NO950731L - Optisk aktive karboksamidderivater - Google Patents

Optisk aktive karboksamidderivater

Info

Publication number
NO950731L
NO950731L NO950731A NO950731A NO950731L NO 950731 L NO950731 L NO 950731L NO 950731 A NO950731 A NO 950731A NO 950731 A NO950731 A NO 950731A NO 950731 L NO950731 L NO 950731L
Authority
NO
Norway
Prior art keywords
optically active
carboxamide derivatives
active carboxamide
rer
halogen atom
Prior art date
Application number
NO950731A
Other languages
English (en)
Other versions
NO950731D0 (no
Inventor
Atsusuke Terada
Yoshio Iizuka
Kazuyuki Wachi
Kenji Fujibayashi
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of NO950731D0 publication Critical patent/NO950731D0/no
Publication of NO950731L publication Critical patent/NO950731L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)

Abstract

Optisk aktive karboksamidderivater med den generelle formel:. (i formelen ovenfor er Ret hydrogen-eller halogenatom; Rer et halogenatom; Rer en pyrrolidino- eller piperidinogruppe; Y er en metylen-eller karbonylgruppe; og n er et helt tall 1 eller 2) og farmakologisk aksep-table salter derav.Forbindelsene ifølge foreliggende oppfinnelse har en utmerket analgetisk aktivitet og kan anvendes som et analgetisk middel.
NO950731A 1992-08-28 1995-02-27 Optisk aktive karboksamidderivater NO950731L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP22997092 1992-08-28
PCT/JP1993/001210 WO1994005646A1 (en) 1992-08-28 1993-08-27 Optically active carboxamide derivative

Publications (2)

Publication Number Publication Date
NO950731D0 NO950731D0 (no) 1995-02-27
NO950731L true NO950731L (no) 1995-04-21

Family

ID=16900566

Family Applications (1)

Application Number Title Priority Date Filing Date
NO950731A NO950731L (no) 1992-08-28 1995-02-27 Optisk aktive karboksamidderivater

Country Status (13)

Country Link
US (1) US5679674A (no)
EP (1) EP0657443A4 (no)
JP (1) JPH06122677A (no)
KR (1) KR950702972A (no)
AU (2) AU4981693A (no)
CA (1) CA2143449A1 (no)
CZ (1) CZ280931B6 (no)
FI (1) FI950878A (no)
HU (1) HUT72636A (no)
NO (1) NO950731L (no)
NZ (1) NZ255572A (no)
RU (1) RU2101284C1 (no)
WO (1) WO1994005646A1 (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE291429T1 (de) * 1996-11-25 2005-04-15 Toray Industries Mittel gegen juckreiz
US6191126B1 (en) * 1996-12-16 2001-02-20 Alcon Laboratories, Inc. Topical use of κ opioid agonists to treat ocular pain
US6174878B1 (en) 1999-08-31 2001-01-16 Alcon Laboratories, Inc. Topical use of kappa opioid agonists to treat otic pain
US6645990B2 (en) * 2000-08-15 2003-11-11 Amgen Inc. Thiazolyl urea compounds and methods of uses
ES2319265T3 (es) * 2001-03-30 2009-05-06 Toray Industries, Inc. Farmacos para el sindrome de piernas inquietas.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5021413B1 (en) * 1988-08-24 1994-12-13 Sankyo Co Analgesic thiomorpholins, their preparation, and pharmaceutical compositions containing them
JPH0735373B2 (ja) * 1989-08-11 1995-04-19 三共株式会社 カルボン酸アミド化合物

Also Published As

Publication number Publication date
EP0657443A1 (en) 1995-06-14
EP0657443A4 (en) 1995-09-06
KR950702972A (ko) 1995-08-23
FI950878A0 (fi) 1995-02-27
NO950731D0 (no) 1995-02-27
JPH06122677A (ja) 1994-05-06
CZ52595A3 (en) 1995-10-18
NZ255572A (en) 1996-10-28
AU4981693A (en) 1994-03-29
RU2101284C1 (ru) 1998-01-10
FI950878A (fi) 1995-03-29
RU95106652A (ru) 1996-12-10
CA2143449A1 (en) 1994-03-17
WO1994005646A1 (en) 1994-03-17
US5679674A (en) 1997-10-21
CZ280931B6 (cs) 1996-05-15
HUT72636A (en) 1996-05-28
AU4001797A (en) 1998-01-15
HU9500598D0 (en) 1995-04-28

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application