PL2938194T3 - Pochodne n-podstawionego 5-fluoro-4-imino-3-metylo-2-okso-3,4-dihydropirymidyno-1(2h)-karboksylanu - Google Patents

Pochodne n-podstawionego 5-fluoro-4-imino-3-metylo-2-okso-3,4-dihydropirymidyno-1(2h)-karboksylanu

Info

Publication number
PL2938194T3
PL2938194T3 PL13868013T PL13868013T PL2938194T3 PL 2938194 T3 PL2938194 T3 PL 2938194T3 PL 13868013 T PL13868013 T PL 13868013T PL 13868013 T PL13868013 T PL 13868013T PL 2938194 T3 PL2938194 T3 PL 2938194T3
Authority
PL
Poland
Prior art keywords
dihydropyrimidine
imino
oxo
fluoro
substituted
Prior art date
Application number
PL13868013T
Other languages
English (en)
Polish (pl)
Inventor
Beth Lorsbach
W. John Owen
Chenglin Yao
Lindsay Stelzer
Original Assignee
Adama Makhteshim Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd. filed Critical Adama Makhteshim Ltd.
Publication of PL2938194T3 publication Critical patent/PL2938194T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22—O-Aryl or S-Aryl esters thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
PL13868013T 2012-12-28 2013-12-23 Pochodne n-podstawionego 5-fluoro-4-imino-3-metylo-2-okso-3,4-dihydropirymidyno-1(2h)-karboksylanu PL2938194T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747086P 2012-12-28 2012-12-28
PCT/US2013/077540 WO2014105844A1 (en) 2012-12-28 2013-12-23 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
EP13868013.7A EP2938194B1 (en) 2012-12-28 2013-12-23 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives

Publications (1)

Publication Number Publication Date
PL2938194T3 true PL2938194T3 (pl) 2020-09-21

Family

ID=51022033

Family Applications (1)

Application Number Title Priority Date Filing Date
PL13868013T PL2938194T3 (pl) 2012-12-28 2013-12-23 Pochodne n-podstawionego 5-fluoro-4-imino-3-metylo-2-okso-3,4-dihydropirymidyno-1(2h)-karboksylanu

Country Status (18)

Country Link
US (2) US9622474B2 (enExample)
EP (1) EP2938194B1 (enExample)
JP (1) JP6324994B2 (enExample)
KR (1) KR20150103096A (enExample)
CN (2) CN104902757B (enExample)
AU (1) AU2013370493B2 (enExample)
BR (1) BR102013033709B1 (enExample)
CA (1) CA2893778A1 (enExample)
CR (1) CR20150382A (enExample)
DK (1) DK2938194T3 (enExample)
EC (1) ECSP15032859A (enExample)
HU (1) HUE047711T2 (enExample)
IL (1) IL239561B (enExample)
MX (1) MX2015008441A (enExample)
PL (1) PL2938194T3 (enExample)
RU (1) RU2638556C2 (enExample)
UA (1) UA115462C2 (enExample)
WO (1) WO2014105844A1 (enExample)

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CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
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JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
CR20160344A (es) 2013-12-31 2016-12-19 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas para el control fúngico en cereales
UA129860C2 (uk) 2013-12-31 2025-08-27 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
CN107426999B (zh) 2014-12-30 2023-01-20 美国陶氏益农公司 具有杀真菌活性的吡啶酰胺化合物
AU2015374379B2 (en) 2014-12-30 2018-10-04 Dow Agrosciences Llc Picolinamides as fungicides
UA121561C2 (uk) 2014-12-30 2020-06-25 Дау Аґросаєнсиз Елелсі Застосування сполук аміду як фунгіцидів
KR20170100549A (ko) 2014-12-30 2017-09-04 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
US10173971B2 (en) 2014-12-30 2019-01-08 Dow Agrosciences Llc Picolinamides with fungicidal activity
CA3118729A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound

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UA129860C2 (uk) 2013-12-31 2025-08-27 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
CR20160344A (es) 2013-12-31 2016-12-19 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas para el control fúngico en cereales
MA41272A (fr) 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences

Also Published As

Publication number Publication date
CN110003118A (zh) 2019-07-12
IL239561A0 (en) 2015-08-31
DK2938194T3 (da) 2020-01-02
CR20150382A (es) 2015-08-21
US9908855B2 (en) 2018-03-06
KR20150103096A (ko) 2015-09-09
US20160192653A1 (en) 2016-07-07
BR102013033709B1 (pt) 2019-05-14
EP2938194A1 (en) 2015-11-04
HUE047711T2 (hu) 2020-05-28
EP2938194B1 (en) 2019-11-27
BR102013033709A2 (pt) 2015-10-06
RU2015131095A (ru) 2017-02-06
EP2938194A4 (en) 2016-08-31
IL239561B (en) 2018-01-31
RU2638556C2 (ru) 2017-12-14
HK1214475A1 (en) 2016-07-29
CN104902757A (zh) 2015-09-09
UA115462C2 (uk) 2017-11-10
MX2015008441A (es) 2015-09-23
CN104902757B (zh) 2019-01-08
ECSP15032859A (es) 2015-11-30
CA2893778A1 (en) 2014-07-03
JP6324994B2 (ja) 2018-05-16
US9622474B2 (en) 2017-04-18
JP2016507512A (ja) 2016-03-10
US20170204069A1 (en) 2017-07-20
WO2014105844A1 (en) 2014-07-03
AU2013370493B2 (en) 2017-08-17
AU2013370493A1 (en) 2015-07-02

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