HUE047711T2 - N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok - Google Patents

N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok

Info

Publication number
HUE047711T2
HUE047711T2 HUE13868013A HUE13868013A HUE047711T2 HU E047711 T2 HUE047711 T2 HU E047711T2 HU E13868013 A HUE13868013 A HU E13868013A HU E13868013 A HUE13868013 A HU E13868013A HU E047711 T2 HUE047711 T2 HU E047711T2
Authority
HU
Hungary
Prior art keywords
dihydropyrimidine
imino
oxo
fluoro
substituted
Prior art date
Application number
HUE13868013A
Other languages
English (en)
Hungarian (hu)
Inventor
Beth Lorsbach
W Owen
Chenglin Yao
Lindsay Stelzer
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of HUE047711T2 publication Critical patent/HUE047711T2/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22O-Aryl or S-Aryl esters thereof
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
HUE13868013A 2012-12-28 2013-12-23 N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok HUE047711T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261747086P 2012-12-28 2012-12-28

Publications (1)

Publication Number Publication Date
HUE047711T2 true HUE047711T2 (hu) 2020-05-28

Family

ID=51022033

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE13868013A HUE047711T2 (hu) 2012-12-28 2013-12-23 N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok

Country Status (18)

Country Link
US (2) US9622474B2 (enExample)
EP (1) EP2938194B1 (enExample)
JP (1) JP6324994B2 (enExample)
KR (1) KR20150103096A (enExample)
CN (2) CN110003118A (enExample)
AU (1) AU2013370493B2 (enExample)
BR (1) BR102013033709B1 (enExample)
CA (1) CA2893778A1 (enExample)
CR (1) CR20150382A (enExample)
DK (1) DK2938194T3 (enExample)
EC (1) ECSP15032859A (enExample)
HU (1) HUE047711T2 (enExample)
IL (1) IL239561B (enExample)
MX (1) MX2015008441A (enExample)
PL (1) PL2938194T3 (enExample)
RU (1) RU2638556C2 (enExample)
UA (1) UA115462C2 (enExample)
WO (1) WO2014105844A1 (enExample)

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EP3240413B1 (en) 2014-12-30 2020-05-13 Dow Agrosciences LLC Picolinamide compounds with fungicidal activity
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UA121561C2 (uk) 2014-12-30 2020-06-25 Дау Аґросаєнсиз Елелсі Застосування сполук аміду як фунгіцидів
WO2016109302A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
EP4034529A1 (en) 2019-09-23 2022-08-03 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one

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SG11201605377VA (en) 2013-12-31 2016-08-30 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
MA41272A (fr) 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences

Also Published As

Publication number Publication date
BR102013033709B1 (pt) 2019-05-14
HK1214475A1 (en) 2016-07-29
KR20150103096A (ko) 2015-09-09
US20170204069A1 (en) 2017-07-20
US9622474B2 (en) 2017-04-18
RU2638556C2 (ru) 2017-12-14
AU2013370493B2 (en) 2017-08-17
CR20150382A (es) 2015-08-21
US20160192653A1 (en) 2016-07-07
MX2015008441A (es) 2015-09-23
IL239561B (en) 2018-01-31
CN110003118A (zh) 2019-07-12
EP2938194A4 (en) 2016-08-31
WO2014105844A1 (en) 2014-07-03
CA2893778A1 (en) 2014-07-03
AU2013370493A1 (en) 2015-07-02
CN104902757A (zh) 2015-09-09
JP2016507512A (ja) 2016-03-10
BR102013033709A2 (pt) 2015-10-06
EP2938194A1 (en) 2015-11-04
IL239561A0 (en) 2015-08-31
EP2938194B1 (en) 2019-11-27
JP6324994B2 (ja) 2018-05-16
US9908855B2 (en) 2018-03-06
CN104902757B (zh) 2019-01-08
PL2938194T3 (pl) 2020-09-21
DK2938194T3 (da) 2020-01-02
ECSP15032859A (es) 2015-11-30
RU2015131095A (ru) 2017-02-06
UA115462C2 (uk) 2017-11-10

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