PL3141552T3 - Pochodne tienopiryimidyny wykazujące aktywność hamującą względem kinazy białkowej - Google Patents

Pochodne tienopiryimidyny wykazujące aktywność hamującą względem kinazy białkowej

Info

Publication number
PL3141552T3
PL3141552T3 PL16190699T PL16190699T PL3141552T3 PL 3141552 T3 PL3141552 T3 PL 3141552T3 PL 16190699 T PL16190699 T PL 16190699T PL 16190699 T PL16190699 T PL 16190699T PL 3141552 T3 PL3141552 T3 PL 3141552T3
Authority
PL
Poland
Prior art keywords
protein kinase
inhibitory activity
thienopyrimidine derivatives
thienopyrimidine
derivatives
Prior art date
Application number
PL16190699T
Other languages
English (en)
Inventor
Seung Hyun Jung
Young Hee Jung
Wha II Choi
Jung Beom Son
Eun Ju Jeon
In Ho Yang
Tae Hun Song
Mi Kyoung Lee
Mi Kyoung Ko
Young Gil Ahn
Maeng Sup Kim
Young Jin Ham
Tae Bo Sim
Hwan Geun Choi
Jung Mi Hah
Dong-Sik Park
Hwan Kim
Original Assignee
Hanmi Pharm. Co., Ltd.
Hanmi Science Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hanmi Pharm. Co., Ltd., Hanmi Science Co., Ltd. filed Critical Hanmi Pharm. Co., Ltd.
Publication of PL3141552T3 publication Critical patent/PL3141552T3/pl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Communicable Diseases (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
PL16190699T 2010-01-29 2011-01-28 Pochodne tienopiryimidyny wykazujące aktywność hamującą względem kinazy białkowej PL3141552T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
KR20100008720A KR101483215B1 (ko) 2010-01-29 2010-01-29 단백질 키나아제 저해활성을 갖는 비시클릭 헤테로아릴 유도체
EP11737311.8A EP2528920A4 (en) 2010-01-29 2011-01-28 BICYCLIC HETEROARYL DERIVATIVES HAVING PROTEIN KINASE INHIBITORY ACTIVITY
EP16190699.5A EP3141552B1 (en) 2010-01-29 2011-01-28 Thienopyrimidine derivatives having inhibitory activity for protein kinase
PCT/KR2011/000615 WO2011093672A2 (en) 2010-01-29 2011-01-28 Bicyclic heteroaryl derivatives having inhibitory activity for protein kinase

Publications (1)

Publication Number Publication Date
PL3141552T3 true PL3141552T3 (pl) 2019-08-30

Family

ID=44320004

Family Applications (1)

Application Number Title Priority Date Filing Date
PL16190699T PL3141552T3 (pl) 2010-01-29 2011-01-28 Pochodne tienopiryimidyny wykazujące aktywność hamującą względem kinazy białkowej

Country Status (9)

Country Link
US (1) US10112954B2 (pl)
EP (2) EP2528920A4 (pl)
JP (1) JP5844284B2 (pl)
KR (1) KR101483215B1 (pl)
CN (1) CN102741256B (pl)
ES (1) ES2726882T3 (pl)
PL (1) PL3141552T3 (pl)
TR (1) TR201906936T4 (pl)
WO (1) WO2011093672A2 (pl)

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WO2011093672A3 (en) 2012-01-05
EP2528920A2 (en) 2012-12-05
KR20110088960A (ko) 2011-08-04
CN102741256B (zh) 2015-12-02
KR101483215B1 (ko) 2015-01-16
EP2528920A4 (en) 2013-08-07
EP3141552A1 (en) 2017-03-15
US10112954B2 (en) 2018-10-30
ES2726882T3 (es) 2019-10-10
JP2013518098A (ja) 2013-05-20
EP3141552B1 (en) 2019-04-17
US20120302567A1 (en) 2012-11-29
TR201906936T4 (tr) 2019-06-21
WO2011093672A2 (en) 2011-08-04
CN102741256A (zh) 2012-10-17
JP5844284B2 (ja) 2016-01-13

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