PL3668859T3 - Stałe postacie inhibitora kapsydu HIV - Google Patents

Stałe postacie inhibitora kapsydu HIV

Info

Publication number
PL3668859T3
PL3668859T3 PL18766406.5T PL18766406T PL3668859T3 PL 3668859 T3 PL3668859 T3 PL 3668859T3 PL 18766406 T PL18766406 T PL 18766406T PL 3668859 T3 PL3668859 T3 PL 3668859T3
Authority
PL
Poland
Prior art keywords
solid forms
hiv capsid
capsid inhibitor
inhibitor
hiv
Prior art date
Application number
PL18766406.5T
Other languages
English (en)
Inventor
Bing Shi
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of PL3668859T3 publication Critical patent/PL3668859T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Compounds Of Unknown Constitution (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
PL18766406.5T 2017-08-17 2018-08-16 Stałe postacie inhibitora kapsydu HIV PL3668859T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762546968P 2017-08-17 2017-08-17
PCT/US2018/000172 WO2019035904A1 (en) 2017-08-17 2018-08-16 SOLID FORMS OF HIV CAPSID INHIBITOR

Publications (1)

Publication Number Publication Date
PL3668859T3 true PL3668859T3 (pl) 2022-07-18

Family

ID=63528873

Family Applications (2)

Application Number Title Priority Date Filing Date
PL18766406.5T PL3668859T3 (pl) 2017-08-17 2018-08-16 Stałe postacie inhibitora kapsydu HIV
PL22165005.4T PL4092020T3 (pl) 2017-08-17 2018-08-16 Stałe postacie inhibitora kapsydu hiv

Family Applications After (1)

Application Number Title Priority Date Filing Date
PL22165005.4T PL4092020T3 (pl) 2017-08-17 2018-08-16 Stałe postacie inhibitora kapsydu hiv

Country Status (14)

Country Link
US (3) US11267799B2 (pl)
EP (3) EP4458415A3 (pl)
JP (2) JP7136886B2 (pl)
KR (2) KR102399483B1 (pl)
CN (2) CN117285514A (pl)
AR (1) AR112413A1 (pl)
AU (4) AU2018317833C1 (pl)
CA (2) CA3070141C (pl)
ES (2) ES2991698T3 (pl)
PL (2) PL3668859T3 (pl)
PT (1) PT3668859T (pl)
SI (1) SI3668859T1 (pl)
TW (2) TW202024061A (pl)
WO (1) WO2019035904A1 (pl)

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