BE818989A - Amides n -(1-(omega)-phenylalcoyl-piperidyl-4)-n -(alpha -pyriyl)- carboxyliques, leurs sels d'addition d'acide, leur procede de preparation et leur application comme medicaments - Google Patents
Amides n -(1-(omega)-phenylalcoyl-piperidyl-4)-n -(alpha -pyriyl)- carboxyliques, leurs sels d'addition d'acide, leur procede de preparation et leur application comme medicamentsInfo
- Publication number
- BE818989A BE818989A BE147736A BE147736A BE818989A BE 818989 A BE818989 A BE 818989A BE 147736 A BE147736 A BE 147736A BE 147736 A BE147736 A BE 147736A BE 818989 A BE818989 A BE 818989A
- Authority
- BE
- Belgium
- Prior art keywords
- phenylalcoyl
- pyriyl
- carboxylics
- piperidyl
- omega
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE2341965A DE2341965C3 (de) | 1973-08-20 | 1973-08-20 | 4- [N- (o-PyridyD- N-acyl] -aminolphenäthylpiperidine, Verfahren zu deren Herstellung sowie deren Verwendung bei der Bekämpfung von Schmerzzuständen |
Publications (1)
Publication Number | Publication Date |
---|---|
BE818989A true BE818989A (fr) | 1975-02-19 |
Family
ID=5890196
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE147736A BE818989A (fr) | 1973-08-20 | 1974-08-19 | Amides n -(1-(omega)-phenylalcoyl-piperidyl-4)-n -(alpha -pyriyl)- carboxyliques, leurs sels d'addition d'acide, leur procede de preparation et leur application comme medicaments |
Country Status (26)
Country | Link |
---|---|
US (1) | US3933832A (fr) |
JP (1) | JPS5049285A (fr) |
AT (2) | AT334900B (fr) |
BE (1) | BE818989A (fr) |
BG (1) | BG24669A3 (fr) |
CA (1) | CA1041513A (fr) |
CH (2) | CH603630A5 (fr) |
CS (2) | CS181767B2 (fr) |
DD (1) | DD114260A5 (fr) |
DE (1) | DE2341965C3 (fr) |
DK (1) | DK141097C (fr) |
ES (2) | ES429234A1 (fr) |
FI (1) | FI57749C (fr) |
FR (1) | FR2241314B1 (fr) |
GB (1) | GB1468283A (fr) |
HU (1) | HU167563B (fr) |
IE (1) | IE40511B1 (fr) |
IL (1) | IL45494A (fr) |
NL (1) | NL7410989A (fr) |
NO (1) | NO140594C (fr) |
PH (1) | PH11999A (fr) |
PL (2) | PL91562B1 (fr) |
RO (2) | RO63050A (fr) |
SE (1) | SE402285B (fr) |
SU (2) | SU504480A3 (fr) |
ZA (1) | ZA745306B (fr) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4191683A (en) * | 1975-05-28 | 1980-03-04 | Ciba-Geigy Corporation | Derivatives of 4-aminopiperidine as stabilizers for polymers |
US4225606A (en) * | 1975-09-23 | 1980-09-30 | Janssen Pharmaceutica N.V. | N-Aryl-N-(1-L-4-piperidinyl)arylacetamides |
US4791112A (en) * | 1987-02-02 | 1988-12-13 | The Boc Group, Inc. | N-heterocyclic-N-(4-piperidyl)amides and pharmaceutical compositions and methods employing such compounds |
USRE34201E (en) * | 1989-04-20 | 1993-03-23 | Anaquest, Inc. | N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds |
NZ527365A (en) | 2001-02-23 | 2005-08-26 | Merck & Co Inc | N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists |
US20060263401A1 (en) * | 2001-07-13 | 2006-11-23 | Flow Focusing, Inc. | Formulation and Method for Preventing Infection |
US20030055075A1 (en) * | 2001-07-13 | 2003-03-20 | Rubsamen Reid M. | Programmable controlled release injectable opioid formulation |
US20040142013A1 (en) * | 2001-07-13 | 2004-07-22 | Flow Focusing, Inc. | Implantable orthopedic surgical devices with controlled release antimicrobial component |
US20070254009A1 (en) * | 2001-07-13 | 2007-11-01 | Flow Focusing, Inc. | Antibiotic/bone morphogenic protein formulation and method of treatment |
US20070254008A1 (en) * | 2001-07-13 | 2007-11-01 | Flow Focusing, Inc. | Antibiotic formulation and method of treatment |
US7592360B2 (en) * | 2003-06-04 | 2009-09-22 | Merck & Co., Inc. | 3-fluoro-piperidines as NMDA/NR2B antagonists |
JO2769B1 (en) | 2005-10-26 | 2014-03-15 | جانسين فارماسوتيكا ان. في | Rapid decomposition of physiologically antagonistic agents of the 2-dopamine receptor |
JO2642B1 (en) * | 2006-12-08 | 2012-06-17 | جانسين فارماسوتيكا ان. في | Dopamine 2 receptor antagonists are rapidly hydrolyzed |
JO2849B1 (en) | 2007-02-13 | 2015-03-15 | جانسين فارماسوتيكا ان. في | Dopamine 2 receptor antagonists are rapidly hydrolyzed |
CA2682668A1 (fr) * | 2007-04-23 | 2008-10-30 | Janssen Pharmaceutica N.V. | Derives de pyridine comme antagonistes des recepteurs d2 de la dopamine a dissociation rapide |
US8933101B2 (en) * | 2007-04-23 | 2015-01-13 | Janssen Pharmaceutica Nv | Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists |
SI2148873T1 (sl) * | 2007-04-23 | 2013-01-31 | Janssen Pharmaceutica, N.V. | Derivati 4-alkoksipiridazina kot antagonisti receptorja dopamina 2 s hitro disociacijo |
US8530474B2 (en) * | 2008-07-03 | 2013-09-10 | Janssen Pharmaceutica Nv | Substituted 6-(1-piperazinyl)-pyridazines as 5-HT6 receptor antagonists |
CA2730774C (fr) * | 2008-07-31 | 2016-09-13 | Janssen Pharmaceutica Nv | Pyridines substituees par piperazin-1-yl-trifluoromethyle en tant qu'antagonistes des recepteurs d2 de la dopamine a dissociation rapide |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1232147B (de) * | 1961-04-13 | 1967-01-12 | Bayer Ag | Verfahren zur Herstellung von acylierten N-(Alkylaminoalkyl)-aminopyridinen |
NL135583C (fr) * | 1961-10-10 | |||
US3141823A (en) * | 1962-09-04 | 1964-07-21 | Res Lab Dr C Janssen N V | Method for producing analgesia |
IL25840A (en) * | 1965-07-24 | 1969-12-31 | Bayer Ag | Optically active pyridine derivatives and their production |
-
1973
- 1973-08-20 DE DE2341965A patent/DE2341965C3/de not_active Expired
-
1974
- 1974-07-31 CS CS7400005454A patent/CS181767B2/cs unknown
- 1974-07-31 CS CS7400005455A patent/CS182263B2/cs unknown
- 1974-08-07 FI FI2349/74A patent/FI57749C/fi active
- 1974-08-08 AT AT651274A patent/AT334900B/de not_active IP Right Cessation
- 1974-08-08 AT AT651374A patent/AT334901B/de not_active IP Right Cessation
- 1974-08-13 ES ES429234A patent/ES429234A1/es not_active Expired
- 1974-08-13 ES ES429221A patent/ES429221A1/es not_active Expired
- 1974-08-14 US US05/497,455 patent/US3933832A/en not_active Expired - Lifetime
- 1974-08-15 PH PH16171A patent/PH11999A/en unknown
- 1974-08-16 SU SU2055577A patent/SU504480A3/ru active
- 1974-08-16 RO RO7400079806A patent/RO63050A/ro unknown
- 1974-08-16 CH CH1118674A patent/CH603630A5/xx not_active IP Right Cessation
- 1974-08-16 DK DK439974A patent/DK141097C/da active
- 1974-08-16 SU SU2056122A patent/SU507229A3/ru active
- 1974-08-16 CH CH1119074A patent/CH603631A5/xx not_active IP Right Cessation
- 1974-08-16 NL NL7410989A patent/NL7410989A/xx not_active Application Discontinuation
- 1974-08-16 BG BG7400027507A patent/BG24669A3/xx unknown
- 1974-08-16 RO RO7400079805A patent/RO63458A/fr unknown
- 1974-08-17 HU HUBO1516A patent/HU167563B/hu unknown
- 1974-08-19 PL PL1974173565A patent/PL91562B1/pl unknown
- 1974-08-19 SE SE7410540A patent/SE402285B/xx unknown
- 1974-08-19 IL IL45494A patent/IL45494A/en unknown
- 1974-08-19 DD DD180589A patent/DD114260A5/xx unknown
- 1974-08-19 ZA ZA00745306A patent/ZA745306B/xx unknown
- 1974-08-19 PL PL1974173564A patent/PL91512B1/pl unknown
- 1974-08-19 CA CA207,296A patent/CA1041513A/fr not_active Expired
- 1974-08-19 GB GB3645574A patent/GB1468283A/en not_active Expired
- 1974-08-19 JP JP49094904A patent/JPS5049285A/ja active Pending
- 1974-08-19 BE BE147736A patent/BE818989A/fr unknown
- 1974-08-19 NO NO742970A patent/NO140594C/no unknown
- 1974-08-20 IE IE1734/74A patent/IE40511B1/xx unknown
- 1974-08-20 FR FR7428596A patent/FR2241314B1/fr not_active Expired
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