PL365443A1 - Pochodne amidów kwasu tiazolilo-, oksazolilo-, pirolilo-i imidazolilokarboksylowego użyteczne jako inhibitory izoenzymów PDE4 - Google Patents

Pochodne amidów kwasu tiazolilo-, oksazolilo-, pirolilo-i imidazolilokarboksylowego użyteczne jako inhibitory izoenzymów PDE4

Info

Publication number
PL365443A1
PL365443A1 PL01365443A PL36544301A PL365443A1 PL 365443 A1 PL365443 A1 PL 365443A1 PL 01365443 A PL01365443 A PL 01365443A PL 36544301 A PL36544301 A PL 36544301A PL 365443 A1 PL365443 A1 PL 365443A1
Authority
PL
Poland
Prior art keywords
oxazolyl
pyrrolyl
thiazolyl
imidazolyl
inhibitors
Prior art date
Application number
PL01365443A
Other languages
English (en)
Inventor
Anthony Marfat
Michael William Mckechney
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of PL365443A1 publication Critical patent/PL365443A1/pl

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    • C—CHEMISTRY; METALLURGY
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • AIDS & HIV (AREA)
PL01365443A 2001-01-31 2001-12-24 Pochodne amidów kwasu tiazolilo-, oksazolilo-, pirolilo-i imidazolilokarboksylowego użyteczne jako inhibitory izoenzymów PDE4 PL365443A1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26548601P 2001-01-31 2001-01-31
PCT/IB2001/002728 WO2002060898A1 (en) 2001-01-31 2001-12-24 Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes

Publications (1)

Publication Number Publication Date
PL365443A1 true PL365443A1 (pl) 2005-01-10

Family

ID=23010641

Family Applications (1)

Application Number Title Priority Date Filing Date
PL01365443A PL365443A1 (pl) 2001-01-31 2001-12-24 Pochodne amidów kwasu tiazolilo-, oksazolilo-, pirolilo-i imidazolilokarboksylowego użyteczne jako inhibitory izoenzymów PDE4

Country Status (24)

Country Link
US (3) US6559168B2 (pl)
EP (1) EP1355907A1 (pl)
JP (1) JP2004518691A (pl)
KR (1) KR20030072614A (pl)
CN (1) CN1489588A (pl)
BG (1) BG108039A (pl)
BR (1) BR0116850A (pl)
CA (1) CA2436551A1 (pl)
CR (1) CR7038A (pl)
CZ (1) CZ20031903A3 (pl)
EA (1) EA200300622A1 (pl)
EC (1) ECSP034683A (pl)
EE (1) EE200300362A (pl)
HU (1) HUP0401305A2 (pl)
IL (1) IL156412A0 (pl)
IS (1) IS6844A (pl)
MA (1) MA26985A1 (pl)
MX (1) MXPA03006886A (pl)
NO (1) NO20033398L (pl)
OA (1) OA12542A (pl)
PL (1) PL365443A1 (pl)
TN (1) TNSN03050A1 (pl)
WO (1) WO2002060898A1 (pl)
ZA (1) ZA200305769B (pl)

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WO2003020313A1 (fr) * 2001-09-04 2003-03-13 Ono Pharmaceutical Co., Ltd. Medicaments contre les maladies respiratoires renfermant un agent de regulation du recepteur de la sphingosine-1-phosphate
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FI114917B (fi) * 2002-08-29 2005-01-31 Hormos Nutraceutical Oy Ltd Lignaanikomplekseja
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GB0317482D0 (en) * 2003-07-25 2003-08-27 Pfizer Ltd Nicotinamide derivatives useful as pde4 inhibitors
GB0317498D0 (en) * 2003-07-25 2003-08-27 Pfizer Ltd Compounds
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