NO (1) NO140594C (instruction)
PH (1) PH11999A (instruction)
PL (2) PL91562B1 (instruction)
RO (2) RO63458A (instruction)
SE (1) SE402285B (instruction)
SU (2) SU507229A3 (instruction)
ZA (1) ZA745306B (instruction)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4191683A (en) * 1975-05-28 1980-03-04 Ciba-Geigy Corporation Derivatives of 4-aminopiperidine as stabilizers for polymers
US4225606A (en) * 1975-09-23 1980-09-30 Janssen Pharmaceutica N.V. N-Aryl-N-(1-L-4-piperidinyl)arylacetamides
US4791112A (en) * 1987-02-02 1988-12-13 The Boc Group, Inc. N-heterocyclic-N-(4-piperidyl)amides and pharmaceutical compositions and methods employing such compounds
USRE34201E (en) * 1989-04-20 1993-03-23 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
PT1379520E (pt) 2001-02-23 2006-08-31 Merck & Co Inc Antagonistas (nao-aril)-heterociclicos n-substituidos de nmda/nr2b
US20040142013A1 (en) * 2001-07-13 2004-07-22 Flow Focusing, Inc. Implantable orthopedic surgical devices with controlled release antimicrobial component
US20030055075A1 (en) * 2001-07-13 2003-03-20 Rubsamen Reid M. Programmable controlled release injectable opioid formulation
US20060263401A1 (en) * 2001-07-13 2006-11-23 Flow Focusing, Inc. Formulation and Method for Preventing Infection
US20070254009A1 (en) * 2001-07-13 2007-11-01 Flow Focusing, Inc. Antibiotic/bone morphogenic protein formulation and method of treatment
US20070254008A1 (en) * 2001-07-13 2007-11-01 Flow Focusing, Inc. Antibiotic formulation and method of treatment
US7592360B2 (en) * 2003-06-04 2009-09-22 Merck & Co., Inc. 3-fluoro-piperidines as NMDA/NR2B antagonists
JO2769B1 (en) 2005-10-26 2014-03-15 جانسين فارماسوتيكا ان. في Rapid decomposition of physiologically antagonistic agents of the 2-dopamine receptor
JO2642B1 (en) * 2006-12-08 2012-06-17 جانسين فارماسوتيكا ان. في Dopamine 2 receptor antagonists are rapidly hydrolyzed
JO2849B1 (en) 2007-02-13 2015-03-15 جانسين فارماسوتيكا ان. في Dopamine 2 receptor antagonists are rapidly hydrolyzed
JP2010525013A (ja) * 2007-04-23 2010-07-22 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 高速解離性ドパミン2受容体アンタゴニストとしてのピリジン誘導体
US8906921B2 (en) * 2007-04-23 2014-12-09 Janssen Pharmaceutica Nv 4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists
US8933101B2 (en) * 2007-04-23 2015-01-13 Janssen Pharmaceutica Nv Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists
CN102159554B (zh) * 2008-07-03 2014-09-24 詹森药业有限公司 作为5-ht6受体拮抗剂的取代的6-(1-哌嗪基)-哒嗪
WO2010012758A1 (en) * 2008-07-31 2010-02-04 Janssen Pharmaceutica Nv Piperazin-1-yl-trifluoromethyl-substituted-pyridines as fast dissociating dopamine 2 receptor antagonists

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1232147B (de) * 1961-04-13 1967-01-12 Bayer Ag Verfahren zur Herstellung von acylierten N-(Alkylaminoalkyl)-aminopyridinen
NL284196A (instruction) * 1961-10-10
US3141823A (en) * 1962-09-04 1964-07-21 Res Lab Dr C Janssen N V Method for producing analgesia
IL25840A (en) * 1965-07-24 1969-12-31 Bayer Ag Optically active pyridine derivatives and their production

Also Published As

Publication number Publication date
ATA651374A (de) 1976-06-15
BG24669A3 (bg) 1978-04-12
ZA745306B (en) 1976-04-28
AT334901B (de) 1977-02-10
NO140594C (no) 1979-10-03
CS181767B2 (en) 1978-03-31
PL91562B1 (instruction) 1977-03-31
DK141097B (da) 1980-01-14
ES429221A1 (es) 1976-08-16
ES429234A1 (es) 1976-08-16
DE2341965B2 (de) 1978-06-01
NO742970L (instruction) 1975-03-17
CH603631A5 (instruction) 1978-08-31
RO63458A (fr) 1978-06-15
FR2241314A1 (instruction) 1975-03-21
PH11999A (en) 1978-10-06
DE2341965C3 (de) 1979-01-25
GB1468283A (en) 1977-03-23
DE2341965A1 (de) 1975-03-06
AT334900B (de) 1977-02-10
SU504480A3 (ru) 1976-02-25
SE7410540L (instruction) 1975-02-21
FI57749C (fi) 1980-10-10
CS182263B2 (en) 1978-04-28
IL45494A (en) 1977-07-31
CH603630A5 (instruction) 1978-08-31
IL45494A0 (en) 1974-11-29
SE402285B (sv) 1978-06-26
IE40511L (en) 1975-02-20
NO140594B (no) 1979-06-25
AU7248974A (en) 1976-02-19
BE818989A (fr) 1975-02-19
IE40511B1 (en) 1979-06-20
DK439974A (instruction) 1975-04-28
RO63050A (instruction) 1978-05-15
SU507229A3 (ru) 1976-03-15
FI234974A7 (instruction) 1975-02-21
NL7410989A (nl) 1975-02-24
US3933832A (en) 1976-01-20
FI57749B (fi) 1980-06-30
HU167563B (instruction) 1975-11-28
FR2241314B1 (instruction) 1977-11-10
DK141097C (da) 1980-08-18
CA1041513A (en) 1978-10-31
ATA651274A (de) 1976-06-15
JPS5049285A (instruction) 1975-05-01
DD114260A5 (instruction) 1975-07-20

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