NZ574654A - Crystalline forms of rapamycin analogs - Google Patents

Crystalline forms of rapamycin analogs

Info

Publication number
NZ574654A
NZ574654A NZ574654A NZ57465407A NZ574654A NZ 574654 A NZ574654 A NZ 574654A NZ 574654 A NZ574654 A NZ 574654A NZ 57465407 A NZ57465407 A NZ 57465407A NZ 574654 A NZ574654 A NZ 574654A
Authority
NZ
New Zealand
Prior art keywords
powder
ray diffraction
diffraction pattern
rapamycin analog
composition
Prior art date
Application number
NZ574654A
Other languages
English (en)
Inventor
Shekhar Viswanath
Larry Bartelt
Robert Leanna
Michael Rasmussen
Madhup Dhaon
Rodger Henry
Thomas Borchardt
Shuang Chen
Geoff Zhang
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/781,804 external-priority patent/US7812032B2/en
Priority claimed from US11/781,807 external-priority patent/US7820812B2/en
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of NZ574654A publication Critical patent/NZ574654A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
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  • Health & Medical Sciences (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Neurology (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Communicable Diseases (AREA)
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  • Toxicology (AREA)
  • Obesity (AREA)
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  • Pain & Pain Management (AREA)
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NZ574654A 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs NZ574654A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US82031706P 2006-07-25 2006-07-25
US11/781,804 US7812032B2 (en) 2006-07-25 2007-07-23 Crystalline forms of rapamycin analogs
US11/781,807 US7820812B2 (en) 2006-07-25 2007-07-23 Methods of manufacturing crystalline forms of rapamycin analogs
PCT/US2007/074159 WO2008014222A1 (en) 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs

Publications (1)

Publication Number Publication Date
NZ574654A true NZ574654A (en) 2012-03-30

Family

ID=38562825

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ574654A NZ574654A (en) 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs

Country Status (10)

Country Link
EP (2) EP2051984A1 (https=)
JP (1) JP2010500286A (https=)
KR (1) KR20090035716A (https=)
AU (1) AU2007276837B2 (https=)
BR (1) BRPI0714945B8 (https=)
CA (1) CA2658896A1 (https=)
IL (1) IL196706A0 (https=)
MX (1) MX2009001067A (https=)
NZ (1) NZ574654A (https=)
WO (1) WO2008014222A1 (https=)

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US7820812B2 (en) 2006-07-25 2010-10-26 Abbott Laboratories Methods of manufacturing crystalline forms of rapamycin analogs
US7812032B2 (en) 2006-07-25 2010-10-12 Abbott Laboratories Crystalline forms of rapamycin analogs
CA2673991C (en) 2007-01-21 2012-02-07 Hemoteq Ag Methods for coating catheter balloons with a defined quantity of active agent
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EP2380006A4 (en) * 2009-01-21 2012-05-16 Biocon Ltd PROCESS FOR DETERMINING THE SIROLIMUS STABILITY AND METHOD FOR PRODUCING ITS STABLE FORM
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WO2013022458A1 (en) * 2011-08-05 2013-02-14 Boston Scientific Scimed, Inc. Methods of converting amorphous drug substance into crystalline form
WO2013028208A1 (en) 2011-08-25 2013-02-28 Boston Scientific Scimed, Inc. Medical device with crystalline drug coating
US9439892B2 (en) 2013-05-16 2016-09-13 Surmodics, Inc. Macrolide particulates, methods for preparation, and medical devices associated therewith
CA2915704C (en) 2013-06-12 2022-06-21 Surmodics, Inc. Solvent methods for preparing crystalline macrolide particulates, compositions, and articles containing particulates
DE102013110294B4 (de) * 2013-09-18 2016-07-07 Innora Gmbh Limus-Depot-Formulierung auf Ballonkathetern
EP3435988B1 (en) 2016-03-31 2021-10-06 Surmodics, Inc. Drug-containing particulate composition with cationic agent, associated medical devices, and methods for treatment
US11123459B2 (en) 2016-12-16 2021-09-21 Surmodics, Inc. Hydrophobic active agent particle coatings and methods for treatment
CN108144131A (zh) * 2017-12-22 2018-06-12 上海微创医疗器械（集团）有限公司 一种载药植入医疗器械及其制备方法
CN119431400A (zh) * 2020-03-27 2025-02-14 波士顿科学国际有限公司 用于使药物结晶的方法
JP2024503898A (ja) * 2021-01-22 2024-01-29 ヤンセン ファーマシューティカ エヌ．ベー． ラパマイシン類似体及びその使用

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EP2407471A3 (en) 2012-06-20
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BRPI0714945B1 (pt) 2020-11-10
WO2008014222A1 (en) 2008-01-31
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AU2007276837B2 (en) 2013-02-07

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