PE20061297A1 - Compuestos derivados de cromano y cromeno moduladores del receptor de serotonina 5-ht2c - Google Patents

Compuestos derivados de cromano y cromeno moduladores del receptor de serotonina 5-ht2c

Info

Publication number
PE20061297A1
PE20061297A1 PE2006000415A PE2006000415A PE20061297A1 PE 20061297 A1 PE20061297 A1 PE 20061297A1 PE 2006000415 A PE2006000415 A PE 2006000415A PE 2006000415 A PE2006000415 A PE 2006000415A PE 20061297 A1 PE20061297 A1 PE 20061297A1
Authority
PE
Peru
Prior art keywords
chrome
aliphatic
serotonin
ht2c receptor
chromen
Prior art date
Application number
PE2006000415A
Other languages
English (en)
Spanish (es)
Inventor
Gavin David Heffernan
Gary Paul Stack
Dahui Zhou
Hong Gao
Jonathan Laird Gross
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of PE20061297A1 publication Critical patent/PE20061297A1/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/06—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2
    • C07D311/20—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 2 hydrogenated in the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
    • C07D313/02—Seven-membered rings
    • C07D313/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D313/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
PE2006000415A 2005-04-22 2006-04-21 Compuestos derivados de cromano y cromeno moduladores del receptor de serotonina 5-ht2c PE20061297A1 (es)

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US67382005P 2005-04-22 2005-04-22

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EP (1) EP1874756A1 (US20060258714A1-20061116-C00165.png)
JP (1) JP2008538576A (US20060258714A1-20061116-C00165.png)
KR (1) KR20080008378A (US20060258714A1-20061116-C00165.png)
CN (1) CN101203505A (US20060258714A1-20061116-C00165.png)
AR (1) AR056320A1 (US20060258714A1-20061116-C00165.png)
AU (1) AU2006239937A1 (US20060258714A1-20061116-C00165.png)
BR (1) BRPI0610027A2 (US20060258714A1-20061116-C00165.png)
CA (1) CA2605587A1 (US20060258714A1-20061116-C00165.png)
CO (1) CO6321153A2 (US20060258714A1-20061116-C00165.png)
GT (1) GT200600166A (US20060258714A1-20061116-C00165.png)
IL (1) IL186837A0 (US20060258714A1-20061116-C00165.png)
MX (1) MX2007013163A (US20060258714A1-20061116-C00165.png)
NO (1) NO20075641L (US20060258714A1-20061116-C00165.png)
PE (1) PE20061297A1 (US20060258714A1-20061116-C00165.png)
RU (1) RU2007139541A (US20060258714A1-20061116-C00165.png)
TW (1) TW200716595A (US20060258714A1-20061116-C00165.png)
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AU2006239937A1 (en) 2006-11-02
TW200716595A (en) 2007-05-01
US20080182891A1 (en) 2008-07-31
WO2006116165A1 (en) 2006-11-02
KR20080008378A (ko) 2008-01-23
GT200600166A (es) 2007-03-14
US7365095B2 (en) 2008-04-29
CN101203505A (zh) 2008-06-18
JP2008538576A (ja) 2008-10-30
BRPI0610027A2 (pt) 2010-05-18
US20060258714A1 (en) 2006-11-16
CO6321153A2 (es) 2011-09-20
CA2605587A1 (en) 2006-11-02
ZA200709052B (en) 2009-08-26
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IL186837A0 (en) 2008-02-09

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