NZ597638A - 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives - Google Patents

5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Info

Publication number
NZ597638A
NZ597638A NZ597638A NZ59763810A NZ597638A NZ 597638 A NZ597638 A NZ 597638A NZ 597638 A NZ597638 A NZ 597638A NZ 59763810 A NZ59763810 A NZ 59763810A NZ 597638 A NZ597638 A NZ 597638A
Authority
NZ
New Zealand
Prior art keywords
fluoro
oxopyrimidine
amino
carboxylate
optionally substituted
Prior art date
Application number
NZ597638A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ597638(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of NZ597638A publication Critical patent/NZ597638A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
NZ597638A 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives NZ597638A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07
PCT/US2010/044585 WO2011017544A1 (en) 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Publications (1)

Publication Number Publication Date
NZ597638A true NZ597638A (en) 2014-06-27

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ597638A NZ597638A (en) 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Country Status (28)

Country Link
US (1) US8318758B2 (esLanguage)
EP (1) EP2462133B1 (esLanguage)
JP (1) JP5818791B2 (esLanguage)
KR (1) KR101792286B1 (esLanguage)
CN (1) CN102548979B (esLanguage)
AU (1) AU2010279408B2 (esLanguage)
BR (1) BR112012002807B1 (esLanguage)
CA (1) CA2769251C (esLanguage)
CL (1) CL2012000314A1 (esLanguage)
CO (1) CO6491089A2 (esLanguage)
CR (1) CR20120033A (esLanguage)
DK (1) DK2462133T3 (esLanguage)
EA (1) EA022930B1 (esLanguage)
EC (1) ECSP12011651A (esLanguage)
ES (1) ES2506169T3 (esLanguage)
HN (1) HN2012000261A (esLanguage)
IL (1) IL217954A (esLanguage)
IN (1) IN2012DN00695A (esLanguage)
MX (1) MX2012001623A (esLanguage)
NI (1) NI201200019A (esLanguage)
NZ (1) NZ597638A (esLanguage)
PE (1) PE20120689A1 (esLanguage)
PL (1) PL2462133T3 (esLanguage)
PT (1) PT2462133E (esLanguage)
RS (1) RS53658B1 (esLanguage)
UA (1) UA106086C2 (esLanguage)
WO (1) WO2011017544A1 (esLanguage)
ZA (1) ZA201305992B (esLanguage)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2769073C (en) * 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
CN110003118A (zh) * 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 制备羧酸酯衍生物的方法
CA2893776A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
KR20150100869A (ko) 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
SG11201605372QA (en) 2013-12-31 2016-08-30 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
HUE072634T2 (hu) 2013-12-31 2025-11-28 Adama Makhteshim Ltd Szinergikus fungicid keverékek gomba elleni védekezésre gabonafélékben
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
CN108472290A (zh) 2015-11-06 2018-08-31 萨穆梅德有限公司 治疗骨关节炎
PT3464285T (pt) 2016-06-01 2022-12-20 Biosplice Therapeutics Inc Processo para preparar n-(5-(3-(7-(3-fluorofenil)-3himidazo[4,5-c]piridin-2-il)-1h-indazol-5-il)piridin-3-il)-3-metilbutanamida
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
MA54148A (fr) 2018-11-05 2022-02-09 Adama Makhteshim Ltd Mélanges et compositions comprenant de la 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one et leurs procédés d'utilisation
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US6262058B1 (en) 1996-03-11 2001-07-17 Syngenta Crop Protection, Inc. Pyrimidin-4-one derivatives as pesticide
AU2003274652A1 (en) * 2002-10-23 2004-05-13 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
PL2151439T3 (pl) * 2007-04-27 2014-08-29 Daiichi Sankyo Co Ltd Pochodna z wprowadzonym atomem azotu i 6-członowym pierścieniem aromatycznym oraz zawierający ją środek farmaceutyczny
JP5580310B2 (ja) 2008-08-01 2014-08-27 ダウ アグロサイエンシィズ エルエルシー 殺真菌剤としての５−フルオロシトシンの使用

Also Published As

Publication number Publication date
JP5818791B2 (ja) 2015-11-18
RS53658B1 (sr) 2015-04-30
US20110034491A1 (en) 2011-02-10
PE20120689A1 (es) 2012-06-06
DK2462133T3 (en) 2015-01-05
ES2506169T3 (es) 2014-10-13
KR20120043069A (ko) 2012-05-03
BR112012002807A2 (pt) 2015-10-13
BR112012002807A8 (pt) 2017-07-11
IL217954A (en) 2016-02-29
CA2769251A1 (en) 2011-02-10
EP2462133A4 (en) 2013-01-16
CR20120033A (es) 2012-03-22
CN102548979B (zh) 2015-05-13
EA022930B1 (ru) 2016-03-31
BR112012002807B1 (pt) 2018-07-10
IL217954A0 (en) 2012-03-29
KR101792286B1 (ko) 2017-10-31
US8318758B2 (en) 2012-11-27
CN102548979A (zh) 2012-07-04
HN2012000261A (es) 2015-01-05
AU2010279408B2 (en) 2015-09-10
PL2462133T3 (pl) 2015-03-31
UA106086C2 (uk) 2014-07-25
ZA201305992B (en) 2014-10-29
AU2010279408A1 (en) 2012-02-09
CA2769251C (en) 2018-05-15
CL2012000314A1 (es) 2012-10-05
EA201270255A1 (ru) 2012-07-30
PT2462133E (pt) 2014-12-26
EP2462133B1 (en) 2014-09-24
EP2462133A1 (en) 2012-06-13
JP2013501726A (ja) 2013-01-17
WO2011017544A1 (en) 2011-02-10
ECSP12011651A (es) 2012-03-30
MX2012001623A (es) 2012-04-11
NI201200019A (es) 2012-05-22
CO6491089A2 (es) 2012-07-31
HK1172892A1 (en) 2013-05-03
IN2012DN00695A (esLanguage) 2015-06-19

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