PL168456B1 - Sposób wytwarzania cyklopeptydów PL PL PL - Google Patents
Sposób wytwarzania cyklopeptydów PL PL PLInfo
- Publication number
- PL168456B1 PL168456B1 PL91299317A PL29931791A PL168456B1 PL 168456 B1 PL168456 B1 PL 168456B1 PL 91299317 A PL91299317 A PL 91299317A PL 29931791 A PL29931791 A PL 29931791A PL 168456 B1 PL168456 B1 PL 168456B1
- Authority
- PL
- Poland
- Prior art keywords
- arg
- gly
- ile
- phe
- fmoc
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/58—Atrial natriuretic factor complex; Atriopeptin; Atrial natriuretic peptide [ANP]; Cardionatrin; Cardiodilatin
- C07K14/582—Atrial natriuretic factor complex; Atriopeptin; Atrial natriuretic peptide [ANP]; Cardionatrin; Cardiodilatin at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Biochemistry (AREA)
- Heart & Thoracic Surgery (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Diabetes (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Toxicology (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19904032268 DE4032268A1 (de) | 1990-10-11 | 1990-10-11 | Cyclopeptide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
DE19904032269 DE4032269A1 (de) | 1990-10-11 | 1990-10-11 | Cyclopeptide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
DE19904032271 DE4032271A1 (de) | 1990-10-11 | 1990-10-11 | Cyclopeptide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
DE19914117733 DE4117733A1 (de) | 1991-05-30 | 1991-05-30 | Cyclopeptide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
PCT/EP1991/001934 WO1992006998A1 (de) | 1990-10-11 | 1991-10-10 | Cyclopeptide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
PL168456B1 true PL168456B1 (pl) | 1996-02-29 |
Family
ID=27435038
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL91299317A PL168456B1 (pl) | 1990-10-11 | 1991-10-10 | Sposób wytwarzania cyklopeptydów PL PL PL |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0552238A1 (de) |
JP (1) | JPH06501950A (de) |
KR (1) | KR930702395A (de) |
AU (1) | AU8736691A (de) |
CA (1) | CA2089747A1 (de) |
CZ (1) | CZ61893A3 (de) |
FI (1) | FI931499A0 (de) |
HU (1) | HUT63859A (de) |
IE (1) | IE913582A1 (de) |
PL (1) | PL168456B1 (de) |
SK (1) | SK32693A3 (de) |
WO (1) | WO1992006998A1 (de) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6525022B1 (en) | 1993-11-12 | 2003-02-25 | Genentech, Inc. | Receptor specific atrial natriuretic peptides |
US5665704A (en) * | 1993-11-12 | 1997-09-09 | Genentech, Inc. | Receptor specific atrial natriuretic peptides |
US5846932A (en) * | 1993-11-12 | 1998-12-08 | Genentech, Inc. | Receptor specific atrial natriuretic peptides |
AU769791B2 (en) * | 1998-06-24 | 2004-02-05 | New York University | Novel Staphylococcus peptides for bacterial interference |
US6337385B1 (en) | 1998-06-24 | 2002-01-08 | The Rockefeller University | Staphylococcus peptides for bacterial interference |
FR2797689B1 (fr) * | 1999-08-16 | 2003-06-27 | Pasteur Sanofi Diagnostics | Utilisation de composes synthetiques pour des immunodosages |
US6455587B1 (en) * | 2000-03-15 | 2002-09-24 | Pharmacor Inc. | Amino acid derivatives as HIV aspartyl protease inhibitors |
US7388008B2 (en) | 2004-08-02 | 2008-06-17 | Ambrilia Biopharma Inc. | Lysine based compounds |
CA2632095A1 (en) | 2005-11-30 | 2007-06-07 | Ambrilia Biopharma Inc. | Lysine-based prodrugs of aspartyl protease inhibitors and processes for their preparation |
AU2007233116B2 (en) | 2006-03-30 | 2013-05-09 | Palatin Technologies, Inc. | Cyclic natriuretic peptide constructs |
US8580746B2 (en) | 2006-03-30 | 2013-11-12 | Palatin Technologies, Inc. | Amide linkage cyclic natriuretic peptide constructs |
CA2647146A1 (en) | 2006-03-30 | 2007-10-11 | Palatin Technologies, Inc. | Linear natriuretic peptide constructs |
WO2008078200A2 (en) | 2006-09-21 | 2008-07-03 | Ambrilia Biopharma Inc. | Protease inhibitors |
JP5649825B2 (ja) | 2007-01-31 | 2015-01-07 | デイナ ファーバー キャンサー インスティチュート,インコーポレイテッド | 安定化させたp53ペプチドおよびその使用法 |
KR101525754B1 (ko) | 2007-03-28 | 2015-06-09 | 프레지던트 앤드 펠로우즈 오브 하바드 칼리지 | 스티칭된 폴리펩티드 |
CN108570097A (zh) | 2010-08-13 | 2018-09-25 | 爱勒让治疗公司 | 拟肽大环化合物 |
MX358886B (es) | 2011-10-18 | 2018-08-31 | Aileron Therapeutics Inc | Macrociclos peptidomimeticos. |
US8987414B2 (en) | 2012-02-15 | 2015-03-24 | Aileron Therapeutics, Inc. | Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles |
SG11201404648PA (en) | 2012-02-15 | 2014-09-26 | Aileron Therapeutics Inc | Peptidomimetic macrocycles |
EP2914256B1 (de) | 2012-11-01 | 2019-07-31 | Aileron Therapeutics, Inc. | Disubstituierte aminosäuren und verfahren zur herstellung und verwendung davon |
US10736932B2 (en) * | 2014-05-20 | 2020-08-11 | Ohio State Innovation Foundation | Small molecule Ras inhibitors |
CN112972378A (zh) | 2014-09-24 | 2021-06-18 | 艾瑞朗医疗公司 | 拟肽大环化合物及其制剂 |
JP2017533889A (ja) | 2014-09-24 | 2017-11-16 | エルロン・セラピューティクス・インコーポレイテッドAileron Therapeutics,Inc. | ペプチド模倣大環状分子およびその使用 |
EP3294318A4 (de) | 2015-03-20 | 2019-04-03 | Aileron Therapeutics, Inc. | Peptidomimetische makrozyklen und verwendungen davon |
US10023613B2 (en) | 2015-09-10 | 2018-07-17 | Aileron Therapeutics, Inc. | Peptidomimetic macrocycles as modulators of MCL-1 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1337891C (en) * | 1987-12-16 | 1996-01-02 | John Dimaio | Anf derivatives with novel bridging |
US4935492A (en) * | 1987-12-24 | 1990-06-19 | California Biotechnology Inc. | Cyclic analogs of atrial natriuretic peptides |
DK380288D0 (da) * | 1988-07-07 | 1988-07-07 | Novo Industri As | Hidtil ukendet peptider |
-
1991
- 1991-10-10 CZ CS93618A patent/CZ61893A3/cs unknown
- 1991-10-10 PL PL91299317A patent/PL168456B1/pl unknown
- 1991-10-10 CA CA002089747A patent/CA2089747A1/en not_active Abandoned
- 1991-10-10 SK SK32693A patent/SK32693A3/sk unknown
- 1991-10-10 WO PCT/EP1991/001934 patent/WO1992006998A1/de not_active Application Discontinuation
- 1991-10-10 JP JP3516845A patent/JPH06501950A/ja active Pending
- 1991-10-10 EP EP91918322A patent/EP0552238A1/de not_active Withdrawn
- 1991-10-10 HU HU931054A patent/HUT63859A/hu unknown
- 1991-10-10 AU AU87366/91A patent/AU8736691A/en not_active Abandoned
- 1991-10-16 IE IE358291A patent/IE913582A1/en not_active Application Discontinuation
-
1993
- 1993-04-02 FI FI931499A patent/FI931499A0/fi not_active Application Discontinuation
- 1993-04-10 KR KR1019930701088A patent/KR930702395A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CA2089747A1 (en) | 1992-04-12 |
IE913582A1 (en) | 1992-04-22 |
FI931499A (fi) | 1993-04-02 |
FI931499A0 (fi) | 1993-04-02 |
HU9301054D0 (en) | 1993-07-28 |
WO1992006998A1 (de) | 1992-04-30 |
AU8736691A (en) | 1992-05-20 |
HUT63859A (en) | 1993-10-28 |
EP0552238A1 (de) | 1993-07-28 |
CZ61893A3 (en) | 1994-01-19 |
SK32693A3 (en) | 1993-09-09 |
KR930702395A (ko) | 1993-09-09 |
JPH06501950A (ja) | 1994-03-03 |
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