CS181767B2 - Method of producing new amides n-(1-(u phenylalkyl)-piperidyl-4)-n-/alfa-pyridyl/carboxylic acid - Google Patents
Method of producing new amides n-(1-(u phenylalkyl)-piperidyl-4)-n-/alfa-pyridyl/carboxylic acidInfo
- Publication number
- CS181767B2 CS181767B2 CS7400005454A CS545474A CS181767B2 CS 181767 B2 CS181767 B2 CS 181767B2 CS 7400005454 A CS7400005454 A CS 7400005454A CS 545474 A CS545474 A CS 545474A CS 181767 B2 CS181767 B2 CS 181767B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- phenylalkyl
- alfa
- piperidyl
- pyridyl
- carboxylic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE2341965A DE2341965C3 (de) | 1973-08-20 | 1973-08-20 | 4- [N- (o-PyridyD- N-acyl] -aminolphenäthylpiperidine, Verfahren zu deren Herstellung sowie deren Verwendung bei der Bekämpfung von Schmerzzuständen |
Publications (1)
Publication Number | Publication Date |
---|---|
CS181767B2 true CS181767B2 (en) | 1978-03-31 |
Family
ID=5890196
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS7400005455A CS182263B2 (en) | 1973-08-20 | 1974-07-31 | Method of producing new amides of n-(1-w-phenylalkyl/-piperidyl-4)-n-/alfa-pyridyl/-carboxylic acid |
CS7400005454A CS181767B2 (en) | 1973-08-20 | 1974-07-31 | Method of producing new amides n-(1-(u phenylalkyl)-piperidyl-4)-n-/alfa-pyridyl/carboxylic acid |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS7400005455A CS182263B2 (en) | 1973-08-20 | 1974-07-31 | Method of producing new amides of n-(1-w-phenylalkyl/-piperidyl-4)-n-/alfa-pyridyl/-carboxylic acid |
Country Status (26)
Country | Link |
---|---|
US (1) | US3933832A (fr) |
JP (1) | JPS5049285A (fr) |
AT (2) | AT334900B (fr) |
BE (1) | BE818989A (fr) |
BG (1) | BG24669A3 (fr) |
CA (1) | CA1041513A (fr) |
CH (2) | CH603630A5 (fr) |
CS (2) | CS182263B2 (fr) |
DD (1) | DD114260A5 (fr) |
DE (1) | DE2341965C3 (fr) |
DK (1) | DK141097C (fr) |
ES (2) | ES429221A1 (fr) |
FI (1) | FI57749C (fr) |
FR (1) | FR2241314B1 (fr) |
GB (1) | GB1468283A (fr) |
HU (1) | HU167563B (fr) |
IE (1) | IE40511B1 (fr) |
IL (1) | IL45494A (fr) |
NL (1) | NL7410989A (fr) |
NO (1) | NO140594C (fr) |
PH (1) | PH11999A (fr) |
PL (2) | PL91512B1 (fr) |
RO (2) | RO63458A (fr) |
SE (1) | SE402285B (fr) |
SU (2) | SU504480A3 (fr) |
ZA (1) | ZA745306B (fr) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4191683A (en) * | 1975-05-28 | 1980-03-04 | Ciba-Geigy Corporation | Derivatives of 4-aminopiperidine as stabilizers for polymers |
US4225606A (en) * | 1975-09-23 | 1980-09-30 | Janssen Pharmaceutica N.V. | N-Aryl-N-(1-L-4-piperidinyl)arylacetamides |
US4791112A (en) * | 1987-02-02 | 1988-12-13 | The Boc Group, Inc. | N-heterocyclic-N-(4-piperidyl)amides and pharmaceutical compositions and methods employing such compounds |
USRE34201E (en) * | 1989-04-20 | 1993-03-23 | Anaquest, Inc. | N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds |
PT1379520E (pt) * | 2001-02-23 | 2006-08-31 | Merck & Co Inc | Antagonistas (nao-aril)-heterociclicos n-substituidos de nmda/nr2b |
US20040142013A1 (en) * | 2001-07-13 | 2004-07-22 | Flow Focusing, Inc. | Implantable orthopedic surgical devices with controlled release antimicrobial component |
US20070254008A1 (en) * | 2001-07-13 | 2007-11-01 | Flow Focusing, Inc. | Antibiotic formulation and method of treatment |
US20070254009A1 (en) * | 2001-07-13 | 2007-11-01 | Flow Focusing, Inc. | Antibiotic/bone morphogenic protein formulation and method of treatment |
US20030055075A1 (en) * | 2001-07-13 | 2003-03-20 | Rubsamen Reid M. | Programmable controlled release injectable opioid formulation |
US20060263401A1 (en) * | 2001-07-13 | 2006-11-23 | Flow Focusing, Inc. | Formulation and Method for Preventing Infection |
US7592360B2 (en) * | 2003-06-04 | 2009-09-22 | Merck & Co., Inc. | 3-fluoro-piperidines as NMDA/NR2B antagonists |
JO2769B1 (en) * | 2005-10-26 | 2014-03-15 | جانسين فارماسوتيكا ان. في | Rapid decomposition of physiologically antagonistic agents of the 2-dopamine receptor |
JO2642B1 (en) * | 2006-12-08 | 2012-06-17 | جانسين فارماسوتيكا ان. في | Dopamine 2 receptor antagonists are rapidly hydrolyzed |
JO2849B1 (en) * | 2007-02-13 | 2015-03-15 | جانسين فارماسوتيكا ان. في | Dopamine 2 receptor antagonists are rapidly hydrolyzed |
US20100137368A1 (en) * | 2007-04-23 | 2010-06-03 | Janssen Pharmaceutica N.V. | Pyridine derivatives as fast dissociating dopamine 2 receptor antagonists |
EP2148879B1 (fr) * | 2007-04-23 | 2012-11-28 | Janssen Pharmaceutica, N.V. | Thia(dia)zoles en tant qu'antagonistes du récepteur de la dopamine à dissociation rapide |
US8906921B2 (en) * | 2007-04-23 | 2014-12-09 | Janssen Pharmaceutica Nv | 4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists |
MX2011000043A (es) * | 2008-07-03 | 2011-02-22 | Janssen Pharmaceutica Nv | 6-(1-piperazinil)-piridazinas sustituidas como antagonistas del receptor 5-ht6. |
EP2307374B1 (fr) * | 2008-07-31 | 2017-01-25 | Janssen Pharmaceutica NV | Pyridines à substitution pipérazin-1-yl-trifluorométhyle en tant qu'antagonistes du récepteur de la dopamine 2 à dissociation rapide |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1232147B (de) * | 1961-04-13 | 1967-01-12 | Bayer Ag | Verfahren zur Herstellung von acylierten N-(Alkylaminoalkyl)-aminopyridinen |
NL284196A (fr) * | 1961-10-10 | |||
US3141823A (en) * | 1962-09-04 | 1964-07-21 | Res Lab Dr C Janssen N V | Method for producing analgesia |
IL25840A (en) * | 1965-07-24 | 1969-12-31 | Bayer Ag | Optically active pyridine derivatives and their production |
-
1973
- 1973-08-20 DE DE2341965A patent/DE2341965C3/de not_active Expired
-
1974
- 1974-07-31 CS CS7400005455A patent/CS182263B2/cs unknown
- 1974-07-31 CS CS7400005454A patent/CS181767B2/cs unknown
- 1974-08-07 FI FI2349/74A patent/FI57749C/fi active
- 1974-08-08 AT AT651274A patent/AT334900B/de not_active IP Right Cessation
- 1974-08-08 AT AT651374A patent/AT334901B/de not_active IP Right Cessation
- 1974-08-13 ES ES429221A patent/ES429221A1/es not_active Expired
- 1974-08-13 ES ES429234A patent/ES429234A1/es not_active Expired
- 1974-08-14 US US05/497,455 patent/US3933832A/en not_active Expired - Lifetime
- 1974-08-15 PH PH16171A patent/PH11999A/en unknown
- 1974-08-16 DK DK439974A patent/DK141097C/da active
- 1974-08-16 NL NL7410989A patent/NL7410989A/xx not_active Application Discontinuation
- 1974-08-16 CH CH1118674A patent/CH603630A5/xx not_active IP Right Cessation
- 1974-08-16 SU SU2055577A patent/SU504480A3/ru active
- 1974-08-16 CH CH1119074A patent/CH603631A5/xx not_active IP Right Cessation
- 1974-08-16 RO RO7400079805A patent/RO63458A/fr unknown
- 1974-08-16 RO RO7400079806A patent/RO63050A/ro unknown
- 1974-08-16 BG BG7400027507A patent/BG24669A3/xx unknown
- 1974-08-16 SU SU2056122A patent/SU507229A3/ru active
- 1974-08-17 HU HUBO1516A patent/HU167563B/hu unknown
- 1974-08-19 GB GB3645574A patent/GB1468283A/en not_active Expired
- 1974-08-19 BE BE147736A patent/BE818989A/fr unknown
- 1974-08-19 PL PL1974173564A patent/PL91512B1/pl unknown
- 1974-08-19 PL PL1974173565A patent/PL91562B1/pl unknown
- 1974-08-19 NO NO742970A patent/NO140594C/no unknown
- 1974-08-19 SE SE7410540A patent/SE402285B/xx unknown
- 1974-08-19 ZA ZA00745306A patent/ZA745306B/xx unknown
- 1974-08-19 IL IL45494A patent/IL45494A/en unknown
- 1974-08-19 DD DD180589A patent/DD114260A5/xx unknown
- 1974-08-19 JP JP49094904A patent/JPS5049285A/ja active Pending
- 1974-08-19 CA CA207,296A patent/CA1041513A/fr not_active Expired
- 1974-08-20 IE IE1734/74A patent/IE40511B1/xx unknown
- 1974-08-20 FR FR7428596A patent/FR2241314B1/fr not_active Expired
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