NO981131L - Diarylalkenylamin-derivater - Google Patents
Diarylalkenylamin-derivaterInfo
- Publication number
- NO981131L NO981131L NO981131A NO981131A NO981131L NO 981131 L NO981131 L NO 981131L NO 981131 A NO981131 A NO 981131A NO 981131 A NO981131 A NO 981131A NO 981131 L NO981131 L NO 981131L
- Authority
- NO
- Norway
- Prior art keywords
- derivatives
- diarylalkenylamin
- analgesics
- potent
- antagonists
- Prior art date
Links
- 229940127450 Opioid Agonists Drugs 0.000 abstract 1
- 229940035676 analgesics Drugs 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 239000000730 antalgic agent Substances 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/28—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
- C07C237/30—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to hydrogen atoms or to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Transplantation (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT95MI001930A IT1277597B1 (it) | 1995-09-15 | 1995-09-15 | Derivati di diarilalchenilammina |
| PCT/EP1996/003988 WO1997010230A1 (en) | 1995-09-15 | 1996-09-09 | Diarylalkenylamine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO981131D0 NO981131D0 (no) | 1998-03-13 |
| NO981131L true NO981131L (no) | 1998-03-16 |
Family
ID=11372254
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO981131A NO981131L (no) | 1995-09-15 | 1998-03-13 | Diarylalkenylamin-derivater |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US6262104B1 (cs) |
| EP (1) | EP0873330B1 (cs) |
| JP (1) | JPH11512413A (cs) |
| KR (1) | KR19990044675A (cs) |
| CN (1) | CN1202164A (cs) |
| AR (1) | AR004205A1 (cs) |
| AT (1) | ATE240307T1 (cs) |
| AU (1) | AU706980B2 (cs) |
| BR (1) | BR9610597A (cs) |
| CA (1) | CA2232161A1 (cs) |
| CZ (1) | CZ78598A3 (cs) |
| DE (1) | DE69628200T2 (cs) |
| ES (1) | ES2195010T3 (cs) |
| HU (1) | HUP9900374A3 (cs) |
| IL (1) | IL123621A0 (cs) |
| IT (1) | IT1277597B1 (cs) |
| NO (1) | NO981131L (cs) |
| NZ (1) | NZ318774A (cs) |
| PL (1) | PL325552A1 (cs) |
| TR (1) | TR199800478T1 (cs) |
| WO (1) | WO1997010230A1 (cs) |
| ZA (1) | ZA967741B (cs) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5985880A (en) | 1996-06-05 | 1999-11-16 | Delta Pharmaceuticals | Compositions and methods for reducing respiratory depression and attendant side effects of mu opioid compounds |
| US6103722A (en) * | 1997-07-23 | 2000-08-15 | The Medical College Of Wisconsin Research Foundation Inc. | Ischemic preconditioning |
| DE69831876T2 (de) * | 1997-12-24 | 2006-07-27 | Ortho-Mcneil Pharmaceutical, Inc. | (4)-[aryl(piperidin-4-yl) aminobenzamidderivate die an delta-opioid rezeptor binden |
| US6436959B1 (en) | 1998-12-23 | 2002-08-20 | Ortho-Mcneil Pharmaceutical, Inc. | 4-[aryl(piperidin-4-yl)]aminobenzamides |
| AU2001232319B2 (en) * | 2000-02-18 | 2005-01-13 | Meiji Seika Kaisha, Ltd. | Phenoxyalkylamine derivates useful as opioid delta receptor ligands |
| CA2404280A1 (en) | 2000-03-24 | 2002-09-23 | Meiji Seika Kaisha, Ltd. | Diphenylalkylamine derivatives useful as opioid .delta. receptor agonists |
| JP4667384B2 (ja) * | 2003-10-07 | 2011-04-13 | レノビス， インコーポレイテッド | イオンチャネルリガンドとしてのアミド誘導体および薬学的組成物、ならびにこれらを使用する方法 |
| WO2006023757A2 (en) * | 2004-08-19 | 2006-03-02 | University Of Virginia Patent Foundation | Novel tricyclic, bicyclic, monocyclic, and acyclic amines as potent sodium channel blocking agents |
| US20080045610A1 (en) * | 2004-09-23 | 2008-02-21 | Alexander Michalow | Methods for regulating neurotransmitter systems by inducing counteradaptations |
| US20060069086A1 (en) * | 2004-09-23 | 2006-03-30 | Alexander Michalow | Methods for regulating neurotransmitter systems by inducing counteradaptations |
| EA200701835A1 (ru) * | 2005-02-28 | 2008-02-28 | Реновис, Инк. | Амидные производные в качестве лигандов ионных каналов, их фармацевтические композиции и способы их применения |
| US7576099B2 (en) | 2005-02-28 | 2009-08-18 | Renovis, Inc. | Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0000322B1 (en) * | 1977-07-04 | 1982-05-05 | Astra Läkemedel Aktiebolag | Compounds having an anti-depressive or tranquilizing activity, pharmaceutical compositions containing them, and processes and intermediates for their preparation |
| SI8310221A8 (en) | 1982-02-04 | 1995-10-31 | Wellcome Found | Process for obtaining new pyridil compounds |
| US4514414A (en) * | 1982-10-25 | 1985-04-30 | Smithkline Beckman Corporation | N-Substituted pyrrolidineacetic acids and their esters |
| US4564685A (en) * | 1983-03-10 | 1986-01-14 | Findlay John W A | Diphenylmethane compounds |
| ES2061432T3 (es) * | 1985-10-09 | 1994-12-16 | Shell Int Research | Nuevas amidas de acido acrilico. |
| PT94402A (pt) | 1989-06-19 | 1991-03-20 | Wellcome Found | Processo para a preparacao de compostos azotados que contem sistemas de aneis ciclicos aromaticos e de composicoes farmaceuticas que os contem |
-
1995
- 1995-09-15 IT IT95MI001930A patent/IT1277597B1/it active IP Right Grant
-
1996
- 1996-09-09 WO PCT/EP1996/003988 patent/WO1997010230A1/en not_active Ceased
- 1996-09-09 BR BR9610597A patent/BR9610597A/pt unknown
- 1996-09-09 HU HU9900374A patent/HUP9900374A3/hu unknown
- 1996-09-09 NZ NZ318774A patent/NZ318774A/en unknown
- 1996-09-09 AU AU70847/96A patent/AU706980B2/en not_active Ceased
- 1996-09-09 CA CA002232161A patent/CA2232161A1/en not_active Abandoned
- 1996-09-09 PL PL96325552A patent/PL325552A1/xx unknown
- 1996-09-09 TR TR1998/00478T patent/TR199800478T1/xx unknown
- 1996-09-09 CN CN96198240A patent/CN1202164A/zh active Pending
- 1996-09-09 KR KR1019980701930A patent/KR19990044675A/ko not_active Withdrawn
- 1996-09-09 EP EP96931791A patent/EP0873330B1/en not_active Expired - Lifetime
- 1996-09-09 IL IL12362196A patent/IL123621A0/xx unknown
- 1996-09-09 US US09/029,892 patent/US6262104B1/en not_active Expired - Fee Related
- 1996-09-09 CZ CZ98785A patent/CZ78598A3/cs unknown
- 1996-09-09 ES ES96931791T patent/ES2195010T3/es not_active Expired - Lifetime
- 1996-09-09 AT AT96931791T patent/ATE240307T1/de not_active IP Right Cessation
- 1996-09-09 JP JP9511657A patent/JPH11512413A/ja not_active Withdrawn
- 1996-09-09 DE DE69628200T patent/DE69628200T2/de not_active Expired - Fee Related
- 1996-09-12 AR ARP960104332A patent/AR004205A1/es unknown
- 1996-09-13 ZA ZA9607741A patent/ZA967741B/xx unknown
-
1998
- 1998-03-13 NO NO981131A patent/NO981131L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| TR199800478T1 (xx) | 1998-06-22 |
| IL123621A0 (en) | 1998-10-30 |
| AU706980B2 (en) | 1999-07-01 |
| ATE240307T1 (de) | 2003-05-15 |
| KR19990044675A (ko) | 1999-06-25 |
| HUP9900374A2 (hu) | 1999-06-28 |
| WO1997010230A1 (en) | 1997-03-20 |
| ITMI951930A0 (it) | 1995-09-15 |
| AU7084796A (en) | 1997-04-01 |
| ITMI951930A1 (it) | 1997-03-15 |
| DE69628200D1 (de) | 2003-06-18 |
| JPH11512413A (ja) | 1999-10-26 |
| IT1277597B1 (it) | 1997-11-11 |
| AR004205A1 (es) | 1998-11-04 |
| ZA967741B (en) | 1998-03-13 |
| NZ318774A (en) | 1998-08-26 |
| HUP9900374A3 (en) | 1999-11-29 |
| EP0873330B1 (en) | 2003-05-14 |
| MX9802024A (es) | 1998-08-30 |
| ES2195010T3 (es) | 2003-12-01 |
| PL325552A1 (en) | 1998-08-03 |
| BR9610597A (pt) | 1999-07-06 |
| CZ78598A3 (cs) | 1998-08-12 |
| DE69628200T2 (de) | 2003-11-27 |
| NO981131D0 (no) | 1998-03-13 |
| CN1202164A (zh) | 1998-12-16 |
| CA2232161A1 (en) | 1997-03-20 |
| US6262104B1 (en) | 2001-07-17 |
| EP0873330A1 (en) | 1998-10-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PL335484A1 (en) | Derivatives of heteroarylhexamide, their production and application as selective inhibitors of mip-1a being assimilated by its ccr1 receptor | |
| NO991732L (no) | Nye heterocyklylmetylsubstituerte pyrazolderivater | |
| ATE192153T1 (de) | Amino-imidazo (4,5-c) chinoline | |
| YU49898A (sh) | Hemijska jedinjenja | |
| NO942618L (no) | Imidazolderivater og deres anvendelse som cytokin-inhibitorer | |
| MY133647A (en) | Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates | |
| NO964871L (no) | Nye agonistforbindelser | |
| MD1233C2 (ro) | Derivaţi de eritromicină, procedeu de preparare a lor şi compoziţie farmaceutică pe baza acestora | |
| TR200100623T2 (tr) | 5-Tia-w-ikameli fenil-prostaglandin türevleri, bunları üretme yöntemleri ve müessir madde olarak bunları ihtiva eden ilaçlar | |
| NO20000311L (no) | Nye forbindelser | |
| GB9914486D0 (en) | Medicaments | |
| DK0970095T3 (da) | Hidtil ukendte benzimidazolinhibitorer for fructose-1,6-bisphosphase | |
| NZ233735A (en) | Heterocyclic substituted aminophenol derivatives | |
| NO981131L (no) | Diarylalkenylamin-derivater | |
| MXPA03012013A (es) | Derivados de 1-oxa-2,8-diaza-spiro[4,5]dec-2-eno sustituidos como medicamento para el tratamiento de dolor. | |
| NO305657B1 (no) | 4-substituerte piperidinderivater og farmas°ytisk preparat derav | |
| NO20062239L (no) | Nye tetrahydrospiro[piperidin-2,7'-pyrrolo[3,2-b]pyridinderivater og nye indolderivater nyttige i behandlingen av 5-HT6 reseptorrelaterte forstyrrelser | |
| DK0944643T3 (da) | Oxyiminopregnancarbolactoner. | |
| BR0007589A (pt) | Inibidores da proliferação de células | |
| MX9801890A (es) | Nuevos compuestos antagonistas selectivos del receptor nk3 humano, procedimiento para su obtencion y composiciones farmaceuticas que los contienen. | |
| NO984740L (no) | Isatinderivater som acetylcholinesteraseinhibitorer og analgetiske midler | |
| YU49276B (sh) | Postupak za dobijanje olanzapina | |
| MX9700373A (es) | Derivados morfinoides de heterociclo condensado. | |
| GR1000156B (el) | ΜΕΘΟΔΟΣ ΠΑΡΑΣΚΕΥΗΣ ΝΕΩΝ ΠΑΡΑΓΩΓΩΝ ΤΡΙΚΥΚΛΙΚΩΝ ΑΜΙΝΩΝ ΤΗΣ ΤΕΤΡΑΥΔΡΟ-5,6,7,8ΝΑΦΘΟ[2,3b] ΔΙΥΔΡΟ-2,3 ΦΟΥΡΑΝΗΣ & ΤΗΣ ΤΕΤΡΑΥΔΡΟ-6,7,8,9 5Η-ΒΕΝΖΟΚΥΚΛΟΕΠΤΑ[2,3Β] ΔΙΥΔΡΟ-2,3 ΦΟΥΡΑΝΗΣ. | |
| NO990914L (no) | Amorfe benzotiofener, fremgangsmÕter for fremstilling og fremgangsmÕter for anvendelse |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |