JP2010500286A - 結晶形態のラパマイシン類似体 - Google Patents

結晶形態のラパマイシン類似体 Download PDF

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JP2010500286A
JP2010500286A JP2009521936A JP2009521936A JP2010500286A JP 2010500286 A JP2010500286 A JP 2010500286A JP 2009521936 A JP2009521936 A JP 2009521936A JP 2009521936 A JP2009521936 A JP 2009521936A JP 2010500286 A JP2010500286 A JP 2010500286A
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Prior art keywords
powder
ray diffraction
diffraction pattern
rapamycin analog
composition
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JP2009521936A
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JP2010500286A5 (https=
Inventor
シェカー ヴィズワナス，
ラリー バートエルト，
ロバート レアンナ，
マイケル ラスムッセン，
マドハップ ダオン，
ロジャー ヘンリー，
トーマス ボーチャード，
シャング チェン，
ジェフ ツァン，
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Abbott Laboratories
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Abbott Laboratories
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Priority claimed from US11/781,804 external-priority patent/US7812032B2/en
Priority claimed from US11/781,807 external-priority patent/US7820812B2/en
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of JP2010500286A publication Critical patent/JP2010500286A/ja
Publication of JP2010500286A5 publication Critical patent/JP2010500286A5/ja
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    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
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JP2009521936A 2006-07-25 2007-07-24 結晶形態のラパマイシン類似体 Pending JP2010500286A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US82031706P 2006-07-25 2006-07-25
US11/781,804 US7812032B2 (en) 2006-07-25 2007-07-23 Crystalline forms of rapamycin analogs
US11/781,807 US7820812B2 (en) 2006-07-25 2007-07-23 Methods of manufacturing crystalline forms of rapamycin analogs
PCT/US2007/074159 WO2008014222A1 (en) 2006-07-25 2007-07-24 Crystalline forms of rapamycin analogs

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JP2010500286A true JP2010500286A (ja) 2010-01-07
JP2010500286A5 JP2010500286A5 (https=) 2010-09-09

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JP2009521936A Pending JP2010500286A (ja) 2006-07-25 2007-07-24 結晶形態のラパマイシン類似体

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EP (2) EP2051984A1 (https=)
JP (1) JP2010500286A (https=)
KR (1) KR20090035716A (https=)
AU (1) AU2007276837B2 (https=)
BR (1) BRPI0714945B8 (https=)
CA (1) CA2658896A1 (https=)
IL (1) IL196706A0 (https=)
MX (1) MX2009001067A (https=)
NZ (1) NZ574654A (https=)
WO (1) WO2008014222A1 (https=)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016521751A (ja) * 2013-06-12 2016-07-25 サーモディクス，インコーポレイティド 結晶性マクロライド微粒子を調製するための溶剤法、組成物、および微粒子を含む物品
JP2016530975A (ja) * 2013-09-18 2016-10-06 イノラ ゲーエムベーハ バルーンカテーテルに対する長時間作用型リムス製剤
JP2021506467A (ja) * 2017-12-22 2021-02-22 シャンハイ マイクロポート メディカル （グループ） シーオー．， エルティーディー． 装薬式埋め込み医療デバイスおよびその準備方法
JP2023519875A (ja) * 2020-03-27 2023-05-15 ボストン サイエンティフィック サイムド，インコーポレイテッド 薬品の結晶化のための方法
JP2024503898A (ja) * 2021-01-22 2024-01-29 ヤンセン ファーマシューティカ エヌ．ベー． ラパマイシン類似体及びその使用

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7820812B2 (en) 2006-07-25 2010-10-26 Abbott Laboratories Methods of manufacturing crystalline forms of rapamycin analogs
US7812032B2 (en) 2006-07-25 2010-10-12 Abbott Laboratories Crystalline forms of rapamycin analogs
CA2673991C (en) 2007-01-21 2012-02-07 Hemoteq Ag Methods for coating catheter balloons with a defined quantity of active agent
US9192697B2 (en) 2007-07-03 2015-11-24 Hemoteq Ag Balloon catheter for treating stenosis of body passages and for preventing threatening restenosis
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