NZ594010A - Novel forms of bendamustine free base - Google Patents

Novel forms of bendamustine free base

Info

Publication number
NZ594010A
NZ594010A NZ594010A NZ59401010A NZ594010A NZ 594010 A NZ594010 A NZ 594010A NZ 594010 A NZ594010 A NZ 594010A NZ 59401010 A NZ59401010 A NZ 59401010A NZ 594010 A NZ594010 A NZ 594010A
Authority
NZ
New Zealand
Prior art keywords
free base
bendamustine free
forms
novel forms
bendamustine
Prior art date
Application number
NZ594010A
Other languages
English (en)
Inventor
Mark Eddleston
Curtis R Haltiwanger
Laurent D Courvoisier
Robert E Mckean
Original Assignee
Cephalon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42008533&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ594010(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cephalon Inc filed Critical Cephalon Inc
Publication of NZ594010A publication Critical patent/NZ594010A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/16—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
NZ594010A 2009-01-15 2010-01-14 Novel forms of bendamustine free base NZ594010A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14484309P 2009-01-15 2009-01-15
PCT/US2010/020992 WO2010083276A1 (en) 2009-01-15 2010-01-14 Novel forms of bendamustine free base

Publications (1)

Publication Number Publication Date
NZ594010A true NZ594010A (en) 2013-08-30

Family

ID=42008533

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ594010A NZ594010A (en) 2009-01-15 2010-01-14 Novel forms of bendamustine free base

Country Status (16)

Country Link
US (1) US8076366B2 (cg-RX-API-DMAC7.html)
EP (1) EP2387400A1 (cg-RX-API-DMAC7.html)
JP (1) JP2012515210A (cg-RX-API-DMAC7.html)
KR (1) KR20110110293A (cg-RX-API-DMAC7.html)
CN (2) CN102281877B (cg-RX-API-DMAC7.html)
AU (2) AU2010204765A1 (cg-RX-API-DMAC7.html)
BR (1) BRPI1004922A2 (cg-RX-API-DMAC7.html)
CA (1) CA2749101A1 (cg-RX-API-DMAC7.html)
EA (1) EA020767B1 (cg-RX-API-DMAC7.html)
IL (1) IL213725A0 (cg-RX-API-DMAC7.html)
MX (1) MX2011007557A (cg-RX-API-DMAC7.html)
NZ (1) NZ594010A (cg-RX-API-DMAC7.html)
SG (1) SG172810A1 (cg-RX-API-DMAC7.html)
UA (1) UA109109C2 (cg-RX-API-DMAC7.html)
WO (1) WO2010083276A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA201105099B (cg-RX-API-DMAC7.html)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9376394B2 (en) * 2009-12-23 2016-06-28 Dr. Reddy's Laboratories Ltd. Preparation of bendamustine and its salts
EP3895694A1 (en) 2010-01-28 2021-10-20 Eagle Pharmaceuticals, Inc. Formulations of bendamustine
WO2012176214A2 (en) * 2011-06-20 2012-12-27 Hetero Research Foundation Process for bendamustine hydrochloride
RS58744B1 (sr) 2012-03-20 2019-06-28 Eagle Pharmaceuticals Inc Tečna kompozicija za upotrebu u postupku lečenja stanja koja reaguju na bendamustin kod pacijenata kojima su potrebne smanjene zapremine za davanje
DK2827862T3 (da) 2012-03-20 2024-02-12 Eagle Pharmaceuticals Inc Formuleringer af bendamustin
US20230241218A1 (en) * 2012-07-10 2023-08-03 Eagle Pharmaceuticals, Inc. Formulations of bendamustine
MX362032B (es) 2013-03-12 2019-01-04 Cephalon Inc Formulaciones nanoparticuladas y macroparticuladas.
EP2988655B1 (en) 2013-04-26 2023-04-12 Genentech, Inc. Contour integration perimetry vision test
US20240148696A1 (en) 2022-10-25 2024-05-09 Softkemo Pharma Inc. Lyophilized bendamustine-cyclodextrin composition

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DE10306724A1 (de) 2002-02-28 2003-09-18 G O T Therapeutics Gmbh Vesikuläre Verkapselung von Bendamustin
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Also Published As

Publication number Publication date
KR20110110293A (ko) 2011-10-06
MX2011007557A (es) 2011-08-12
BRPI1004922A2 (pt) 2019-09-24
ZA201105099B (en) 2012-03-28
EA020767B1 (ru) 2015-01-30
EA201170934A1 (ru) 2011-12-30
CA2749101A1 (en) 2010-07-22
CN102281877A (zh) 2011-12-14
CN103554030A (zh) 2014-02-05
AU2016204902A1 (en) 2016-08-04
SG172810A1 (en) 2011-08-29
EP2387400A1 (en) 2011-11-23
UA109109C2 (uk) 2015-07-27
IL213725A0 (en) 2011-07-31
US8076366B2 (en) 2011-12-13
CN102281877B (zh) 2014-07-23
WO2010083276A1 (en) 2010-07-22
JP2012515210A (ja) 2012-07-05
AU2010204765A1 (en) 2011-07-28
US20100210701A1 (en) 2010-08-19

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Effective date: 20140828

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Effective date: 20140829