NZ575030A - Histone deacetylase inhibitors with combined activity on class-I and class-IIb histone deacetylases in combination with proteasome inhibitors - Google Patents

Histone deacetylase inhibitors with combined activity on class-I and class-IIb histone deacetylases in combination with proteasome inhibitors

Info

Publication number
NZ575030A
NZ575030A NZ575030A NZ57503007A NZ575030A NZ 575030 A NZ575030 A NZ 575030A NZ 575030 A NZ575030 A NZ 575030A NZ 57503007 A NZ57503007 A NZ 57503007A NZ 575030 A NZ575030 A NZ 575030A
Authority
NZ
New Zealand
Prior art keywords
leukemia
combination
drug resistant
acute
inhibitor
Prior art date
Application number
NZ575030A
Other languages
English (en)
Inventor
Janine Arts
Peter Willem Jan Hellemans
Michel Marie Francois Janicot
Martin John Page
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Priority claimed from PCT/EP2007/059518 external-priority patent/WO2008031817A2/en
Publication of NZ575030A publication Critical patent/NZ575030A/en

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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NZ575030A 2006-09-15 2007-09-11 Histone deacetylase inhibitors with combined activity on class-I and class-IIb histone deacetylases in combination with proteasome inhibitors NZ575030A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP06120726 2006-09-15
US91589507P 2007-05-03 2007-05-03
PCT/EP2007/059518 WO2008031817A2 (en) 2006-09-15 2007-09-11 Histone deacetylase inhibitors with combined activity on class-i and class-iib histone deacetylases in combination with proteasome inhibitors

Publications (1)

Publication Number Publication Date
NZ575030A true NZ575030A (en) 2012-07-27

Family

ID=41040414

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ575030A NZ575030A (en) 2006-09-15 2007-09-11 Histone deacetylase inhibitors with combined activity on class-I and class-IIb histone deacetylases in combination with proteasome inhibitors

Country Status (12)

Country Link
CN (1) CN101516374B (zh)
BR (1) BRPI0716992A2 (zh)
DK (1) DK2066327T3 (zh)
ES (1) ES2399670T3 (zh)
ME (1) ME01514B (zh)
NZ (1) NZ575030A (zh)
PT (1) PT2066327E (zh)
RS (1) RS52638B (zh)
SG (1) SG177219A1 (zh)
SI (1) SI2066327T1 (zh)
UA (1) UA97249C2 (zh)
ZA (1) ZA200901818B (zh)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8957066B2 (en) * 2011-02-28 2015-02-17 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
CN107095871A (zh) * 2016-02-22 2017-08-29 中国科学院上海巴斯德研究所 Quisinostat,一种新型的高效抗疟药物
KR20190030693A (ko) * 2016-07-20 2019-03-22 더 트러스티이스 오브 콜롬비아 유니버시티 인 더 시티 오브 뉴욕 히스톤 아세틸트랜스퍼라제 활성화제 및 이의 조성물 및 용도
CN114409638B (zh) * 2022-02-09 2023-02-14 深圳大学 组蛋白去乙酰化酶8选择性降解剂、制备方法及其在抗肿瘤活性中的应用
CN115028678A (zh) * 2022-07-08 2022-09-09 杭州医学院 基于vhl配体诱导bcr-abl蛋白降解的双功能分子及其制备方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006010750A1 (en) * 2004-07-28 2006-02-02 Janssen Pharmaceutica N.V. Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase

Also Published As

Publication number Publication date
BRPI0716992A2 (pt) 2013-09-17
ZA200901818B (en) 2010-05-26
PT2066327E (pt) 2013-02-06
ME01514B (me) 2014-04-20
SI2066327T1 (sl) 2013-04-30
SG177219A1 (en) 2012-01-30
CN101516374A (zh) 2009-08-26
UA97249C2 (ru) 2012-01-25
CN101516374B (zh) 2013-04-24
RS52638B (en) 2013-06-28
DK2066327T3 (da) 2013-02-11
ES2399670T3 (es) 2013-04-02

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