PL3150610T3 - Sole i polimorfy 8-fluoro-2-{4-[(metyloamino}metylo]fenylo}-1,3,4,5-tetrahydro-6Hazepino[5,4,3-cd]indol-6-onu - Google Patents
Sole i polimorfy 8-fluoro-2-{4-[(metyloamino}metylo]fenylo}-1,3,4,5-tetrahydro-6Hazepino[5,4,3-cd]indol-6-onuInfo
- Publication number
- PL3150610T3 PL3150610T3 PL16183844T PL16183844T PL3150610T3 PL 3150610 T3 PL3150610 T3 PL 3150610T3 PL 16183844 T PL16183844 T PL 16183844T PL 16183844 T PL16183844 T PL 16183844T PL 3150610 T3 PL3150610 T3 PL 3150610T3
- Authority
- PL
- Poland
- Prior art keywords
- 6hazepino
- polymorphs
- indol
- methylamino
- tetrahydro
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
- C07C309/19—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
- C07C57/13—Dicarboxylic acids
- C07C57/145—Maleic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
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- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
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- General Chemical & Material Sciences (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Physical Education & Sports Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Reproductive Health (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Dermatology (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Gastroenterology & Hepatology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Gynecology & Obstetrics (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30427710P | 2010-02-12 | 2010-02-12 | |
| PCT/IB2011/050571 WO2011098971A1 (en) | 2010-02-12 | 2011-02-10 | Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one |
| EP16183844.6A EP3150610B1 (en) | 2010-02-12 | 2011-02-10 | Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one |
| EP11708094.5A EP2534153B2 (en) | 2010-02-12 | 2011-02-10 | Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL3150610T3 true PL3150610T3 (pl) | 2020-02-28 |
Family
ID=43859823
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL16183844T PL3150610T3 (pl) | 2010-02-12 | 2011-02-10 | Sole i polimorfy 8-fluoro-2-{4-[(metyloamino}metylo]fenylo}-1,3,4,5-tetrahydro-6Hazepino[5,4,3-cd]indol-6-onu |
| PL11708094.5T PL2534153T5 (pl) | 2010-02-12 | 2011-02-10 | Sole i polimorfy 8-fluoro-2-{4-[(metyloamino}metylo]fenylo}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-onu |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL11708094.5T PL2534153T5 (pl) | 2010-02-12 | 2011-02-10 | Sole i polimorfy 8-fluoro-2-{4-[(metyloamino}metylo]fenylo}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-onu |
Country Status (32)
| Country | Link |
|---|---|
| US (5) | US8754072B2 (OSRAM) |
| EP (4) | EP3597651A1 (OSRAM) |
| JP (6) | JP5745283B2 (OSRAM) |
| KR (2) | KR20120127495A (OSRAM) |
| CN (2) | CN104876937B (OSRAM) |
| AR (2) | AR080164A1 (OSRAM) |
| AU (1) | AU2011213944B2 (OSRAM) |
| BR (1) | BR112012019050B1 (OSRAM) |
| CA (2) | CA2787881C (OSRAM) |
| CY (3) | CY1118319T1 (OSRAM) |
| DK (2) | DK3150610T3 (OSRAM) |
| ES (2) | ES2753748T3 (OSRAM) |
| FI (1) | FI2534153T4 (OSRAM) |
| FR (1) | FR18C1049I2 (OSRAM) |
| HR (2) | HRP20161742T4 (OSRAM) |
| HU (3) | HUE047248T2 (OSRAM) |
| IL (1) | IL220921B (OSRAM) |
| LT (3) | LT3150610T (OSRAM) |
| LU (1) | LUC00093I2 (OSRAM) |
| MX (1) | MX343383B (OSRAM) |
| NL (1) | NL300958I2 (OSRAM) |
| NO (1) | NO2018039I1 (OSRAM) |
| NZ (1) | NZ601445A (OSRAM) |
| PL (2) | PL3150610T3 (OSRAM) |
| PT (2) | PT2534153T (OSRAM) |
| RS (2) | RS55487B2 (OSRAM) |
| RU (1) | RU2570198C2 (OSRAM) |
| SG (2) | SG10201406805RA (OSRAM) |
| SI (2) | SI3150610T1 (OSRAM) |
| SM (3) | SMT201600462T1 (OSRAM) |
| TW (1) | TWI545123B (OSRAM) |
| WO (1) | WO2011098971A1 (OSRAM) |
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| JP5745283B2 (ja) | 2010-02-12 | 2015-07-08 | ファイザー・インク | 8−フルオロ−2−{4−[(メチルアミノ)メチル]フェニル}−1,3,4,5−テトラヒドロ−6H−アゼピノ[5,4,3−cd]インドール−6−オンの塩および多形体 |
| TW201516636A (zh) * | 2013-10-22 | 2015-05-01 | Hon Hai Prec Ind Co Ltd | 電子裝置及其供電方法 |
| LT3182975T (lt) * | 2014-08-22 | 2025-11-25 | Tabletės su didele rukaparibo doze | |
| BR112018073667A2 (pt) * | 2016-05-16 | 2019-03-12 | Pulmagen Therapeutics (Asthma) Limited | cristal de derivado de quinolina |
| DE102016218772A1 (de) * | 2016-09-28 | 2018-03-29 | Bruker Biospin Gmbh | Verbesserte Temperierung eines NMR-MAS-Rotors |
| HRP20241280T1 (hr) * | 2017-01-24 | 2024-12-06 | Assia Chemical Industries Ltd. | Kruti oblici rukapariba i soli rukapariba |
| CN109651377B (zh) * | 2017-10-12 | 2020-10-20 | 成都海创药业有限公司 | 一种治疗癌症的化合物及其用途 |
| CA3080657A1 (en) | 2017-11-03 | 2019-05-09 | Sandoz Ag | Crystalline salt of a tricyclic poly(adp-ribose) polymerase inhibitor |
| WO2019115000A1 (en) * | 2017-12-15 | 2019-06-20 | Advitech Advisory And Technologies Sa | Process for the preparation of rucaparib and novel synthesis intermediates |
| WO2019130229A1 (en) | 2017-12-28 | 2019-07-04 | Mylan Laboratories Ltd | Methods and intermediates for preparing rucaparib |
| PE20211305A1 (es) | 2018-01-05 | 2021-07-20 | Cybrexa 1 Inc | Compuestos, composiciones y metodos para tratar enfermedades que involucren tejidos con enfermedades acidas o hipoxicas |
| US10442813B2 (en) | 2018-01-30 | 2019-10-15 | RK Pharma Solutions LLC | Polymorphs of rucaparib camsylate and methods of making same |
| WO2019207596A1 (en) | 2018-04-25 | 2019-10-31 | Mylan Laboratories Limited | Novel crystalline forms of rucaparib (s)-camsylate salt and rucaparib free base |
| WO2019207498A1 (en) * | 2018-04-25 | 2019-10-31 | Biophore India Pharmaceuticals Pvt. Ltd | Solid forms of 8-fluoro-2-{4-[(methylamino)methyl] phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd] indol-6-one ((1s,4r)-7,7dimethyl-2-oxobicyclo [2.2.1] hept-1-yl) methanesulfonic acid salt (rucaparib camsylate) and the prerparation thereof |
| CN108743557A (zh) * | 2018-06-27 | 2018-11-06 | 李莉 | 一种磷酸瑞卡帕布软胶囊及其制备方法 |
| CN109111454A (zh) * | 2018-08-01 | 2019-01-01 | 宁波金未生物科技有限公司 | 一种瑞卡帕布s-樟脑磺酸盐 |
| CN113454080B (zh) | 2018-10-30 | 2025-10-28 | 修复治疗公司 | 化合物、药物组合物和制备化合物的方法以及其使用方法 |
| CN111217818A (zh) * | 2018-11-27 | 2020-06-02 | 台耀化学股份有限公司 | 芦卡帕尼樟脑磺酸盐的结晶、及制备三环化合物、芦卡帕尼及其樟脑磺酸盐结晶的方法 |
| CN111542527A (zh) * | 2018-12-06 | 2020-08-14 | 上海诚妙医药科技有限公司 | 芦卡帕利樟脑磺酸盐的新晶型和制备方法及其用途 |
| MX2021006841A (es) | 2018-12-10 | 2021-07-02 | Ideaya Biosciences Inc | Derivados de 2-oxoquinazolina como inhibidores de metionina adenosiltransferasa 2?. |
| CR20220058A (es) | 2019-07-10 | 2022-07-19 | Cybrexa 2 Inc | Conjugados peptídicos de citotoxinas como terapéuticos |
| JP7675060B2 (ja) | 2019-07-10 | 2025-05-12 | サイブレクサ 3,インコーポレイテッド | 治療薬としての微小管標的化剤のペプチドコンジュゲート |
| CN111004244A (zh) * | 2019-12-27 | 2020-04-14 | 重庆市碚圣医药科技股份有限公司 | 一种瑞卡帕布樟脑磺酸盐的合成方法 |
| WO2021156140A1 (en) | 2020-02-03 | 2021-08-12 | Sandoz Ag | Polymorph of rucaparib mesylate |
| BR112022021089A2 (pt) * | 2020-04-24 | 2022-12-06 | Astrazeneca Ab | Formulações farmacêuticas |
| CA3176206A1 (en) | 2020-04-28 | 2021-11-04 | Debnath Bhuniya | Novel compounds useful as poly(adp-ribose) polymerase (parp) inhibitors |
| EP4178571A4 (en) | 2020-07-10 | 2024-07-17 | The Regents Of The University Of Michigan | GAS41 INHIBITORS AND METHODS OF USE |
| WO2022015557A1 (en) | 2020-07-14 | 2022-01-20 | Assia Chemical Industries Ltd | Solid state forms of rucaparib salts |
| WO2022090938A1 (en) | 2020-10-31 | 2022-05-05 | Rhizen Pharmaceuticals Ag | Phthalazinone derivatives useful as parp inhibitors |
| MX2023011793A (es) | 2021-04-08 | 2023-10-12 | Rhizen Pharmaceuticals Ag | Inhibidores de poli(adenosin difosfato-ribosa) polimerasa. |
| EP4463232A1 (en) | 2022-01-11 | 2024-11-20 | Assia Chemical Industries Ltd. | Solid state forms of rucaparib tosylate |
| WO2023152754A1 (en) * | 2022-02-08 | 2023-08-17 | Sawant, Mohit Manikrao | Crystalline form of rosuvastatin allyl ester |
| CN120693324A (zh) * | 2022-11-30 | 2025-09-23 | 艾迪亚生物科学公司 | 2-氧代喹唑啉的晶型 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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