PH12014501653A1 - Metalloenzyme inhibitor compounds - Google Patents
Metalloenzyme inhibitor compoundsInfo
- Publication number
- PH12014501653A1 PH12014501653A1 PH12014501653A PH12014501653A PH12014501653A1 PH 12014501653 A1 PH12014501653 A1 PH 12014501653A1 PH 12014501653 A PH12014501653 A PH 12014501653A PH 12014501653 A PH12014501653 A PH 12014501653A PH 12014501653 A1 PH12014501653 A1 PH 12014501653A1
- Authority
- PH
- Philippines
- Prior art keywords
- inhibitor compounds
- metalloenzyme inhibitor
- metalloenzyme
- compounds
- present disclosure
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/713—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
- A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
- A01N57/16—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing heterocyclic radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Wood Science & Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Preventing Corrosion Or Incrustation Of Metals (AREA)
- Catching Or Destruction (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261589064P | 2012-01-20 | 2012-01-20 | |
| PCT/US2013/022317 WO2013110002A1 (en) | 2012-01-20 | 2013-01-18 | Metalloenzyme inhibitor compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH12014501653A1 true PH12014501653A1 (en) | 2014-10-13 |
Family
ID=48799720
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH12014501653A PH12014501653A1 (en) | 2012-01-20 | 2014-07-18 | Metalloenzyme inhibitor compounds |
Country Status (17)
Families Citing this family (46)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR201900242T4 (tr) | 2009-10-07 | 2019-02-21 | Dow Agrosciences Llc | Hububatta Mantarın Kontrol Altına Alınmasına Yönelik Sinerjistik Fungisidal Karışımlar |
| JP6223329B2 (ja) | 2011-06-23 | 2017-11-01 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素化合物 |
| IN2014DN06792A (cg-RX-API-DMAC10.html) | 2012-01-20 | 2015-05-22 | Viamet Pharmaceuticals Inc | |
| PL2938191T3 (pl) | 2012-12-28 | 2018-07-31 | Dow Agrosciences Llc | Synergistyczne mieszaniny grzybobójcze do zwalczania grzybów w zbożach |
| MX2015008562A (es) | 2012-12-31 | 2015-09-07 | Dow Agrosciences Llc | Pocolinamidas macrociclicas como fungicidas. |
| WO2015100181A1 (en) | 2013-12-26 | 2015-07-02 | Dow Agrosciences Llc | Macrocyclic picolinamide compounds with fungicidal activity |
| WO2015100183A1 (en) | 2013-12-26 | 2015-07-02 | Dow Agrosciences Llc | Macrocyclic picolinamides as fungicides |
| JP6518683B2 (ja) * | 2014-03-19 | 2019-05-22 | ヴィアメット ファーマスーティカルズ（エヌシー），インコーポレイテッド | 抗真菌化合物の調製方法 |
| AU2015231234B2 (en) * | 2014-03-19 | 2019-04-04 | Mycovia Pharmaceuticals, Inc. | Antifungal compound process |
| US9802914B2 (en) | 2014-03-19 | 2017-10-31 | Viamet Pharmaceuticals, Inc. | Antifungal compound process |
| BR112016021282A8 (pt) | 2014-03-19 | 2021-07-20 | The Us Secretary Department Of Health & Human Services | processos para a preparação de compostos antifúngicos e os referidos compostos |
| AU2015231220B2 (en) * | 2014-03-19 | 2019-04-04 | The United States Of America, As Represented By The Secretary, Department Of Health & Human Services | Antifungal compound process |
| AU2015231216B2 (en) * | 2014-03-19 | 2019-04-04 | Mycovia Pharmaceuticals, Inc. | Antifungal compound process |
| JP6633539B2 (ja) | 2014-03-19 | 2020-01-22 | ダウ アグロサイエンシィズ エルエルシー | ２−（２，４−ジフルオロフェニル）−１，１−ジフルオロ−１−（５−置換−ピリジン−２−イル）−３−（１ｈ−テトラゾール−１−イル）プロパン−２−オールおよびその調製工程 |
| JP2017514790A (ja) * | 2014-03-19 | 2017-06-08 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 抗真菌化合物の調製方法 |
| US9914726B2 (en) | 2014-03-19 | 2018-03-13 | Vps-3, Inc. | 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1H-tetrazol-1-yl)propan-2-ols and processes for their preparation |
| EP3119745B1 (en) | 2014-03-19 | 2020-08-05 | Mycovia Pharmaceuticals, Inc. | Antifungal compound process |
| CA2945674A1 (en) | 2014-04-15 | 2015-10-22 | Dow Agrosciences Llc | Metalloenzyme inhibitor compounds as fungicides |
| US9663491B2 (en) | 2014-04-15 | 2017-05-30 | Dow Agrosciences Llc | Metalloenzyme inhibitor compounds as fungicides |
| BR112016025397A2 (pt) | 2014-05-06 | 2017-08-15 | Dow Agrosciences Llc | picolinamidas macrocíclicas como fungicidas |
| CN106470982A (zh) | 2014-07-08 | 2017-03-01 | 美国陶氏益农公司 | 作为杀真菌剂的大环吡啶酰胺 |
| US9686984B2 (en) | 2014-07-08 | 2017-06-27 | Dow Agrosciences Llc | Macrocyclic picolinamides as fungicides |
| US10188109B2 (en) | 2014-12-30 | 2019-01-29 | Dow Agrosciences Llc | Picolinamide compounds with fungicidal activity |
| BR112017013589A2 (pt) | 2014-12-30 | 2018-03-06 | Dow Agrosciences Llc | picolinamidas com atividade fungicida |
| CN107105654B (zh) | 2014-12-30 | 2021-03-02 | 美国陶氏益农公司 | 杀真菌组合物 |
| KR20170100620A (ko) | 2014-12-30 | 2017-09-04 | 다우 아그로사이언시즈 엘엘씨 | 살진균제로서의 피콜린아미드의 용도 |
| MX2017008422A (es) * | 2014-12-30 | 2017-10-02 | Dow Agrosciences Llc | Compuestos de picolinamida con actividad fungicida. |
| CN107426999B (zh) | 2014-12-30 | 2023-01-20 | 美国陶氏益农公司 | 具有杀真菌活性的吡啶酰胺化合物 |
| SI3271347T1 (sl) * | 2015-03-19 | 2022-11-30 | Mycovia Pharmaceuticals, Inc. | Protiglivične spojine in postopki za izdelavo |
| AU2016323782B2 (en) | 2015-09-18 | 2020-11-26 | Nqp 1598, Ltd. | Antifungal compound process |
| EA038421B1 (ru) * | 2015-12-30 | 2021-08-26 | ВиПиЭс-3, ИНК. | Соединения, ингибирующие металлоферменты |
| WO2018045003A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Picolinamide n-oxide compounds with fungicidal activity |
| WO2018045012A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Pyrido-1,3-oxazine-2,4-dione compounds with fungicidal activity |
| US10172358B2 (en) | 2016-08-30 | 2019-01-08 | Dow Agrosciences Llc | Thiopicolinamide compounds with fungicidal activity |
| WO2018045000A1 (en) | 2016-08-30 | 2018-03-08 | Dow Agrosciences Llc | Picolinamides as fungicides |
| BR102018000183B1 (pt) | 2017-01-05 | 2023-04-25 | Dow Agrosciences Llc | Picolinamidas, composição para controle de um patógeno fúngico, e método para controle e prevenção de um ataque por fungos em uma planta |
| US20200045967A1 (en) * | 2017-02-08 | 2020-02-13 | Bayer Cropscience Aktiengesellschaft | Novel triazole derivatives |
| TW201842851A (zh) | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
| TWI774761B (zh) | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
| CN110996665B (zh) | 2017-05-02 | 2021-10-26 | 陶氏益农公司 | 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途 |
| BR102019004480B1 (pt) | 2018-03-08 | 2023-03-28 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
| CA3115684A1 (en) | 2018-10-15 | 2020-04-23 | Dow Agrosciences Llc | Methods for sythesis of oxypicolinamides |
| CN114554848A (zh) | 2019-10-18 | 2022-05-27 | 科迪华农业科技有限责任公司 | 用于合成吡啶酰胺的方法 |
| CN110981810A (zh) * | 2019-12-19 | 2020-04-10 | 东莞市维琪科技有限公司 | 一种脱羧肌肽的合成方法 |
| TW202140445A (zh) * | 2020-01-17 | 2021-11-01 | 大陸商上海森輝醫藥有限公司 | 四氮唑類化合物的可藥用鹽及其結晶形式、製備方法和用途 |
| WO2026006142A1 (en) * | 2024-06-24 | 2026-01-02 | The United States Of America, As Represented By The Secretary, Dept. Of Health And Human Services | Azole compounds useful as inhibitors of voltage-dependent anion channel oligomerization |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0117100B1 (en) * | 1983-02-16 | 1986-12-10 | Pfizer Limited | Triazole antifungal agents |
| GB8304282D0 (en) * | 1983-02-16 | 1983-03-23 | Pfizer Ltd | Antifungal agents |
| US5358939A (en) * | 1992-06-25 | 1994-10-25 | Rohm And Haas Company | Fungicidal 2-aryl-2,2-disubstituted ethyl-1,2,4-triazoles |
| MY115814A (en) | 1995-06-16 | 2003-09-30 | Bayer Ip Gmbh | Crop protection compositions |
| CN1187756A (zh) * | 1995-06-16 | 1998-07-15 | 诺瓦提斯公司 | 保护作物的组合物 |
| JP2006143593A (ja) * | 2004-11-16 | 2006-06-08 | Hokko Chem Ind Co Ltd | Ｎ−ベンジルテトラゾール誘導体および農園芸用殺菌剤 |
| WO2010005572A2 (en) * | 2008-07-09 | 2010-01-14 | The Scripps Research Institute | Alpha-keto heterocycles as faah inhibitors |
| BRPI0918058A8 (pt) * | 2008-09-03 | 2016-03-01 | Bayer Cropscience Ag | Uso de composições de composto fungicida para o controle de certos fungos da ferrugem |
| CA2785898C (en) * | 2009-12-31 | 2018-07-03 | Viamet Pharmaceuticals, Inc. | Metalloenzyme inhibitor compounds |
| KR101379370B1 (ko) * | 2010-04-24 | 2014-03-28 | 비아멧 파마슈티컬즈, 인코포레이티드 | 금속효소 억제제 화합물 |
| JP6223329B2 (ja) * | 2011-06-23 | 2017-11-01 | ヴィアメット ファーマスーティカルズ，インコーポレイテッド | 金属酵素化合物 |
-
2013
- 2013-01-18 BR BR112014017799A patent/BR112014017799A8/pt not_active IP Right Cessation
- 2013-01-18 CA CA2861341A patent/CA2861341A1/en not_active Abandoned
- 2013-01-18 EA EA201491386A patent/EA201491386A1/ru unknown
- 2013-01-18 CN CN201380010205.1A patent/CN104135861A/zh active Pending
- 2013-01-18 KR KR1020147023021A patent/KR20140116515A/ko not_active Withdrawn
- 2013-01-18 WO PCT/US2013/022317 patent/WO2013110002A1/en not_active Ceased
- 2013-01-18 AU AU2013209520A patent/AU2013209520A1/en not_active Abandoned
- 2013-01-18 US US14/373,304 patent/US9414596B2/en not_active Expired - Fee Related
- 2013-01-18 EP EP13739106.6A patent/EP2804479A4/en not_active Withdrawn
- 2013-01-18 IN IN6812DEN2014 patent/IN2014DN06812A/en unknown
- 2013-01-18 MX MX2014008729A patent/MX2014008729A/es unknown
- 2013-01-18 JP JP2014553493A patent/JP2015505538A/ja not_active Ceased
-
2014
- 2014-07-17 CL CL2014001892A patent/CL2014001892A1/es unknown
- 2014-07-18 PH PH12014501653A patent/PH12014501653A1/en unknown
- 2014-08-14 CO CO14178605A patent/CO7111289A2/es not_active Application Discontinuation
- 2014-08-18 EC ECIEPI201414530A patent/ECSP14014530A/es unknown
- 2014-08-18 CR CR20140387A patent/CR20140387A/es unknown
-
2016
- 2016-12-15 JP JP2016243478A patent/JP2017110004A/ja active Pending
-
2019
- 2019-02-05 JP JP2019018600A patent/JP2019116476A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU2013209520A1 (en) | 2014-08-28 |
| BR112014017799A8 (pt) | 2017-07-11 |
| KR20140116515A (ko) | 2014-10-02 |
| WO2013110002A1 (en) | 2013-07-25 |
| JP2017110004A (ja) | 2017-06-22 |
| IN2014DN06812A (cg-RX-API-DMAC10.html) | 2015-05-22 |
| ECSP14014530A (es) | 2015-06-30 |
| EA201491386A1 (ru) | 2014-11-28 |
| EP2804479A1 (en) | 2014-11-26 |
| CO7111289A2 (es) | 2014-11-10 |
| BR112014017799A2 (cg-RX-API-DMAC10.html) | 2017-06-20 |
| MX2014008729A (es) | 2015-02-04 |
| JP2019116476A (ja) | 2019-07-18 |
| JP2015505538A (ja) | 2015-02-23 |
| CA2861341A1 (en) | 2013-07-25 |
| CL2014001892A1 (es) | 2014-11-14 |
| CR20140387A (es) | 2014-11-27 |
| CN104135861A (zh) | 2014-11-05 |
| US20150024938A1 (en) | 2015-01-22 |
| US9414596B2 (en) | 2016-08-16 |
| EP2804479A4 (en) | 2015-07-22 |
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