PH20168A - 7-carboxymethoxyphenylacetamino-3-cephem derivatives and their pharmaceutical compositions - Google Patents
7-carboxymethoxyphenylacetamino-3-cephem derivatives and their pharmaceutical compositionsInfo
- Publication number
- PH20168A PH20168A PH29873A PH29873A PH20168A PH 20168 A PH20168 A PH 20168A PH 29873 A PH29873 A PH 29873A PH 29873 A PH29873 A PH 29873A PH 20168 A PH20168 A PH 20168A
- Authority
- PH
- Philippines
- Prior art keywords
- carboxymethoxyphenylacetamino
- pharmaceutical compositions
- cephem derivatives
- cephem
- derivatives
- Prior art date
Links
- LXXZHWKZKHWWSS-OGVSOVDVSA-N 2-[[(6R)-4-acetamido-8-oxo-4-phenyl-5-thia-1-azabicyclo[4.2.0]oct-2-en-7-yl]oxy]acetic acid Chemical class C(=O)(O)COC1[C@@H]2N(C=CC(S2)(NC(=O)C)C2=CC=CC=C2)C1=O LXXZHWKZKHWWSS-OGVSOVDVSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/36—Methylene radicals, substituted by sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP21772682A JPS59108791A (ja) | 1982-12-14 | 1982-12-14 | ７−カルボキシメトキシフエニルアセトアミド−３−セフエム誘導体、その製造方法およびそれからなる抗菌剤 |
| JP3601783A JPS59161389A (ja) | 1983-03-07 | 1983-03-07 | ７−カルボキシメトキシフエニルアセトアミドセフエム誘導体，その製造法およびそれからなる抗菌剤 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH20168A true PH20168A (en) | 1986-10-09 |
Family
ID=26375029
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH29873A PH20168A (en) | 1982-12-14 | 1983-11-23 | 7-carboxymethoxyphenylacetamino-3-cephem derivatives and their pharmaceutical compositions |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4546176A (it) |
| KR (1) | KR840007012A (it) |
| AT (1) | ATA435283A (it) |
| AU (1) | AU2082783A (it) |
| BE (1) | BE898442A (it) |
| CH (1) | CH656131A5 (it) |
| DE (1) | DE3345093A1 (it) |
| DK (1) | DK572183A (it) |
| ES (2) | ES8506025A1 (it) |
| FR (1) | FR2569195B1 (it) |
| GB (1) | GB2132613B (it) |
| IT (1) | IT1169969B (it) |
| NL (1) | NL8304272A (it) |
| PH (1) | PH20168A (it) |
| SE (1) | SE8306882L (it) |
| YU (1) | YU237283A (it) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5232918A (en) * | 1987-07-23 | 1993-08-03 | Imperial Chemical Industries Plc | Cephalosporin derivatives |
| US5180719A (en) * | 1988-10-24 | 1993-01-19 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl lactam esters |
| US5328908A (en) * | 1988-10-24 | 1994-07-12 | Procter & Gamble Pharmaceuticals, Inc. | Antimicrobial quinolone thioureas |
| US5273973A (en) * | 1988-10-24 | 1993-12-28 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl esters |
| CA2001203C (en) * | 1988-10-24 | 2001-02-13 | Thomas P. Demuth, Jr. | Novel antimicrobial dithiocarbamoyl quinolones |
| EP0997466A1 (en) * | 1988-10-24 | 2000-05-03 | PROCTER & GAMBLE PHARMACEUTICALS, INC. | Novel antimicrobial lactam-quinolones |
| US5491139A (en) * | 1988-10-24 | 1996-02-13 | The Procter & Gamble Company | Antimicrobial quinolonyl lactams |
| JPH05506033A (ja) * | 1990-04-18 | 1993-09-02 | ノーウィッチ、イートン、ファーマスーティカルズ、インコーポレーテッド | 抗微生物性キノロニルラクタム類 |
| US5244892A (en) * | 1990-10-16 | 1993-09-14 | Kyorin Pharmaceutical Co., Ltd. | Cephem compounds, and antibacterial agents |
| EP0775145A1 (en) * | 1994-08-02 | 1997-05-28 | The Procter & Gamble Company | Process for making quinolonyl lactam antimicrobials and novel intermediate compounds |
| ATE190972T1 (de) * | 1994-08-02 | 2000-04-15 | Procter & Gamble | Verfahren zur herstellung von antimikrobiellen verbindungen |
| TW200420573A (en) * | 2002-09-26 | 2004-10-16 | Rib X Pharmaceuticals Inc | Bifunctional heterocyclic compounds and methods of making and using same |
| JP2006523229A (ja) * | 2003-03-05 | 2006-10-12 | リブ−エックス ファーマシューティカルズ，インコーポレイテッド | 二官能性複素環式化合物ならびにその製造および使用方法 |
| EP1682563A1 (en) * | 2003-10-30 | 2006-07-26 | Rib-X Pharmaceuticals, Inc. | Bifunctional macrolide heterocyclic compounds and mehtods of making and using the same |
| JP2007512256A (ja) * | 2003-11-18 | 2007-05-17 | リブ−エックス ファーマシューティカルズ，インコーポレイテッド | 二官能性マクロライド複素環化合物ならびにこれらを製造する方法およびこれらを使用する方法 |
| JP5383037B2 (ja) * | 2004-02-27 | 2014-01-08 | リブ−エックス ファーマシューティカルズ，インコーポレイテッド | 大環状化合物およびそれらを製造し使用する方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR208171A1 (es) * | 1972-09-29 | 1976-12-09 | Ciba Geigy Ag | Procedimiento para la obtencion de nuevos derivados del acido cef-3-em-4-carboxilico |
| US4338439A (en) * | 1976-08-26 | 1982-07-06 | Eli Lilly And Company | 7-[2-[(Substituted benzoyl]amino]acetamido]cephalosporins |
| SE8009049L (sv) * | 1980-03-04 | 1981-09-05 | Eisai Co Ltd | 7alfa-metoxicefalosporinderivat, sett for framstellning derav och antibakteriella lekemedel innehallande dessa foreningar |
| US4468394A (en) * | 1981-04-02 | 1984-08-28 | Eisai Co., Ltd. | Cephalosporin compounds |
-
1983
- 1983-10-20 US US06/544,406 patent/US4546176A/en not_active Expired - Fee Related
- 1983-10-31 AU AU20827/83A patent/AU2082783A/en not_active Abandoned
- 1983-11-04 GB GB08329554A patent/GB2132613B/en not_active Expired
- 1983-11-23 PH PH29873A patent/PH20168A/en unknown
- 1983-12-05 YU YU02372/83A patent/YU237283A/xx unknown
- 1983-12-12 IT IT24122/83A patent/IT1169969B/it active
- 1983-12-12 NL NL8304272A patent/NL8304272A/nl not_active Application Discontinuation
- 1983-12-12 FR FR8319876A patent/FR2569195B1/fr not_active Expired
- 1983-12-13 DE DE19833345093 patent/DE3345093A1/de not_active Withdrawn
- 1983-12-13 CH CH6649/83A patent/CH656131A5/de not_active IP Right Cessation
- 1983-12-13 ES ES528003A patent/ES8506025A1/es not_active Expired
- 1983-12-13 SE SE8306882A patent/SE8306882L/xx not_active Application Discontinuation
- 1983-12-13 DK DK572183A patent/DK572183A/da not_active Application Discontinuation
- 1983-12-13 BE BE0/212036A patent/BE898442A/fr not_active IP Right Cessation
- 1983-12-14 KR KR1019830005939A patent/KR840007012A/ko not_active Application Discontinuation
- 1983-12-14 AT AT0435283A patent/ATA435283A/de not_active Application Discontinuation
-
1984
- 1984-07-13 ES ES534297A patent/ES534297A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| ES8505691A1 (es) | 1985-06-01 |
| BE898442A (fr) | 1984-06-13 |
| GB2132613B (en) | 1986-05-08 |
| FR2569195B1 (fr) | 1987-01-09 |
| YU237283A (en) | 1986-04-30 |
| US4546176A (en) | 1985-10-08 |
| NL8304272A (nl) | 1984-07-02 |
| KR840007012A (ko) | 1984-12-04 |
| AU2082783A (en) | 1984-06-21 |
| DK572183A (da) | 1984-06-27 |
| ES528003A0 (es) | 1985-06-16 |
| DK572183D0 (da) | 1983-12-13 |
| ES534297A0 (es) | 1985-06-01 |
| ATA435283A (de) | 1986-12-15 |
| GB8329554D0 (en) | 1983-12-07 |
| DE3345093A1 (de) | 1984-06-14 |
| FR2569195A1 (fr) | 1986-02-21 |
| ES8506025A1 (es) | 1985-06-16 |
| GB2132613A (en) | 1984-07-11 |
| CH656131A5 (de) | 1986-06-13 |
| IT8324122A0 (it) | 1983-12-12 |
| SE8306882D0 (sv) | 1983-12-13 |
| SE8306882L (sv) | 1984-06-15 |
| IT1169969B (it) | 1987-06-03 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL72028A0 (en) | Aminomethyl-oxooxazolidinylbenzene derivatives and pharmaceutical compositions containing them | |
| IL69955A0 (en) | 1-phenyl-2-piperidinoalkanol derivatives,their preparation and pharmaceutical compositions containing them | |
| IL68913A (en) | 3-aminoalkyl-1h-indole-5-alkan-sulphonamide derivatives,their preparation and pharmaceutical compositions containing them | |
| IL69157A0 (en) | Fluoromorphinan derivatives,their preparation and pharmaceutical compositions containing them | |
| IL72566A (en) | Androst-5-en-17-one and 5alpha-androstan-17-one derivatives and pharmaceutical compositions containing the same | |
| GB2091262B (en) | 3-aminoprpoxyaryl derivatives their preparation and pharmaceutical compositions containing them | |
| NZ210633A (en) | Glycerol derivatives and pharmaceutical compositions thereof | |
| NZ201520A (en) | Substituted aminopyridazines and pharmaceutical compositions | |
| IL68360A0 (en) | Imidazopyrazolopyrimidine derivatives,their preparation and pharmaceutical compositions containing them | |
| NZ209064A (en) | N 6 -diarylalkyl-adenosine derivatives and pharmaceutical compositions | |
| NZ206636A (en) | Pyridine derivatives and pharmaceutical compositions | |
| PH17562A (en) | 2-guanidino-4-heteroarylthiazoles and pharmaceutical compositions | |
| PH20168A (en) | 7-carboxymethoxyphenylacetamino-3-cephem derivatives and their pharmaceutical compositions | |
| IL68817A0 (en) | Oxoazetidine derivatives,their preparation and pharmaceutical compositions containing them | |
| ZW16583A1 (en) | Milbemycind derivatives their preparation and compositions containing them | |
| NZ209095A (en) | Piperidinoquinazolines and pharmaceutical compositions | |
| NZ208244A (en) | Phenyl-pyrazol-3-ones and pharmaceutical compositions | |
| NZ208694A (en) | Rooperol derivatives and pharmaceutical compositions | |
| DE3473444D1 (en) | Acylindole derivatives and pharmaceutical compositions containing them | |
| IL68496A (en) | 8-heteroarylalkyl-ergoline derivatives,their preparation and pharmaceutical compositions containing them | |
| AU576739B2 (en) | 2-piperazinyl-or-homo-piperazinyl-quinazoline derivatives and pharmaceutical compositions | |
| PH19575A (en) | Cephalosporing derivatives and pharmaceutical compositions thereof | |
| DE3380093D1 (en) | 3-aminopropoxyphenyl derivatives, their preparation and pharmaceutical compositions containing them | |
| IL73224A (en) | 2-dioxacycloalkylthiopenem derivatives and pharmaceutical compositions containing them | |
| NZ205732A (en) | Thiatriazine derivatives and pharmaceutical compositions |