PT2066327E - Inibidores de histona deacetilase com atividade combinada sobre histona deacetilases da classe i e da classe iib, em combinação com inibidores de proteassoma - Google Patents

Inibidores de histona deacetilase com atividade combinada sobre histona deacetilases da classe i e da classe iib, em combinação com inibidores de proteassoma

Info

Publication number
PT2066327E
PT2066327E PT78033974T PT07803397T PT2066327E PT 2066327 E PT2066327 E PT 2066327E PT 78033974 T PT78033974 T PT 78033974T PT 07803397 T PT07803397 T PT 07803397T PT 2066327 E PT2066327 E PT 2066327E
Authority
PT
Portugal
Prior art keywords
class
inhibitors
combination
histone
iib
Prior art date
Application number
PT78033974T
Other languages
English (en)
Portuguese (pt)
Inventor
Janine Arts
Peter Willem Jan Hellemans
Michel Marie Francois Janicot
Martin John Page
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PT2066327E publication Critical patent/PT2066327E/pt

Links

PT78033974T 2006-09-15 2007-09-11 Inibidores de histona deacetilase com atividade combinada sobre histona deacetilases da classe i e da classe iib, em combinação com inibidores de proteassoma PT2066327E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06120726 2006-09-15
US91589507P 2007-05-03 2007-05-03

Publications (1)

Publication Number Publication Date
PT2066327E true PT2066327E (pt) 2013-02-06

Family

ID=41040414

Family Applications (1)

Application Number Title Priority Date Filing Date
PT78033974T PT2066327E (pt) 2006-09-15 2007-09-11 Inibidores de histona deacetilase com atividade combinada sobre histona deacetilases da classe i e da classe iib, em combinação com inibidores de proteassoma

Country Status (12)

Country Link
CN (1) CN101516374B (zh)
BR (1) BRPI0716992A2 (zh)
DK (1) DK2066327T3 (zh)
ES (1) ES2399670T3 (zh)
ME (1) ME01514B (zh)
NZ (1) NZ575030A (zh)
PT (1) PT2066327E (zh)
RS (1) RS52638B (zh)
SG (1) SG177219A1 (zh)
SI (1) SI2066327T1 (zh)
UA (1) UA97249C2 (zh)
ZA (1) ZA200901818B (zh)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8957066B2 (en) * 2011-02-28 2015-02-17 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
CN107095871A (zh) * 2016-02-22 2017-08-29 中国科学院上海巴斯德研究所 Quisinostat,一种新型的高效抗疟药物
JP2019527226A (ja) * 2016-07-20 2019-09-26 ザ トラスティース オブ コロンビア ユニバーシティ イン ザ シティ オブ ニューヨーク ヒストンアセチルトランスフェラーゼ活性化剤及び組成物並びにそれらの使用
CN114409638B (zh) * 2022-02-09 2023-02-14 深圳大学 组蛋白去乙酰化酶8选择性降解剂、制备方法及其在抗肿瘤活性中的应用
CN115028678A (zh) * 2022-07-08 2022-09-09 杭州医学院 基于vhl配体诱导bcr-abl蛋白降解的双功能分子及其制备方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4948403B2 (ja) * 2004-07-28 2012-06-06 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストン・デアセチラーゼの新インヒビターとしての置換インドリルアルキルアミノ誘導体

Also Published As

Publication number Publication date
SI2066327T1 (sl) 2013-04-30
CN101516374A (zh) 2009-08-26
DK2066327T3 (da) 2013-02-11
BRPI0716992A2 (pt) 2013-09-17
CN101516374B (zh) 2013-04-24
ES2399670T3 (es) 2013-04-02
RS52638B (en) 2013-06-28
ME01514B (me) 2014-04-20
NZ575030A (en) 2012-07-27
ZA200901818B (en) 2010-05-26
UA97249C2 (ru) 2012-01-25
SG177219A1 (en) 2012-01-30

Similar Documents

Publication Publication Date Title
HK1136770A1 (en) Histone deacetylase inhibitors with combined activity on class-i and class- iib histone deacetylases in combination with proteasome inhibitors
HK1133199A1 (zh) 組蛋白脫乙酰基酶和微管蛋白脫乙酰基酶抑制劑
ZA200905060B (en) Method of using histone deacetylase inhibitors and monitoring biomarkers in combination therapy
HK1161583A1 (zh) 脫乙酰酶抑制劑和其用途
HK1220179A1 (zh) 組蛋白去乙酰的抑制劑
EP1973872A4 (en) HISTONDEACETYLASE HEMMER AND PROPHARMAKA THEREOF
EP1940805A4 (en) BENZODIAZEPIN AND BENZOPIPERAZINANALOGA AS INHIBITORS OF HISTONDEACETYLASE
EP1991247A4 (en) BIFUNCTIONAL HISTONE DEACETYLASE INHIBITORS
HK1135902A1 (en) Combinations of class-i specific histone deacetylase inhibitors with proteasome inhibitors
EP1991951A4 (en) PORTABLE CASHING SYSTEMS AND METHOD
IL188692A0 (en) Histone deacetylase inhibitors
EP1945617A4 (en) HISTONDEACETYLASEINHIBITORS WITH ARYLPYRAZOLYL MOTIVES
IL193458A0 (en) Histone deacetylase inhibitors
EP1771167A4 (en) INHIBITORS OF HISTONE DEACETYLASE
EP1735319A4 (en) Histone deacetylase INHIBITORS
IL205241A0 (en) Histone deacetylase inhibitors
IL198263A0 (en) Hydroxamates as inhibitors of histone deacetylase
EP1991226A4 (en) Histone deacetylase INHIBITORS
EP2308868A4 (en) HISTONDEACETYLASEINHIBITORS AND APPLICATIONS THEREOF
IL214244A (en) Diastylase Heisone Inhibitors and their use in healing
EP2208721A4 (en) HISTONE DEACETYLASE INHIBITOR, COMPOSITION AND USE THEREOF
EP1784386A4 (en) HISTONE DEACETYLASE INHIBITORS
EP2089354A4 (en) NAPHTHALENYLOXYPROPENYL DERIVATIVES HAVING HISTONE DEACETYLASE INHIBITORY ACTIVITY AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME
EP1784194A4 (en) HISTONE DEACETYLASE INHIBITORS
AP2007004188A0 (en) Hydroxamates as histone deacetylase inhibitors and pharmaceutical formulations containing them