KR20090035716A - 라파마이신 유사체의 결정형 형태 - Google Patents

라파마이신 유사체의 결정형 형태 Download PDF

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KR20090035716A
KR20090035716A KR1020097003955A KR20097003955A KR20090035716A KR 20090035716 A KR20090035716 A KR 20090035716A KR 1020097003955 A KR1020097003955 A KR 1020097003955A KR 20097003955 A KR20097003955 A KR 20097003955A KR 20090035716 A KR20090035716 A KR 20090035716A
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Prior art keywords
powder
ray diffraction
diffraction pattern
composition
peaks
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Korean (ko)
Inventor
셰크하르 비스와나스
래리 바텔트
로버트 레안나
마이클 라스뮤쎈
마드후프 다온
로져 헨리
토마스 보어하르트
솽 천
제프 장
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아보트 러보러터리즈
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Priority claimed from US11/781,804 external-priority patent/US7812032B2/en
Priority claimed from US11/781,807 external-priority patent/US7820812B2/en
Application filed by 아보트 러보러터리즈 filed Critical 아보트 러보러터리즈
Publication of KR20090035716A publication Critical patent/KR20090035716A/ko
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
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KR1020097003955A 2006-07-25 2007-07-24 라파마이신 유사체의 결정형 형태 Ceased KR20090035716A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US82031706P 2006-07-25 2006-07-25
US60/820,317 2006-07-25
US11/781,804 US7812032B2 (en) 2006-07-25 2007-07-23 Crystalline forms of rapamycin analogs
US11/781,804 2007-07-23
US11/781,807 US7820812B2 (en) 2006-07-25 2007-07-23 Methods of manufacturing crystalline forms of rapamycin analogs
US11/781,807 2007-07-23

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KR20090035716A true KR20090035716A (ko) 2009-04-10

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KR1020097003955A Ceased KR20090035716A (ko) 2006-07-25 2007-07-24 라파마이신 유사체의 결정형 형태

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EP (2) EP2051984A1 (https=)
JP (1) JP2010500286A (https=)
KR (1) KR20090035716A (https=)
AU (1) AU2007276837B2 (https=)
BR (1) BRPI0714945B8 (https=)
CA (1) CA2658896A1 (https=)
IL (1) IL196706A0 (https=)
MX (1) MX2009001067A (https=)
NZ (1) NZ574654A (https=)
WO (1) WO2008014222A1 (https=)

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US7820812B2 (en) 2006-07-25 2010-10-26 Abbott Laboratories Methods of manufacturing crystalline forms of rapamycin analogs
US7812032B2 (en) 2006-07-25 2010-10-12 Abbott Laboratories Crystalline forms of rapamycin analogs
CA2673991C (en) 2007-01-21 2012-02-07 Hemoteq Ag Methods for coating catheter balloons with a defined quantity of active agent
US9192697B2 (en) 2007-07-03 2015-11-24 Hemoteq Ag Balloon catheter for treating stenosis of body passages and for preventing threatening restenosis
EP2380006A4 (en) * 2009-01-21 2012-05-16 Biocon Ltd PROCESS FOR DETERMINING THE SIROLIMUS STABILITY AND METHOD FOR PRODUCING ITS STABLE FORM
ES2550634T3 (es) 2009-07-10 2015-11-11 Boston Scientific Scimed, Inc. Uso de nanocristales para un balón de suministro de fármaco
EP2453938B1 (en) 2009-07-17 2015-08-19 Boston Scientific Scimed, Inc. Nucleation of drug delivery balloons to provide improved crystal size and density
US8889211B2 (en) 2010-09-02 2014-11-18 Boston Scientific Scimed, Inc. Coating process for drug delivery balloons using heat-induced rewrap memory
WO2013022458A1 (en) * 2011-08-05 2013-02-14 Boston Scientific Scimed, Inc. Methods of converting amorphous drug substance into crystalline form
WO2013028208A1 (en) 2011-08-25 2013-02-28 Boston Scientific Scimed, Inc. Medical device with crystalline drug coating
US9439892B2 (en) 2013-05-16 2016-09-13 Surmodics, Inc. Macrolide particulates, methods for preparation, and medical devices associated therewith
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